TN2009000100A1 - Silicon derivatives for pet imaging - Google Patents

Silicon derivatives for pet imaging

Info

Publication number: TN2009000100A1
Authority: TN; Tunisia
Prior art keywords: pet imaging; silicon derivatives; compounds; derivatives; silicon
Prior art date: 2006-10-02

Application number

TN2009000100A

Other languages

English (en)

Inventor

Ananth Srinivasan

Lutz Lehmann

Ulrike Voigtmann

Timo Stellfeld

Simon Ametamey

Ulrich Klar

Aileen Hohne

Linjing Mu

Original Assignee

Bayer Schering Pharma Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-10-02

Filing date

2009-03-25

Publication date

2010-08-19

2006-10-02 Priority claimed from EP06076823A external-priority patent/EP1908472A1/fr

2006-10-11 Priority claimed from EP06076869A external-priority patent/EP1911452A1/fr

2007-03-12 Priority claimed from EP07090043A external-priority patent/EP1970064A1/fr

2007-04-23 Priority claimed from EP07090079A external-priority patent/EP1985624A3/fr

2009-03-25 Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag

2010-08-19 Publication of TN2009000100A1 publication Critical patent/TN2009000100A1/fr

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/13—Labelling of peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/695—Silicon compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A61K49/08—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
- A61K49/085—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier conjugated systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A61K49/08—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
- A61K49/10—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/06—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations
- A61K49/08—Nuclear magnetic resonance [NMR] contrast preparations; Magnetic resonance imaging [MRI] contrast preparations characterised by the carrier
- A61K49/10—Organic compounds
- A61K49/14—Peptides, e.g. proteins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0491—Sugars, nucleosides, nucleotides, oligonucleotides, nucleic acids, e.g. DNA, RNA, nucleic acid aptamers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/004—Acyclic, carbocyclic or heterocyclic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen, sulfur, selenium or tellurium
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/008—Peptides; Proteins
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0834—Compounds having one or more O-Si linkage
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0896—Compounds with a Si-H linkage
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/12—Organo silicon halides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
- C07K7/086—Bombesin; Related peptides

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Molecular Biology (AREA)
Epidemiology (AREA)
Biochemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Radiology & Medical Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Analytical Chemistry (AREA)
Biotechnology (AREA)
Physics & Mathematics (AREA)
Optics & Photonics (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Peptides Or Proteins (AREA)
Nuclear Medicine (AREA)

TN2009000100A 2006-10-02 2009-03-25 Silicon derivatives for pet imaging TN2009000100A1 (en)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
EP06076823A EP1908472A1 (fr)	2006-10-02	2006-10-02	Dérivés de silicone pour l'imagerie TEP
EP06076869A EP1911452A1 (fr)	2006-10-11	2006-10-11	Dérivés de silicone pour l'imagerie TEP
EP07090043A EP1970064A1 (fr)	2007-03-12	2007-03-12	Dérivés de silicone pour l'imagerie TEP
EP07090079A EP1985624A3 (fr)	2007-04-23	2007-04-23	Procédé simple de radiofluorination de composés actifs biologiquement ou de biomolécules
PCT/EP2007/008044 WO2008040441A2 (fr)	2006-10-02	2007-09-07	Radiofluoration

Publications (1)

Publication Number	Publication Date
TN2009000100A1 true TN2009000100A1 (en)	2010-08-19

Family

ID=39030886

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TN2009000100A TN2009000100A1 (en)	2006-10-02	2009-03-25	Silicon derivatives for pet imaging

Country Status (21)

