TW200519099A - Novel amines as histamine-3 receptor ligands and their therapeutic applications - Google Patents
Novel amines as histamine-3 receptor ligands and their therapeutic applicationsInfo
- Publication number
- TW200519099A TW200519099A TW093141278A TW93141278A TW200519099A TW 200519099 A TW200519099 A TW 200519099A TW 093141278 A TW093141278 A TW 093141278A TW 93141278 A TW93141278 A TW 93141278A TW 200519099 A TW200519099 A TW 200519099A
- Authority
- TW
- Taiwan
- Prior art keywords
- histamine
- receptor ligands
- therapeutic applications
- novel amines
- amines
- Prior art date
Links
- 239000003446 ligand Substances 0.000 title abstract 2
- 150000001412 amines Chemical class 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 230000001668 ameliorated effect Effects 0.000 abstract 1
- 150000001408 amides Chemical class 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 150000002148 esters Chemical class 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Compounds of formula (I), or a pharmaceutically -acceptable salt, ester, amide, or prodrug thereof, which are useful for the modulation of the histamine-3 receptors in mammals and which are useful for the treatment of disorders ameliorated by histamine-3 receptor ligands.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/810,648 US20020177589A1 (en) | 2001-03-16 | 2001-03-16 | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
| US10/044,495 US20020183309A1 (en) | 2001-03-16 | 2002-01-11 | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
| US10/081,207 US6969730B2 (en) | 2001-03-16 | 2002-02-25 | Amines as histamine-3 receptor ligands and their therapeutic applications |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TW200519099A true TW200519099A (en) | 2005-06-16 |
| TWI333489B TWI333489B (en) | 2010-11-21 |
Family
ID=38812605
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW91104939A TWI335914B (en) | 2001-03-16 | 2002-03-15 | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
| TW93141278A TWI333489B (en) | 2001-03-16 | 2002-03-15 | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW91104939A TWI335914B (en) | 2001-03-16 | 2002-03-15 | Novel amines as histamine-3 receptor ligands and their therapeutic applications |
Country Status (3)
| Country | Link |
|---|---|
| PE (1) | PE20020928A1 (en) |
| TW (2) | TWI335914B (en) |
| UY (1) | UY27212A1 (en) |
-
2002
- 2002-03-15 TW TW91104939A patent/TWI335914B/en not_active IP Right Cessation
- 2002-03-15 TW TW93141278A patent/TWI333489B/en not_active IP Right Cessation
- 2002-03-15 PE PE2002000203A patent/PE20020928A1/en not_active Application Discontinuation
- 2002-03-15 UY UY27212A patent/UY27212A1/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| PE20020928A1 (en) | 2002-10-26 |
| TWI333489B (en) | 2010-11-21 |
| TWI335914B (en) | 2011-01-11 |
| UY27212A1 (en) | 2002-10-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Annulment or lapse of patent due to non-payment of fees |