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UA103031C2 - 1,3-thiazolidine-2,4-dione derivatives and pharmaceutical composition comprising thereof - Google Patents

1,3-thiazolidine-2,4-dione derivatives and pharmaceutical composition comprising thereof

Info

Publication number
UA103031C2
UA103031C2 UAA201100972A UAA201100972A UA103031C2 UA 103031 C2 UA103031 C2 UA 103031C2 UA A201100972 A UAA201100972 A UA A201100972A UA A201100972 A UAA201100972 A UA A201100972A UA 103031 C2 UA103031 C2 UA 103031C2
Authority
UA
Ukraine
Prior art keywords
pim
thiazolidine
pharmaceutical composition
relates
dione derivatives
Prior art date
Application number
UAA201100972A
Other languages
Russian (ru)
Ukrainian (uk)
Inventor
Леслі Дакін
Джеймс Едвард Даулінг
Мішелл Лемб
Джон Рід
Цібінь Су
СяоЛань Чжен
Original Assignee
Астразенека Аб
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Астразенека Аб filed Critical Астразенека Аб
Priority claimed from PCT/GB2009/050773 external-priority patent/WO2010001169A2/en
Publication of UA103031C2 publication Critical patent/UA103031C2/en

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Abstract

The invention relates to chemical compounds of formula (I), and sails thereof. In some embodiments, the invention relates to inhibitors or modulators of PIM-1 and/or PIM-2, and/or PIM-3 protein kinase activity or enzyme function. In still further embodiments, the invention relates to pharmaceutical compositions comprising compounds disclosed herein, and their use in the prevention and treatment of PIM kinase related conditions and diseases, preferably cancer.
UAA201100972A 2008-07-02 2009-07-02 1,3-thiazolidine-2,4-dione derivatives and pharmaceutical composition comprising thereof UA103031C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7763908P 2008-07-02 2008-07-02
PCT/GB2009/050773 WO2010001169A2 (en) 2008-07-02 2009-07-02 Chemical compounds 251

Publications (1)

Publication Number Publication Date
UA103031C2 true UA103031C2 (en) 2013-09-10

Family

ID=52275587

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201100972A UA103031C2 (en) 2008-07-02 2009-07-02 1,3-thiazolidine-2,4-dione derivatives and pharmaceutical composition comprising thereof

Country Status (1)

Country Link
UA (1) UA103031C2 (en)

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