TN2013000494A1 - Combination of panobinostat and ruxolitinib in the treatment of cancer such as a myeloproliferative neoplasm - Google Patents
Combination of panobinostat and ruxolitinib in the treatment of cancer such as a myeloproliferative neoplasmInfo
- Publication number
- TN2013000494A1 TN2013000494A1 TNP2013000494A TN2013000494A TN2013000494A1 TN 2013000494 A1 TN2013000494 A1 TN 2013000494A1 TN P2013000494 A TNP2013000494 A TN P2013000494A TN 2013000494 A TN2013000494 A TN 2013000494A TN 2013000494 A1 TN2013000494 A1 TN 2013000494A1
- Authority
- TN
- Tunisia
- Prior art keywords
- combination
- treatment
- relates
- ruxolitinib
- panobinostat
- Prior art date
Links
- HFNKQEVNSGCOJV-OAHLLOKOSA-N ruxolitinib Chemical compound C1([C@@H](CC#N)N2N=CC(=C2)C=2C=3C=CNC=3N=CN=2)CCCC1 HFNKQEVNSGCOJV-OAHLLOKOSA-N 0.000 title abstract 2
- 239000002144 L01XE18 - Ruxolitinib Substances 0.000 title 1
- 201000007224 Myeloproliferative neoplasm Diseases 0.000 title 1
- 206010028980 Neoplasm Diseases 0.000 title 1
- 201000011510 cancer Diseases 0.000 title 1
- FWZRWHZDXBDTFK-ZHACJKMWSA-N panobinostat Chemical compound CC1=NC2=CC=C[CH]C2=C1CCNCC1=CC=C(\C=C\C(=O)NO)C=C1 FWZRWHZDXBDTFK-ZHACJKMWSA-N 0.000 title 1
- 229960005184 panobinostat Drugs 0.000 title 1
- 229960000215 ruxolitinib Drugs 0.000 title 1
- 201000010099 disease Diseases 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 230000002062 proliferating effect Effects 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 239000000126 substance Substances 0.000 abstract 2
- 229940126062 Compound A Drugs 0.000 abstract 1
- NLDMNSXOCDLTTB-UHFFFAOYSA-N Heterophylliin A Natural products O1C2COC(=O)C3=CC(O)=C(O)C(O)=C3C3=C(O)C(O)=C(O)C=C3C(=O)OC2C(OC(=O)C=2C=C(O)C(O)=C(O)C=2)C(O)C1OC(=O)C1=CC(O)=C(O)C(O)=C1 NLDMNSXOCDLTTB-UHFFFAOYSA-N 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- FPOHNWQLNRZRFC-ZHACJKMWSA-N panobinostat Chemical compound CC=1NC2=CC=CC=C2C=1CCNCC1=CC=C(\C=C\C(=O)NO)C=C1 FPOHNWQLNRZRFC-ZHACJKMWSA-N 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The invention relates to a combination which comprises: (a) Compound A ((R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile) of Formula (A): [Chemical formula should be inserted here as it appears in Abstract in paper form] or a pharmaceutically acceptable salt thereof; and (b) Compound B (N-hydroxy-3-[4-[[[2-(2-methyl-1H-indol-3-yl)-ethyl]-amino]methyl]phenyl]-2E-2-propenamide) of Formula (B): [Chemical formula should be inserted here as it appears in Abstract in paper form] or a pharmaceutically acceptable salt thereof; for simultaneous, concurrent, separate or sequential use, especially for use in the treatment of proliferative diseases. The invention also relates to pharmaceutical compositions comprising such a combination and to a method of treating proliferative diseases, in a mammal, particularly a human, with such a combination. The present invention further also relates to a commercial package or product comprising such a combination.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161568717P | 2011-12-09 | 2011-12-09 | |
| PCT/US2012/042174 WO2012174061A1 (en) | 2011-06-14 | 2012-06-13 | Combination of panobinostat and ruxolitinib in the treatment of cancer such as a myeloproliferative neoplasm |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TN2013000494A1 true TN2013000494A1 (en) | 2015-03-30 |
Family
ID=54359612
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TNP2013000494A TN2013000494A1 (en) | 2011-12-09 | 2013-11-25 | Combination of panobinostat and ruxolitinib in the treatment of cancer such as a myeloproliferative neoplasm |
Country Status (1)
| Country | Link |
|---|---|
| TN (1) | TN2013000494A1 (en) |
-
2013
- 2013-11-25 TN TNP2013000494A patent/TN2013000494A1/en unknown
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