Country	Link
US (1)	US20090035215A1 (fr)
EP (1)	EP2074135A2 (fr)
JP (1)	JP2010505776A (fr)
KR (1)	KR20090085599A (fr)
AR (1)	AR062795A1 (fr)
AU (1)	AU2007304508A1 (fr)
BR (1)	BRPI0719956A2 (fr)
CA (1)	CA2664700A1 (fr)
CO (1)	CO6180444A2 (fr)
CR (1)	CR10703A (fr)
IL (1)	IL197817A0 (fr)
MA (1)	MA30824B1 (fr)
MX (1)	MX2009003617A (fr)
NO (1)	NO20091735L (fr)
PA (1)	PA8747601A1 (fr)
PE (1)	PE20081173A1 (fr)
SV (1)	SV2009003205A (fr)
TN (1)	TN2009000100A1 (fr)
TW (1)	TW200820988A (fr)
UY (1)	UY30596A1 (fr)
WO (1)	WO2008040441A2 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2627486T3 (es)	2010-01-25	2017-07-28	Institut National De La Sante Et De La Recherche Medicale (Inserm)	Biomoléculas sililadas
JP5717138B2 (ja) *	2011-05-23	2015-05-13	独立行政法人産業技術総合研究所	タンパク質固定化表面修飾材料
CN105452262A (zh) *	2013-06-06	2016-03-30	日产化学工业株式会社	烷氧基硅烷化合物、液晶取向剂、液晶取向膜和液晶表示元件
CA2982269C (fr) *	2015-05-26	2023-12-05	The Regents Of The University Of California	Accepteurs silicium-fluorure heteroaromatiques utiles pour de marquage 18f de molecules et de biomolecules, et methodes de preparation
US11464784B2 (en)	2017-09-15	2022-10-11	The Regents Of The University Of California	Inhibition of aminocylase 3 (AA3) in the treatment of cancer
WO2021226076A1 (fr) *	2020-05-04	2021-11-11	The Research Foundation For The State University Of New York	Composition d'agent d'imagerie pour tomographie par émission de positrons et procédé de détection d'infection bactérienne
WO2022064812A1 (fr) *	2020-09-28	2022-03-31	国立研究開発法人量子科学技術研究開発機構	Procédé de production d'une substance marquée radioactive, dispositif de production d'une substance marquée radioactive, et procédé d'évaporation et de concentration de nucléide métallique radioactif

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5084555A (en) *	1989-08-21	1992-01-28	The Administrators Of The Tulane Educational Fund	An octapeptide bombesin analog
US5732578A (en) *	1995-02-24	1998-03-31	Hyundai Metal Co., Ltd.	Device for maintaining the horizontality of a door lock lever
TW432073B (en) *	1995-12-28	2001-05-01	Pfizer	Pyrazolopyridine compounds
US6639076B1 (en) *	1998-08-18	2003-10-28	Eli Lilly And Company	Growth hormone secretagogues
DE60022508T2 (de) *	1999-06-14	2006-06-08	Eli Lilly And Co., Indianapolis	Inhibitoren von serin proteasen
WO2002044144A2 (fr) *	2000-11-30	2002-06-06	Advanced Research And Technology Institute, Inc.	Utilisation de nucleophiles pour preparer des agents d'imagerie radiomarques, et composes associes
GB0206750D0 (en) *	2002-03-22	2002-05-01	Amersham Plc	Radiofluorination methods
US7342095B2 (en) *	2003-02-20	2008-03-11	University Of South Florida	Peptidomimetic inhibitors of STAT activity and uses thereof
GB0305704D0 (en) *	2003-03-13	2003-04-16	Amersham Plc	Radiofluorination methods
WO2005077967A1 (fr) *	2004-02-13	2005-08-25	The University Of British Columbia	Composes et compositions radiomarques, leurs precurseurs et leurs procedes de production
US20080029548A1 (en) *	2006-05-05	2008-02-07	Ann De Wree	Fabric treatment dispensing package

