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TN2009000093A1 - Pharmaceutical compositions comprising nilotinib or its salt - Google Patents

Pharmaceutical compositions comprising nilotinib or its salt

Info

Publication number
TN2009000093A1
TN2009000093A1 TN2009000093A TN2009000093A TN2009000093A1 TN 2009000093 A1 TN2009000093 A1 TN 2009000093A1 TN 2009000093 A TN2009000093 A TN 2009000093A TN 2009000093 A TN2009000093 A TN 2009000093A TN 2009000093 A1 TN2009000093 A1 TN 2009000093A1
Authority
TN
Tunisia
Prior art keywords
salt
nilotinib
pharmaceutical compositions
granules
produced
Prior art date
Application number
TN2009000093A
Other languages
English (en)
Inventor
Nathalie Bruneau
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37684496&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2009000093(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of TN2009000093A1 publication Critical patent/TN2009000093A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1641Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
    • A61K9/1623Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1629Organic macromolecular compounds
    • A61K9/1635Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
TN2009000093A 2006-09-27 2009-03-19 Pharmaceutical compositions comprising nilotinib or its salt TN2009000093A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06121371A EP1923053A1 (fr) 2006-09-27 2006-09-27 Composition pharmaceutique comprenant de la nilotinib ou son sel
PCT/EP2007/060165 WO2008037716A2 (fr) 2006-09-27 2007-09-25 Compositions pharmaceutiques

Publications (1)

Publication Number Publication Date
TN2009000093A1 true TN2009000093A1 (en) 2010-08-19

Family

ID=37684496

Family Applications (1)

Application Number Title Priority Date Filing Date
TN2009000093A TN2009000093A1 (en) 2006-09-27 2009-03-19 Pharmaceutical compositions comprising nilotinib or its salt

Country Status (34)

Country Link
US (2) US8293756B2 (fr)
EP (4) EP1923053A1 (fr)
JP (2) JP5567340B2 (fr)
KR (2) KR101598747B1 (fr)
CN (2) CN101516344A (fr)
AR (1) AR062980A1 (fr)
AU (1) AU2007301977B2 (fr)
BR (1) BRPI0719438B1 (fr)
CA (1) CA2662571C (fr)
CL (1) CL2007002766A1 (fr)
CO (1) CO6160288A2 (fr)
CY (2) CY1117021T1 (fr)
DK (2) DK3984528T3 (fr)
ES (3) ES2957912T3 (fr)
FI (2) FI3984528T3 (fr)
HR (2) HRP20151383T4 (fr)
HU (2) HUE028204T2 (fr)
IL (1) IL197496A (fr)
JO (1) JO3757B1 (fr)
LT (1) LT3984528T (fr)
MA (1) MA30807B1 (fr)
MX (1) MX2009003184A (fr)
MY (1) MY148237A (fr)
NO (2) NO346639B1 (fr)
NZ (1) NZ575317A (fr)
PE (2) PE20120626A1 (fr)
PL (2) PL2068839T5 (fr)
PT (2) PT3984528T (fr)
RU (1) RU2469707C2 (fr)
SI (2) SI2068839T2 (fr)
TN (1) TN2009000093A1 (fr)
TW (3) TWI428333B (fr)
WO (1) WO2008037716A2 (fr)
ZA (1) ZA200901511B (fr)

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EP1923053A1 (fr) 2006-09-27 2008-05-21 Novartis AG Composition pharmaceutique comprenant de la nilotinib ou son sel
CA2775400A1 (fr) 2009-09-28 2011-03-31 Medizinische Universitat Wien Nouvelle utilisation des inhibiteurs de pdgf-beta
NZ599217A (en) * 2009-10-23 2014-05-30 Novartis Ag Method of treating proliferative disorders and other pathological conditions mediated by bcr-abl, c-kit, ddr1, ddr2 or pdgf-r kinase activity
JO3634B1 (ar) 2009-11-17 2020-08-27 Novartis Ag طريقة لعلاج اضطرابات تكاثرية وحالات مرضية أخرى متوسطة بنشاط كيناز bcr-abl، c-kit، ddr1، ddr2، أو pdgf-r
WO2012164578A1 (fr) * 2011-06-02 2012-12-06 Hetero Research Foundation Compositions et procédés de préparation de formulations de nilotinib à libération immédiate
AR086913A1 (es) * 2011-06-14 2014-01-29 Novartis Ag 4-metil-3-[[4-(3-piridinil)-2-pirimidinil]-amino]-n-[5-(4-metil-1h-imidazol-1-il)-3-(trifluoro-metil)-fenil]-benzamida amorfa, forma de dosificacion que la contiene y metodo para prepararlas
CN102321073A (zh) * 2011-08-12 2012-01-18 西安交通大学 一种尼罗替尼的制备方法
WO2013063003A1 (fr) 2011-10-28 2013-05-02 Novartis Ag Méthode de traitement des tumeurs stromales gastro-intestinales
US20140288073A1 (en) 2011-10-28 2014-09-25 Novartis Ag Method of Treating Gastrointestinal Stromal Tumors
US9301957B2 (en) 2011-11-14 2016-04-05 Novartis Ag Immediate release 4-methyl-3-4[[4-(3-pyridinyl)-2-pyrimidinyl]amino]-N-[5-(4-methyl-1H-imidazol-1-YL)-3-(trifluoromethyl)phenyl] benzamide formulation
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AU2017232868B2 (en) * 2016-03-17 2021-07-22 Sun Pharmaceutical Industries Ltd. Pharmaceutical composition of nilotinib
CN107582531B (zh) * 2016-07-06 2020-12-29 四川科伦药物研究院有限公司 一种利伐沙班固体制剂及其制备方法
CN107320460B (zh) * 2017-08-04 2020-11-03 北京化工大学 一种尼罗替尼口服纳米制剂及其制备方法
CN107441094B (zh) * 2017-08-08 2020-05-22 南方医科大学 尼罗替尼作为治疗登革病毒感染的药物及其制药用途
CZ2017821A3 (cs) 2017-12-20 2019-07-03 Zentiva, K.S. Léková forma obsahující krystalický nilotinib
JP7409696B2 (ja) 2018-06-15 2024-01-09 ハンダ ファーマシューティカルズ インコーポレイテッド キナーゼ阻害剤の塩およびその組成物
JP2023513045A (ja) * 2020-01-31 2023-03-30 ナノコピーア リミテッド ライアビリティ カンパニー 非晶質ニロチニブ微粒子及びその使用
IL297776A (en) 2020-04-30 2022-12-01 Nanocopoeia Llc Orally disintegrating tablets containing an amorphous solid dispersion of nalotinib
JP7489849B2 (ja) * 2020-07-20 2024-05-24 日本化薬株式会社 ニロチニブ錠剤
AU2021353684A1 (en) 2020-09-29 2023-06-08 Shenzhen Pharmacin Co., Ltd. Pharmaceutical compositions
WO2022263510A1 (fr) 2021-06-19 2022-12-22 Helm Ag Composition de granulés comprenant de la nisine
WO2023285981A1 (fr) * 2021-07-15 2023-01-19 Torrent Pharmaceuticals Limited Composition pharmaceutique liquide stable de nilotinib
EP4122452A1 (fr) 2021-07-23 2023-01-25 KRKA, d.d., Novo mesto Composition pharmaceutique comprenant du nilotinib et son procédé de fabrication
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WO2024194718A1 (fr) * 2023-03-22 2024-09-26 Unichem Laboratories Limited Composition pharmaceutique stable et son procédé de préparation

