TN2010000588A1 - Substituted isoquinolines and isoquinolinones - Google Patents
Substituted isoquinolines and isoquinolinonesInfo
- Publication number
- TN2010000588A1 TN2010000588A1 TNP2010000588A TN2010000588A TN2010000588A1 TN 2010000588 A1 TN2010000588 A1 TN 2010000588A1 TN P2010000588 A TNP2010000588 A TN P2010000588A TN 2010000588 A TN2010000588 A TN 2010000588A TN 2010000588 A1 TN2010000588 A1 TN 2010000588A1
- Authority
- TN
- Tunisia
- Prior art keywords
- isoquinolinones
- rho
- substituted isoquinolines
- kinase
- substituted
- Prior art date
Links
- VDBNYAPERZTOOF-UHFFFAOYSA-N isoquinolin-1(2H)-one Chemical class C1=CC=C2C(=O)NC=CC2=C1 VDBNYAPERZTOOF-UHFFFAOYSA-N 0.000 title abstract 2
- 150000002537 isoquinolines Chemical class 0.000 title 1
- 102000000568 rho-Associated Kinases Human genes 0.000 abstract 2
- 108010041788 rho-Associated Kinases Proteins 0.000 abstract 2
- -1 6-substituted isoquinoline Chemical class 0.000 abstract 1
- 102000011131 Myosin-Light-Chain Phosphatase Human genes 0.000 abstract 1
- 108010037801 Myosin-Light-Chain Phosphatase Proteins 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000006806 disease prevention Effects 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000026731 phosphorylation Effects 0.000 abstract 1
- 238000006366 phosphorylation reaction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
The invention relates to 6-substituted isoquinoline and isoquinolinone derivatives of the formula (I) useful for the treatment and/or prevention of diseases associated with Rho-kinase and/or Rho-kinase mediated phosphorylation of myosin light chain phosphatase, and compositions containing such compounds.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2009/004420 WO2009156099A1 (en) | 2008-06-24 | 2009-06-19 | 6-substituted isoquinolines and isoquinolinones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TN2010000588A1 true TN2010000588A1 (en) | 2012-05-24 |
Family
ID=55024663
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TNP2010000588A TN2010000588A1 (en) | 2009-06-19 | 2010-12-17 | Substituted isoquinolines and isoquinolinones |
Country Status (1)
| Country | Link |
|---|---|
| TN (1) | TN2010000588A1 (en) |
-
2010
- 2010-12-17 TN TNP2010000588A patent/TN2010000588A1/en unknown
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