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TR200002749T2 - Antibiyotikler olarak siklik aminoguanidin substitüentlerine sahip sefalosporinler. - Google Patents

Antibiyotikler olarak siklik aminoguanidin substitüentlerine sahip sefalosporinler.

Info

Publication number
TR200002749T2
TR200002749T2 TR2000/02749T TR200002749T TR200002749T2 TR 200002749 T2 TR200002749 T2 TR 200002749T2 TR 2000/02749 T TR2000/02749 T TR 2000/02749T TR 200002749 T TR200002749 T TR 200002749T TR 200002749 T2 TR200002749 T2 TR 200002749T2
Authority
TR
Turkey
Prior art keywords
substituents
cephalosporins
antibiotics
cyclic
cyclic aminoguanidine
Prior art date
Application number
TR2000/02749T
Other languages
English (en)
Inventor
Ascher Gerd
Heilmayer Werner
Ludescher Johannes
Hildebrandt Johannes
Schranz M�Chael
Wieser Josef
Original Assignee
Biochemie Gesellschaft M.B.H.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biochemie Gesellschaft M.B.H. filed Critical Biochemie Gesellschaft M.B.H.
Publication of TR200002749T2 publication Critical patent/TR200002749T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
    • C07D501/46—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Farmasötik olarak yararli olan asagidaki formüle sahip bir bilesik olup içersindeki R2, baglandigi nitrojen atomuyla birlikte bir siklik aminoguanidin grubu veya onun türevini olusturmaktadir ve diger substituentler tarifname içersinde belirtilmis olan degisik anlamlara gelmektedir.(Formül).
TR2000/02749T 1998-03-23 1999-03-19 Antibiyotikler olarak siklik aminoguanidin substitüentlerine sahip sefalosporinler. TR200002749T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
AT0051598A AT406772B (de) 1998-03-23 1998-03-23 Antibakterielle 7-acylamino-3-iminomethyl- cephalosporine und verfahren zu deren herstellung

Publications (1)

Publication Number Publication Date
TR200002749T2 true TR200002749T2 (tr) 2000-12-21

Family

ID=3492649

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/02749T TR200002749T2 (tr) 1998-03-23 1999-03-19 Antibiyotikler olarak siklik aminoguanidin substitüentlerine sahip sefalosporinler.

Country Status (25)

Country Link
US (1) US6440957B1 (tr)
EP (2) EP1930335A1 (tr)
JP (1) JP2002507616A (tr)
KR (1) KR100696422B1 (tr)
CN (1) CN1188418C (tr)
AR (1) AR015248A1 (tr)
AT (1) AT406772B (tr)
AU (1) AU749735B2 (tr)
BR (1) BR9908960A (tr)
CA (1) CA2324953C (tr)
CO (1) CO5080739A1 (tr)
HU (1) HUP0101603A3 (tr)
ID (1) ID26567A (tr)
IL (2) IL138477A0 (tr)
MY (1) MY119841A (tr)
NO (1) NO20004760L (tr)
NZ (1) NZ506908A (tr)
PE (1) PE20000360A1 (tr)
PL (1) PL343094A1 (tr)
RU (1) RU2245884C2 (tr)
SK (1) SK14152000A3 (tr)
TR (1) TR200002749T2 (tr)
TW (1) TWI250983B (tr)
WO (1) WO1999048896A1 (tr)
ZA (1) ZA200004850B (tr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6693095B2 (en) * 1997-04-01 2004-02-17 Biochemie Gesellschaft M.B.H. Antibacterial substituted 7-acylamino-3-(methylhydrazono) methyl-cephalosporins and intermediates
DE102007052891A1 (de) 2007-11-02 2009-05-07 Evonik Degussa Gmbh Verfahren zur Stabilisierung von olefinisch ungesättigten Monomeren
DE102013204950A1 (de) 2013-03-20 2014-09-25 Evonik Industries Ag Verfahren und Zusammensetzung zur Inhibierung der Polymerisation von Cyclopentadienverbindungen
ES2624415T3 (es) 2014-09-08 2017-07-14 Evonik Degussa Gmbh (Tio)acetales fenólicos como agentes inhibidores de la polimerización de monómeros olefínicamente insaturados
TWI669317B (zh) 2014-09-22 2019-08-21 德商贏創德固賽有限責任公司 反應性單體的改良製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE943408C (de) * 1953-03-31 1956-05-17 Bayer Ag Verfahren zur Darstellung von Bisguanylhydrazonen
FI851934A7 (fi) * 1984-05-30 1985-12-01 Ici Plc Kefalosporiinijohdannaisia.
GB8721568D0 (en) * 1987-09-14 1987-10-21 Fujisawa Pharmaceutical Co Cephem compounds
JPH11506429A (ja) * 1995-05-11 1999-06-08 ビオヘミー・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング 抗細菌セファロスポリン類
DK0973780T3 (da) * 1997-04-01 2003-10-27 Biochemie Gmbh Antibakterielle substituerede 7-acylamino-3-(methylhydrazono)-methylcephalosporiner og mellemprodukter

Also Published As

Publication number Publication date
AR015248A1 (es) 2001-04-18
TWI250983B (en) 2006-03-11
IL138477A0 (en) 2001-10-31
MY119841A (en) 2005-07-29
PL343094A1 (en) 2001-07-30
ATA51598A (de) 2000-01-15
NO20004760D0 (no) 2000-09-22
CN1294593A (zh) 2001-05-09
NO20004760L (no) 2000-11-21
IL138477A (en) 2007-06-17
CA2324953C (en) 2008-05-13
ID26567A (id) 2001-01-18
AT406772B (de) 2000-08-25
PE20000360A1 (es) 2000-05-17
NZ506908A (en) 2003-04-29
CO5080739A1 (es) 2001-09-25
US6440957B1 (en) 2002-08-27
BR9908960A (pt) 2000-12-05
HUP0101603A3 (en) 2002-10-28
ZA200004850B (en) 2002-02-27
HUP0101603A2 (hu) 2001-12-28
KR100696422B1 (ko) 2007-03-20
EP1082326A1 (en) 2001-03-14
SK14152000A3 (sk) 2001-05-10
KR20010074666A (ko) 2001-08-08
RU2245884C2 (ru) 2005-02-10
EP1930335A1 (en) 2008-06-11
WO1999048896A1 (en) 1999-09-30
CA2324953A1 (en) 1999-09-30
AU3518899A (en) 1999-10-18
JP2002507616A (ja) 2002-03-12
CN1188418C (zh) 2005-02-09
AU749735B2 (en) 2002-07-04

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