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Also Published As

Publication number Publication date
EP3984528B1 (fr) 2023-07-05
ZA200901511B (en) 2010-02-24
HUE028204T2 (en) 2016-12-28
BRPI0719438B1 (pt) 2022-04-19
JP2010504942A (ja) 2010-02-18
HRP20151383T1 (hr) 2016-01-15
TWI428333B (zh) 2014-03-01
CY1126116T1 (el) 2023-11-15
LT3984528T (lt) 2023-08-10
FI2068839T4 (fi) 2023-01-31
SI3984528T1 (sl) 2023-09-29
US8501760B2 (en) 2013-08-06
NO20220946A1 (no) 2009-04-24
AU2007301977A1 (en) 2008-04-03
PE20120626A1 (es) 2012-06-07
CN104306350A (zh) 2015-01-28
AR062980A1 (es) 2008-12-17
TWI540128B (zh) 2016-07-01
RU2469707C2 (ru) 2012-12-20
PT3984528T (pt) 2023-08-07
IL197496A (en) 2016-04-21
ES2951547T3 (es) 2023-10-23
US8293756B2 (en) 2012-10-23
KR101598747B1 (ko) 2016-03-02
TW200821298A (en) 2008-05-16
PL2068839T3 (pl) 2016-06-30
CY1117021T1 (el) 2017-04-05
CA2662571C (fr) 2016-09-27
HRP20151383T4 (hr) 2023-03-03
CL2007002766A1 (es) 2008-08-08
EP3984528A1 (fr) 2022-04-20
PT2068839E (pt) 2015-12-30
AU2007301977B2 (en) 2011-09-08
DK2068839T3 (da) 2016-01-11
KR20140121903A (ko) 2014-10-16
PL3984528T3 (pl) 2023-08-28
HK1133193A1 (en) 2010-03-19
ES2556625T5 (es) 2023-03-02
HRP20230753T3 (hr) 2023-10-27
IL197496A0 (en) 2009-12-24
JO3757B1 (ar) 2021-01-31
PE20081379A1 (es) 2008-11-27
RU2009115782A (ru) 2010-11-10
EP1923053A1 (fr) 2008-05-21
NO346639B1 (no) 2022-11-07
HUE063083T2 (hu) 2023-12-28
JP2014065715A (ja) 2014-04-17
EP3009128B1 (fr) 2023-07-05
US20130023549A1 (en) 2013-01-24
MA30807B1 (fr) 2009-10-01
NO347404B1 (no) 2023-10-16
NZ575317A (en) 2011-12-22
ES2957912T3 (es) 2024-01-29
BRPI0719438A2 (pt) 2013-12-10
EP3009128A1 (fr) 2016-04-20
NO20091501L (no) 2009-04-24
JP5567340B2 (ja) 2014-08-06
DK3984528T3 (da) 2023-07-31
KR20090076931A (ko) 2009-07-13
CN101516344A (zh) 2009-08-26
CA2662571A1 (fr) 2008-04-03
MX2009003184A (es) 2009-04-03
SI2068839T2 (sl) 2023-01-31
EP2068839B1 (fr) 2015-09-23
FI3984528T3 (fi) 2023-07-27
WO2008037716A2 (fr) 2008-04-03
PL2068839T5 (pl) 2023-01-30
US20100087463A1 (en) 2010-04-08
SI2068839T1 (sl) 2016-02-29
WO2008037716A3 (fr) 2008-07-17
ES2556625T3 (es) 2016-01-19
EP2068839A2 (fr) 2009-06-17
CO6160288A2 (es) 2010-05-20
TW201418245A (zh) 2014-05-16
TW201418244A (zh) 2014-05-16
EP2068839B2 (fr) 2022-10-12
MY148237A (en) 2013-03-29

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