TW200635600A - Tetracyclic bicyclolides - Google Patents
Tetracyclic bicyclolidesInfo
- Publication number
- TW200635600A TW200635600A TW094144052A TW94144052A TW200635600A TW 200635600 A TW200635600 A TW 200635600A TW 094144052 A TW094144052 A TW 094144052A TW 94144052 A TW94144052 A TW 94144052A TW 200635600 A TW200635600 A TW 200635600A
- Authority
- TW
- Taiwan
- Prior art keywords
- present
- compounds
- subject
- bicyclolides
- tetracyclic
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 4
- 238000000034 method Methods 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 208000035143 Bacterial infection Diseases 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63565004P | 2004-12-13 | 2004-12-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW200635600A true TW200635600A (en) | 2006-10-16 |
Family
ID=36588440
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW094144052A TW200635600A (en) | 2004-12-13 | 2005-12-13 | Tetracyclic bicyclolides |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US7312201B2 (zh) |
| TW (1) | TW200635600A (zh) |
| WO (1) | WO2006065743A2 (zh) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL1836211T3 (pl) | 2004-12-21 | 2010-07-30 | Pfizer Prod Inc | Makrolidy |
| US7517859B2 (en) * | 2005-05-04 | 2009-04-14 | Enanta Pharmaceuticals, Inc. | Spirocyclic bicyclolides |
| DK1934238T3 (en) | 2005-08-24 | 2017-09-18 | Melinta Therapeutics Inc | TRIAZOL COMPOUNDS AND METHODS FOR THE PREPARATION AND USE OF THESE |
| US7407942B2 (en) * | 2006-03-29 | 2008-08-05 | Emata Pharmaceuticals, Inc | 3,6-bridged 9,12-oxolides |
| AU2007256844A1 (en) * | 2006-06-05 | 2007-12-13 | Auspex Pharmaceuticals, Inc. | Preparation and utility of substituted erythromycin analogs |
| WO2009064953A1 (en) * | 2007-11-15 | 2009-05-22 | Enanta Pharmaceuticals, Inc. | Use of bridged macrolides or tylosin derivatives in treating inflammatory bowel diseases |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2096969C (en) | 1990-11-28 | 2000-11-21 | Masato Kashimura | 6-0-methylerythromycin a derivatives |
| KR0166996B1 (ko) | 1992-04-22 | 1999-01-15 | 우에하라 아키라 | 5-o-데소사미닐에리쓰로노라이드a 유도체 |
| FR2738571B1 (fr) | 1995-09-11 | 1997-10-17 | Roussel Uclaf | Nouveaux derives de la 5-0-desosaminyl 6-0-methyl- erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs |
| US6274715B1 (en) * | 1995-11-08 | 2001-08-14 | Abbott Laboratories | Tricyclic erythromycin derivatives |
| ES2242983T3 (es) * | 1996-09-04 | 2005-11-16 | Abbott Laboratories | Cetolidos 6-0-sustituidos que tienen una actividad antibacteriana. |
| UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
| US6054435A (en) * | 1999-03-19 | 2000-04-25 | Abbott Laboratories | 6-O-substituted macrolides having antibacterial activity |
| US6355620B1 (en) * | 1999-05-14 | 2002-03-12 | Abbott Laboratories | C-2 modified erythromycin derivatives |
| US6437106B1 (en) | 1999-06-24 | 2002-08-20 | Abbott Laboratories | Process for preparing 6-o-substituted erythromycin derivatives |
| CA2483678C (en) | 2002-05-13 | 2010-01-12 | Enanta Pharmaceuticals, Inc. | 6-11 bicyclic ketolide derivatives |
| WO2003095466A1 (en) | 2002-05-13 | 2003-11-20 | Enanta Pharmaceuticals, Inc. | 6,11 bicyclic erythromycin derivatives |
| US7402568B2 (en) * | 2004-09-29 | 2008-07-22 | Enanta Pharmaceuticals, Inc. | Bicyclic 9a-azalide derivatives |
-
2005
- 2005-12-13 TW TW094144052A patent/TW200635600A/zh unknown
- 2005-12-13 US US11/302,525 patent/US7312201B2/en not_active Expired - Fee Related
- 2005-12-13 WO PCT/US2005/044919 patent/WO2006065743A2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| US20060142215A1 (en) | 2006-06-29 |
| US7312201B2 (en) | 2007-12-25 |
| WO2006065743A2 (en) | 2006-06-22 |
| WO2006065743A3 (en) | 2006-09-08 |
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