SV2007002357A - DERIVED FROM QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING IT REF. P-SV-79232 / UG - Google Patents
DERIVED FROM QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING IT REF. P-SV-79232 / UGInfo
- Publication number
- SV2007002357A SV2007002357A SV2005002357A SV2005002357A SV2007002357A SV 2007002357 A SV2007002357 A SV 2007002357A SV 2005002357 A SV2005002357 A SV 2005002357A SV 2005002357 A SV2005002357 A SV 2005002357A SV 2007002357 A SV2007002357 A SV 2007002357A
- Authority
- SV
- El Salvador
- Prior art keywords
- preparation
- quinolina
- ref
- derived
- product containing
- Prior art date
Links
- 229940126601 medicinal product Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- SMWDFEZZVXVKRB-UHFFFAOYSA-N Quinoline Chemical class N1=CC=CC2=CC=CC=C21 SMWDFEZZVXVKRB-UHFFFAOYSA-N 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
LA PRESENTE INVENCION SE REFIERE A UN DERIVADO DE QUINOLINA DE LA FORMULA GENERAL A, VER FORMULA,EN LA QUE R1, R2, R3, X, Y, Z Y A SE INDICAN EN LA DESCRIPCION Y EN LAS REIVINDICACIONES, AL USO DE LOS COMPUESTOS LA FORMULA GENERAL A PARA EL TRATAMIENTO DE DIVERSAS ENFERMEDADES, ASI COMO A LA PREPARACION DE COMPUESTOS LA FORMULA GENERAL ATHE PRESENT INVENTION REFERS TO A QUINOLINE DERIVATIVE OF THE GENERAL FORMULA A, SEE FORMULA, IN WHICH R1, R2, R3, X, Y, ZYA ARE INDICATED IN THE DESCRIPTION AND IN THE CLAIMS, TO THE USE OF THE COMPOUNDS THE FORMULA GENERAL A FOR THE TREATMENT OF VARIOUS DISEASES, AS WELL AS TO THE PREPARATION OF COMPOUNDS THE GENERAL FORMULA A
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004063223A DE102004063223A1 (en) | 2004-12-22 | 2004-12-22 | New quinoline derivatives are ephrin receptor kinase inhibitors useful for the treatment of e.g. blood vessels diseases, hyperproliferations, chronic or acute neurodegenerative diseases, psoriasis, eczema and scleroderma |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2007002357A true SV2007002357A (en) | 2007-02-16 |
Family
ID=36599298
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2005002357A SV2007002357A (en) | 2004-12-22 | 2005-12-22 | DERIVED FROM QUINOLINA, ITS USE, PREPARATION AND MEDICINAL PRODUCT CONTAINING IT REF. P-SV-79232 / UG |
Country Status (7)
| Country | Link |
|---|---|
| CN (1) | CN101087788A (en) |
| AR (1) | AR052544A1 (en) |
| DE (1) | DE102004063223A1 (en) |
| GT (1) | GT200500381A (en) |
| PA (1) | PA8657701A1 (en) |
| SV (1) | SV2007002357A (en) |
| UY (1) | UY29308A1 (en) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103382206B (en) * | 2012-05-04 | 2016-09-28 | 上海恒瑞医药有限公司 | Quinoline or quinazoline derivative, its preparation method and in application pharmaceutically |
| CN106565823B (en) * | 2016-11-10 | 2020-09-11 | 珠海诺贝尔国际生物医药研究院有限公司 | Eph receptor small molecule inhibitor and preparation method thereof |
| CN110577546B (en) * | 2018-06-08 | 2021-09-07 | 江苏威凯尔医药科技有限公司 | VEGFR inhibitor and preparation method and application thereof |
| WO2019233458A1 (en) * | 2018-06-08 | 2019-12-12 | 江苏威凯尔医药科技有限公司 | Vegfr inhibitor, preparation method therefor and use thereof |
| CN113150009B (en) * | 2020-01-07 | 2023-05-23 | 爱科诺生物医药(香港)有限公司 | Heterocyclic compound with activity of inhibiting programmed cell necrosis pathway and application thereof |
| CN113061142B (en) * | 2020-01-02 | 2024-08-27 | 爱科诺生物医药(香港)有限公司 | Heterocyclic compound with activity of inhibiting programmed cell necrosis pathway and application thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3919238A (en) * | 1973-06-06 | 1975-11-11 | Morton Norwich Products Inc | 9-(Substituted amino)imidazo(4,5-f) quinolines |
| EP0187705A3 (en) * | 1985-01-08 | 1988-05-11 | Norwich Eaton Pharmaceuticals, Inc. | Imidazo(4,5-f)quinolines useful as immunomodulating agents |
| FI940469A7 (en) * | 1991-08-02 | 1994-02-01 | Pfizer | Quinoline derivatives as immunostimulants |
-
2004
- 2004-12-22 DE DE102004063223A patent/DE102004063223A1/en not_active Ceased
-
2005
- 2005-12-19 CN CNA2005800444603A patent/CN101087788A/en active Pending
- 2005-12-21 GT GT200500381A patent/GT200500381A/en unknown
- 2005-12-22 SV SV2005002357A patent/SV2007002357A/en not_active Application Discontinuation
- 2005-12-22 UY UY29308A patent/UY29308A1/en not_active Application Discontinuation
- 2005-12-22 PA PA20058657701A patent/PA8657701A1/en unknown
- 2005-12-22 AR ARP050105485A patent/AR052544A1/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| DE102004063223A1 (en) | 2006-07-13 |
| CN101087788A (en) | 2007-12-12 |
| PA8657701A1 (en) | 2006-09-08 |
| GT200500381A (en) | 2006-08-03 |
| UY29308A1 (en) | 2006-06-30 |
| AR052544A1 (en) | 2007-03-21 |
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