UA80474C2 - Aminoheteroaryl compounds as inhibitors of protein kinase - Google Patents
Aminoheteroaryl compounds as inhibitors of protein kinaseInfo
- Publication number
- UA80474C2 UA80474C2 UAA200509044A UA2005009044A UA80474C2 UA 80474 C2 UA80474 C2 UA 80474C2 UA A200509044 A UAA200509044 A UA A200509044A UA 2005009044 A UA2005009044 A UA 2005009044A UA 80474 C2 UA80474 C2 UA 80474C2
- Authority
- UA
- Ukraine
- Prior art keywords
- inhibitors
- protein kinase
- compounds
- aminoheteroaryl compounds
- aminoheteroaryl
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 102000001253 Protein Kinase Human genes 0.000 title 1
- 125000005214 aminoheteroaryl group Chemical group 0.000 title 1
- 108060006633 protein kinase Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003927 aminopyridines Chemical class 0.000 abstract 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000003909 protein kinase inhibitor Substances 0.000 abstract 1
- XFTQRUTUGRCSGO-UHFFFAOYSA-N pyrazin-2-amine Chemical class NC1=CN=CC=N1 XFTQRUTUGRCSGO-UHFFFAOYSA-N 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Aminopyridine and aminopyrazine compounds of formula (1), compositions including these compounds, and methods of their use are provided. Preferred compounds of formula 1 have activity as protein kinase inhibitors, including as inhibitors of c-MET.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US44958803P | 2003-02-26 | 2003-02-26 | |
| PCT/US2004/005495 WO2004076412A2 (en) | 2003-02-26 | 2004-02-26 | Aminoheteroaryl compounds as protein kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA80474C2 true UA80474C2 (en) | 2007-09-25 |
Family
ID=36766604
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UAA200509044A UA80474C2 (en) | 2003-02-26 | 2004-02-26 | Aminoheteroaryl compounds as inhibitors of protein kinase |
Country Status (5)
| Country | Link |
|---|---|
| CN (1) | CN1777427A (en) |
| CR (1) | CR7961A (en) |
| SI (2) | SI2476667T1 (en) |
| UA (1) | UA80474C2 (en) |
| ZA (1) | ZA200506460B (en) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4242911B2 (en) * | 2004-08-26 | 2009-03-25 | ファイザー・インク | Enantiopure aminoheteroaryl compounds as protein kinase inhibitors |
| US7790885B2 (en) * | 2006-08-31 | 2010-09-07 | Eisai R&D Management Co., Ltd. | Process for preparing phenoxypyridine derivatives |
| CN103204844A (en) * | 2012-01-17 | 2013-07-17 | 上海艾力斯医药科技有限公司 | Amino heteroaryl compound, and preparation method and application thereof |
| GB201211310D0 (en) * | 2012-06-26 | 2012-08-08 | Chroma Therapeutics Ltd | CSF-1R kinase inhibitors |
| CN104650049B (en) * | 2013-08-28 | 2018-06-08 | 广东东阳光药业有限公司 | Substituted pyridine compounds and its application method and purposes |
| CN105330697B (en) * | 2014-08-07 | 2019-05-28 | 江苏豪森药业集团有限公司 | A kind of crystal form of anticancer compound and its preparation method and application |
| WO2016019910A1 (en) * | 2014-08-07 | 2016-02-11 | 江苏豪森药业股份有限公司 | Crystal form of anticancer compound and preparation method and use thereof |
| KR102559499B1 (en) * | 2015-01-09 | 2023-07-25 | 오노 야꾸힝 고교 가부시키가이샤 | Tricyclic spiro compound |
| ES2920702T3 (en) * | 2018-03-15 | 2022-08-08 | Fujian Haixi Pharmaceuticals Co Ltd | Heteroaryl Compounds as Kinase Inhibitors |
| CN108947895B (en) * | 2018-08-22 | 2021-09-24 | 肇庆中彩机电技术研发有限公司 | Compound with anticancer activity |
| KR102426921B1 (en) * | 2019-09-24 | 2022-07-29 | 주식회사 이노보테라퓨틱스 | Heteroarylamidopyridinol derivatives and pharmaceutical composition for use in preventing or treating autoimmune diseases containing the same as an active ingredient |
| CN110921918B (en) * | 2019-12-18 | 2021-12-31 | 山东理工大学 | Method for treating amino aromatic sulfonic acid wastewater |
| CN114437058A (en) * | 2020-10-30 | 2022-05-06 | 珠海宇繁生物科技有限责任公司 | Deuterated HPK1 kinase inhibitor and preparation method and application thereof |
-
2004
- 2004-02-26 CN CN 200480010633 patent/CN1777427A/en active Pending
- 2004-02-26 SI SI200432180T patent/SI2476667T1/en unknown
- 2004-02-26 SI SI200431995T patent/SI1603570T1/en unknown
- 2004-02-26 UA UAA200509044A patent/UA80474C2/en unknown
-
2005
- 2005-08-12 ZA ZA200506460A patent/ZA200506460B/en unknown
- 2005-08-24 CR CR7961A patent/CR7961A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1777427A (en) | 2006-05-24 |
| CR7961A (en) | 2006-08-09 |
| SI1603570T1 (en) | 2013-03-29 |
| SI2476667T1 (en) | 2014-10-30 |
| ZA200506460B (en) | 2006-08-30 |
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