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SK16242002A3 - Derivát triazolu a farmaceutický prostriedok, ktorý ho obsahuje - Google Patents

Derivát triazolu a farmaceutický prostriedok, ktorý ho obsahuje Download PDF

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Publication number
SK16242002A3
SK16242002A3 SK1624-2002A SK16242002A SK16242002A3 SK 16242002 A3 SK16242002 A3 SK 16242002A3 SK 16242002 A SK16242002 A SK 16242002A SK 16242002 A3 SK16242002 A3 SK 16242002A3
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SK
Slovakia
Prior art keywords
group
fab
optionally substituted
lower alkyl
atom
Prior art date
Application number
SK1624-2002A
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English (en)
Slovak (sk)
Inventor
Takahiko Tobe
Takashi Sugane
Wataru Hamaguchi
Itsuro Shimada
Kyoichi Maeno
Junji Miyata
Takeshi Suzuki
Atsuyuki Kohara
Takuma Morita
Tetsuya Kimizuka
Michael Arlt
Hartmut Greiner
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Merck Patent Gmbh
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Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SK16242002A3 publication Critical patent/SK16242002A3/sk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/425—Thiazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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    • C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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SK1624-2002A 2000-05-19 2001-05-17 Derivát triazolu a farmaceutický prostriedok, ktorý ho obsahuje SK16242002A3 (sk)

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AR030933A1 (es) 2003-09-03
AU2001256769A1 (en) 2001-11-26
JP3873746B2 (ja) 2007-01-24
KR100776119B1 (ko) 2007-11-16
NO20025517L (no) 2002-11-18
CN1237055C (zh) 2006-01-18
CZ20023763A3 (cs) 2003-03-12
EP1293503A4 (en) 2008-04-02
NO20025517D0 (no) 2002-11-18
RU2002133666A (ru) 2007-05-10
KR20030019386A (ko) 2003-03-06
HUP0302415A2 (hu) 2003-11-28
EP1293503A1 (en) 2003-03-19
US7084164B2 (en) 2006-08-01
US20060025461A1 (en) 2006-02-02
PL359340A1 (en) 2004-08-23
BR0110961A (pt) 2004-06-29
CA2409819C (en) 2009-09-15
CA2409819A1 (en) 2002-11-18
WO2001087855A1 (en) 2001-11-22
CN1429215A (zh) 2003-07-09

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