2007
- 2007-09-07 US US11/851,936 patent/US20090035215A1/en not_active Abandoned
- 2007-09-07 EP EP07818173A patent/EP2074135A2/fr not_active Withdrawn
- 2007-09-07 MX MX2009003617A patent/MX2009003617A/es not_active Application Discontinuation
- 2007-09-07 WO PCT/EP2007/008044 patent/WO2008040441A2/fr not_active Ceased
- 2007-09-07 CA CA002664700A patent/CA2664700A1/fr not_active Abandoned
- 2007-09-07 AU AU2007304508A patent/AU2007304508A1/en not_active Abandoned
- 2007-09-07 KR KR1020097009044A patent/KR20090085599A/ko not_active Withdrawn
- 2007-09-07 JP JP2009530773A patent/JP2010505776A/ja active Pending
- 2007-09-07 BR BRPI0719956-2A2A patent/BRPI0719956A2/pt not_active IP Right Cessation
- 2007-09-10 TW TW096133834A patent/TW200820988A/zh unknown
- 2007-09-14 AR ARP070104086A patent/AR062795A1/es unknown
- 2007-09-14 PE PE2007001246A patent/PE20081173A1/es not_active Application Discontinuation
- 2007-09-14 UY UY30596A patent/UY30596A1/es not_active Application Discontinuation
- 2007-09-14 PA PA20078747601A patent/PA8747601A1/es unknown
2009
- 2009-03-25 TN TN2009000100A patent/TN2009000100A1/fr unknown
- 2009-03-26 IL IL197817A patent/IL197817A0/en unknown
- 2009-04-01 CR CR10703A patent/CR10703A/es not_active Application Discontinuation
- 2009-04-02 CO CO09034043A patent/CO6180444A2/es not_active Application Discontinuation
- 2009-04-02 SV SV2009003205A patent/SV2009003205A/es not_active Application Discontinuation
- 2009-04-30 NO NO20091735A patent/NO20091735L/no not_active Application Discontinuation
- 2009-04-30 MA MA31834A patent/MA30824B1/fr unknown

Also Published As

Publication number	Publication date
AU2007304508A8 (en)	2009-05-14
MX2009003617A (es)	2009-04-22
SV2009003205A (es)	2009-10-19
JP2010505776A (ja)	2010-02-25
WO2008040441A3 (fr)	2009-01-08
UY30596A1 (es)	2008-05-02
CO6180444A2 (es)	2010-07-19
PA8747601A1 (es)	2009-08-26
EP2074135A2 (fr)	2009-07-01
US20090035215A1 (en)	2009-02-05
NO20091735L (no)	2009-06-30
WO2008040441A2 (fr)	2008-04-10
PE20081173A1 (es)	2008-11-06
AU2007304508A1 (en)	2008-04-10
MA30824B1 (fr)	2009-10-01
BRPI0719956A2 (pt)	2014-04-29
TW200820988A (en)	2008-05-16
AR062795A1 (es)	2008-12-03
CR10703A (es)	2009-06-25
IL197817A0 (en)	2009-12-24
CA2664700A1 (fr)	2008-04-10
KR20090085599A (ko)	2009-08-07

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IL181529A0 (en)	2007-07-04	Diagnostic compounds
TN2009000100A1 (en)	2010-08-19	Silicon derivatives for pet imaging
WO2009046842A3 (fr)	2009-06-25	Dérivés de thiazole
MX2009007713A (es)	2009-07-29	Derivados de piridazina, procedimientos para su preparacion y su uso como fungicidas.
ATE522249T1 (de)	2011-09-15	Organische verbindungen
WO2009024342A3 (fr)	2009-04-23	Nouveaux microbiocides
MX2009004435A (es)	2009-05-08	Tinturas dispersas, su preparacion y su uso.
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WO2008151828A8 (fr)	2010-01-07	Nouveaux microbiocides
IL200469A0 (en)	2010-04-29	Benzimidazole derivatives
EA200901142A1 (ru)	2010-04-30	18f фторбензоильные меченые биологически активные соединения в качестве диагностических визуализирующих средств, а также бензотриазол-1-илоксибензоильные, 2,5-(диоксопирролидин-1-илокси)бензоильные и триметиламмониобензоильные предшественники
MX2011007266A (es)	2011-08-08	Microbiocidas nuevos.
WO2009127718A3 (fr)	2010-02-04	Nouveaux microbiocides
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WO2008083191A3 (fr)	2009-08-06	Procédés de radiofluoration
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