[go: up one dir, main page]

UA88448C2 - Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof - Google Patents

Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof

Info

Publication number
UA88448C2
UA88448C2 UAA200600912A UAA200600912A UA88448C2 UA 88448 C2 UA88448 C2 UA 88448C2 UA A200600912 A UAA200600912 A UA A200600912A UA A200600912 A UAA200600912 A UA A200600912A UA 88448 C2 UA88448 C2 UA 88448C2
Authority
UA
Ukraine
Prior art keywords
derivatives
group substituted
cyclopropyl group
substituted oxazolidinone
species
Prior art date
Application number
UAA200600912A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Ясумити Фукуда
Original Assignee
Мерк Энд Ко., Инк.
Керин Фармасьютикал Ко., Лтд.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Мерк Энд Ко., Инк., Керин Фармасьютикал Ко., Лтд. filed Critical Мерк Энд Ко., Инк.
Publication of UA88448C2 publication Critical patent/UA88448C2/en

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

This invention relates to new oxazolidinones having a cyclopropyl moiety, which are effective against aerobic and anerobic pathogens such as multi-resistant staphylococci, streptococci and enterococci, Bacteroides spp., Clostridia spp. species, as well as acid-fast organisms such as Mycobacterium tuberculosis and other mycobactenial species. The compounds are represented by structural formula: (I): its enantiomer, diastereomer, or phaimaceutically acceptable salt or ester thereof.
UAA200600912A 2003-07-02 2004-06-29 Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof UA88448C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US48390403P 2003-07-02 2003-07-02

Publications (1)

Publication Number Publication Date
UA88448C2 true UA88448C2 (en) 2009-10-26

Family

ID=36908184

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200600912A UA88448C2 (en) 2003-07-02 2004-06-29 Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof

Country Status (3)

Country Link
CN (2) CN1816545A (en)
UA (1) UA88448C2 (en)
ZA (1) ZA200510432B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12435077B2 (en) 2020-03-20 2025-10-07 Merck Sharp & Dohme Llc Oxazolidinone compound and methods of use thereof as an antibacterial agent

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013182070A1 (en) * 2012-06-08 2013-12-12 四川贝力克生物技术有限责任公司 Drug for preventing or treating mycobacterial diseases

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6689779B2 (en) * 2000-06-05 2004-02-10 Dong A Pharm. Co., Ltd. Oxazolidinone derivatives and a process for the preparation thereof
DE60206154T2 (en) * 2001-04-17 2006-06-29 Merck & Co., Inc. BICYCLO [3,1,0] HEXANE AS A STRUCTURAL ELEMENT CONTAINING OXAZOLIDINONE ANTIBIOTICS AND THEIR DERIVATIVES
CA2463794A1 (en) * 2001-11-29 2003-06-12 Merck & Co., Inc. Cyclopropyl hexane containing oxazolidinone antibiotics and derivatives thereof

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12435077B2 (en) 2020-03-20 2025-10-07 Merck Sharp & Dohme Llc Oxazolidinone compound and methods of use thereof as an antibacterial agent

Also Published As

Publication number Publication date
CN1816545A (en) 2006-08-09
CN1816548A (en) 2006-08-09
ZA200510432B (en) 2007-03-28
CN1816548B (en) 2011-01-12

Similar Documents

Publication Publication Date Title
MY140137A (en) Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof
ATE304536T1 (en) OXAZOLIDINONE ANTIBIOTICS CONTAINING BICYCLO(3,1,0)HEXANE AS A STRUCTURAL ELEMENT AND THEIR DERIVATIVES
MX9703543A (en) Bicyclic oxazine and thiazine oxazolidinone antibacterials.
MY132698A (en) Herbicidal composition
NO971946L (en) Phenyloxazolidinone antimicrobial agents
HUS1500046I1 (en) Novel oxazolidinone derivatives
MXPA05009205A (en) Hydroxymethyl substituted dihydroisoxazole derivatives useful as antibiotic agents.
LV12605A (en) Substituted oxazine and thiazine oxazlidinone antimicrobials
AU6964096A (en) Aminoaryl oxazolidinone n-oxides
MY161872A (en) Pyrrolidinyl derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors
EP1409464A4 (en) Oxazolidinone derivatives as potential antimicrobials
AU7665196A (en) Oxazolidinone antibacterial agent with tricyclic substituents
EA200500283A1 (en) OXIAZOLIDINON DERIVATIVES AS ANTI-MICROSAL AGENTS
WO2010058423A3 (en) Novel antimicrobials
UA88448C2 (en) Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof
MX9703040A (en) Phenyloxazolidinone antimicrobials.
TW200600011A (en) Silylated carboxamides
WO2006018682A3 (en) Oxazolidinone derivatives as antimicrobials
DOP2004000942A (en) ANTIBIOTICS OF OXAZOLIDINONA REPLACED WITH A CYCLOPROPILE GROUP AND DERIVATIVES OF THE SAME (CYCLOPROPYL GROUP SUBSTITUED OXAZOLDINONE ANTIBIOTICS AND DERIVATIVES THEREOF)
WO2009116090A3 (en) Novel antimicrobials