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SV2005001918A - Metodos para preparar derivados 7-(b-d-ribofuranosilo sustituido en 2')-4 (nr2r3)-5(etin-1-ilo sustituido)-pirrol[2,3-d]pirimidina - Google Patents

Metodos para preparar derivados 7-(b-d-ribofuranosilo sustituido en 2')-4 (nr2r3)-5(etin-1-ilo sustituido)-pirrol[2,3-d]pirimidina

Info

Publication number
SV2005001918A
SV2005001918A SV2004001918A SV2004001918A SV2005001918A SV 2005001918 A SV2005001918 A SV 2005001918A SV 2004001918 A SV2004001918 A SV 2004001918A SV 2004001918 A SV2004001918 A SV 2004001918A SV 2005001918 A SV2005001918 A SV 2005001918A
Authority
SV
El Salvador
Prior art keywords
ribofuranosil
pirrol
etin
ilo
pyrimidine
Prior art date
Application number
SV2004001918A
Other languages
English (en)
Inventor
Jesse D Keicher
Christopher Don Roberts
Natalia B Dyatkina
Original Assignee
Genelabs Tech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US10/861,311 external-priority patent/US7144868B2/en
Priority claimed from US10/861,090 external-priority patent/US7202223B2/en
Application filed by Genelabs Tech Inc filed Critical Genelabs Tech Inc
Publication of SV2005001918A publication Critical patent/SV2005001918A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/14Pyrrolo-pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

METODOS E INTERMEDIARIOS PARA LA PREPARACION DE COMPUESTOS 7-(B-D- RIBOFURANOSILO SUSTITUIDO EN 2-R1) -4-AMINO -5-(ETIN -1-ILO OPCIONALMENTE SUSTITUIDO ) -PIRROL [2,3-D] PIRIMIDINA . ESTOS COMPUESTOS SON DE UTILIDAD EN EL TRATAMIENTO DE LAS INFECCIONES VIRALES CAUSADAS POR LA FAMILIA DE VIRUS, FLAVIVIRIDAE, TAL COMO EL VIRUS DE LA HEPATITIS C
SV2004001918A 2003-10-27 2004-10-27 Metodos para preparar derivados 7-(b-d-ribofuranosilo sustituido en 2')-4 (nr2r3)-5(etin-1-ilo sustituido)-pirrol[2,3-d]pirimidina SV2005001918A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US51515303P 2003-10-27 2003-10-27
US10/861,311 US7144868B2 (en) 2003-10-27 2004-06-04 Nucleoside compounds for treating viral infections
US10/861,090 US7202223B2 (en) 2003-10-27 2004-06-04 Nucleoside compounds for treating viral infections
US60281504P 2004-08-18 2004-08-18

Publications (1)

Publication Number Publication Date
SV2005001918A true SV2005001918A (es) 2005-04-18

Family

ID=34577847

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2004001918A SV2005001918A (es) 2003-10-27 2004-10-27 Metodos para preparar derivados 7-(b-d-ribofuranosilo sustituido en 2')-4 (nr2r3)-5(etin-1-ilo sustituido)-pirrol[2,3-d]pirimidina

Country Status (7)

Country Link
US (1) US7169918B2 (es)
EP (1) EP1682564A1 (es)
AR (1) AR046201A1 (es)
CA (1) CA2543116A1 (es)
SV (1) SV2005001918A (es)
UY (1) UY28582A1 (es)
WO (1) WO2005044835A1 (es)

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Also Published As

Publication number Publication date
CA2543116A1 (en) 2005-05-19
US7169918B2 (en) 2007-01-30
US20050215510A1 (en) 2005-09-29
AR046201A1 (es) 2005-11-30
EP1682564A1 (en) 2006-07-26
UY28582A1 (es) 2005-05-31
WO2005044835A1 (en) 2005-05-19

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