UA84594C2 - 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists - Google Patents
1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonistsInfo
- Publication number
- UA84594C2 UA84594C2 UAA200609435A UAA200609435A UA84594C2 UA 84594 C2 UA84594 C2 UA 84594C2 UA A200609435 A UAA200609435 A UA A200609435A UA A200609435 A UAA200609435 A UA A200609435A UA 84594 C2 UA84594 C2 UA 84594C2
- Authority
- UA
- Ukraine
- Prior art keywords
- pyrazole derivatives
- trisubstituted
- dihydro
- antagonists
- compounds
- Prior art date
Links
- -1 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole Chemical class 0.000 title abstract 2
- 229940124802 CB1 antagonist Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000009286 beneficial effect Effects 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 238000002360 preparation method Methods 0.000 abstract 1
- 150000003217 pyrazoles Chemical class 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The present invention relates to 1,3,5-trisubstituted 4,5-dihydro-1H-pyrazole derivatives as CBantagonists, to methods for the preparation of these compounds and to novel intermediates useful for the synthesis of said pyrazole derivatives. The invention also relates to the use of a compound disclosed herein for the manufacture of a medicament giving a beneficial effect. The compounds have the general formula (I) wherein the symbols have the meanings given in the specification.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UAA200609435A UA84594C2 (en) | 2005-01-27 | 2005-01-27 | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| UAA200609435A UA84594C2 (en) | 2005-01-27 | 2005-01-27 | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA84594C2 true UA84594C2 (en) | 2008-11-10 |
Family
ID=50180792
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200609435A UA84594C2 (en) | 2005-01-27 | 2005-01-27 | 1,3,5-trisubstituted 4,5-dihydro-1h-pyrazole derivatives as cb1 antagonists |
Country Status (1)
| Country | Link |
|---|---|
| UA (1) | UA84594C2 (en) |
-
2005
- 2005-01-27 UA UAA200609435A patent/UA84594C2/en unknown
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