[go: up one dir, main page]

TN2010000561A1 - Novel derivatives of (bridged piperazinyl) 1-alcanone and use thereof as p75 inhibitors - Google Patents

Novel derivatives of (bridged piperazinyl) 1-alcanone and use thereof as p75 inhibitors

Info

Publication number
TN2010000561A1
TN2010000561A1 TNP2010000561A TN2010000561A TN2010000561A1 TN 2010000561 A1 TN2010000561 A1 TN 2010000561A1 TN P2010000561 A TNP2010000561 A TN P2010000561A TN 2010000561 A TN2010000561 A TN 2010000561A TN 2010000561 A1 TN2010000561 A1 TN 2010000561A1
Authority
TN
Tunisia
Prior art keywords
alcanone
inhibitors
novel derivatives
bridged piperazinyl
piperazinyl
Prior art date
Application number
TNP2010000561A
Other languages
French (fr)
Inventor
Marco Baroni
Francoise Bono
Gossart Sandrine Delbary
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/FR2009/051118 external-priority patent/WO2009150388A1/en
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of TN2010000561A1 publication Critical patent/TN2010000561A1/en

Links

Landscapes

  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The invention relates to derivatives of ((phenyl)-3,6-dihydropyridin-1 yl)- (bridged piperazinyl)-1 -alkanone and ((phenyl)-2,5-dihydro-pyrrol-1 yl)-(bridged piperazinyl)-1 – alkanone derivatives of the general formula (I) where A, B, m, W, n, and R5 are such as defined in Claim 1, to a method for preparing the same, and to the therapeutic application thereof.
TNP2010000561A 2009-06-12 2010-12-03 Novel derivatives of (bridged piperazinyl) 1-alcanone and use thereof as p75 inhibitors TN2010000561A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/FR2009/051118 WO2009150388A1 (en) 2008-06-13 2009-06-12 Novel derivatives of (bridged piperazinyl)-1-alcanone and use thereof as p75 inhibitors

Publications (1)

Publication Number Publication Date
TN2010000561A1 true TN2010000561A1 (en) 2012-05-24

Family

ID=55024644

Family Applications (1)

Application Number Title Priority Date Filing Date
TNP2010000561A TN2010000561A1 (en) 2009-06-12 2010-12-03 Novel derivatives of (bridged piperazinyl) 1-alcanone and use thereof as p75 inhibitors

Country Status (1)

Country Link
TN (1) TN2010000561A1 (en)

Similar Documents

Publication Publication Date Title
IL204437A (en) Cyclopropyl aryl amide derivatives and uses thereof
EA018629B8 (en) Phenyl and benzodioxinyl substituted indazoles derivatives
UA109775C2 (en) N-containing heteroaryl derivatives as JAK3 kinase inhibitors
MX2009000884A (en) Pyridizinone derivatives.
TW200621777A (en) New dihydropteridione derivatives, process for their manufacture and their use as medicament
GEP20166432B (en) 3-pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant idh
MY169043A (en) New dihydroquinoline-2-one derivatives
MY186165A (en) New bicyclic dihydroquinoline-2-one derivatives
TW200621262A (en) New dihydropteridione derivatives, process for their manufacture and their use as medicament
TW201713640A (en) Bruton's tyrosine kinase inhibitors
MX2011011661A (en) Substituted 1-cyanoethylheterocyclylcarboxamide compounds 750.
PH12012500752A1 (en) Benzimidazole-imidazole derivatives
MX2010003156A (en) Tetrazole-substituted aryl amide derivatives and uses thereof.
PH12014500814A1 (en) New aryl-quinoline derivatives
MX2010009022A (en) 16 alpha, 17 alpa-acetal glucocorticosteroidal derivatives and their use.
MX2010005649A (en) Novel compounds as cannabinoid receptor ligands and uses thereof.
MX2010007392A (en) Trpa1 antagonists.
TW200745004A (en) Novel compounds, their preparation and use
TN2011000207A1 (en) Akt and p70 s6 kinase inhibitors
MX343225B (en) New aryl-benzocycloalkyl amide derivatives.
MX2012006805A (en) Indolyl-piperidinyl benzylamines as beta-tryptase inhibitors.
GEP20135959B (en) Aryl piperazine and their usage as alpha2c antagonists
MX2008012332A (en) Thiazolyldihydroindazoles.
IL200469A0 (en) Benzimidazole derivatives
MX2010004498A (en) Cyclohexeneamide derivatives and their use as trpv1 antagonist.