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SI2767285T1 - Tableta, ki vsebuje 7-(4-(4-benzo(b)tiofen-4-IL-piperazin-1-IL)butoksi)-1H-kinolin-2-ON ali njegovo sol - Google Patents

Tableta, ki vsebuje 7-(4-(4-benzo(b)tiofen-4-IL-piperazin-1-IL)butoksi)-1H-kinolin-2-ON ali njegovo sol

Info

Publication number
SI2767285T1
SI2767285T1 SI201231718T SI201231718T SI2767285T1 SI 2767285 T1 SI2767285 T1 SI 2767285T1 SI 201231718 T SI201231718 T SI 201231718T SI 201231718 T SI201231718 T SI 201231718T SI 2767285 T1 SI2767285 T1 SI 2767285T1
Authority
SI
Slovenia
Prior art keywords
quinolin
thiophen
piperazin
benzo
butoxy
Prior art date
Application number
SI201231718T
Other languages
English (en)
Other versions
SI2767285T2 (sl
Inventor
Yoshiharu Inoue
Original Assignee
Otsuka Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48081918&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI2767285(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharmaceutical Co., Ltd. filed Critical Otsuka Pharmaceutical Co., Ltd.
Publication of SI2767285T1 publication Critical patent/SI2767285T1/sl
Publication of SI2767285T2 publication Critical patent/SI2767285T2/sl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2813Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Supply Of Fluid Materials To The Packaging Location (AREA)
  • Basic Packing Technique (AREA)
SI201231718T 2011-10-14 2012-10-12 Tableta, ki vsebuje 7-(4-(4-benzo(b)tiofen-4-IL-piperazin-1-IL)butoksi)-1H-kinolin-2-ON ali njegovo sol SI2767285T2 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2011227057 2011-10-14
EP12840025.6A EP2767285B2 (en) 2011-10-14 2012-10-12 TABLET COMPRISING 7-[4-(4-BENZO[b]THIOPHEN-4-YL-PIPERAZIN-1-YL) BUTOXY]-1H-QUINOLIN-2-ONE OR A SALT THEREOF
PCT/JP2012/076415 WO2013054872A1 (ja) 2011-10-14 2012-10-12 7-[4-(4-ベンゾ[b]チオフェン-4-イル-ピペラジン-1-イル)ブトキシ]-1H-キノリン-2-オン又はその塩を含む錠剤

Publications (2)

Publication Number Publication Date
SI2767285T1 true SI2767285T1 (sl) 2020-03-31
SI2767285T2 SI2767285T2 (sl) 2025-06-30

Family

ID=48081918

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201231718T SI2767285T2 (sl) 2011-10-14 2012-10-12 Tableta, ki vsebuje 7-(4-(4-benzo(b)tiofen-4-IL-piperazin-1-IL)butoksi)-1H-kinolin-2-ON ali njegovo sol

Country Status (34)

Country Link
US (8) US20140234417A1 (sl)
EP (1) EP2767285B2 (sl)
JP (2) JP6084161B2 (sl)
KR (1) KR102072371B1 (sl)
CN (2) CN107397730A (sl)
AP (1) AP2014007564A0 (sl)
AR (1) AR088319A1 (sl)
AU (1) AU2012321723C1 (sl)
BR (1) BR112014008603A2 (sl)
CA (1) CA2851588C (sl)
CL (1) CL2014000909A1 (sl)
CO (1) CO6950480A2 (sl)
CY (1) CY1122460T1 (sl)
DK (1) DK2767285T4 (sl)
EA (1) EA032930B1 (sl)
ES (1) ES2762479T5 (sl)
FI (1) FI2767285T4 (sl)
HR (1) HRP20200037T4 (sl)
HU (1) HUE047493T2 (sl)
IL (1) IL231513B (sl)
IN (1) IN2014DN02055A (sl)
JO (1) JO3753B1 (sl)
LT (1) LT2767285T (sl)
MX (1) MX376092B (sl)
MY (1) MY173370A (sl)
PH (1) PH12014500607A1 (sl)
PL (1) PL2767285T5 (sl)
PT (1) PT2767285T (sl)
SG (2) SG2014013783A (sl)
SI (1) SI2767285T2 (sl)
TW (1) TWI634908B (sl)
UA (1) UA114411C2 (sl)
WO (1) WO2013054872A1 (sl)
ZA (1) ZA201402333B (sl)

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JP7060878B2 (ja) * 2016-07-27 2022-04-27 日本臓器製薬株式会社 メトトレキサート含有フィルムコーティング錠
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EP3500247B1 (en) 2016-08-16 2020-05-27 H e x a l Aktiengesellschaft Immediate release tablet of a benzothiophene compound
CN106496206A (zh) * 2016-08-31 2017-03-15 安徽省润生医药股份有限公司 一种依匹哌唑新的制备方法
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JP7166754B2 (ja) * 2017-11-22 2022-11-08 沢井製薬株式会社 ダサチニブ無水物含有製剤
EP3501506B1 (en) 2017-12-19 2019-10-09 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical tablet composition comprising brexpiprazole
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WO2021029020A1 (ja) * 2019-08-13 2021-02-18 大塚製薬株式会社 経口医薬組成物
WO2021095092A1 (ja) * 2019-11-11 2021-05-20 大塚製薬株式会社 口腔内崩壊錠
CN112168794A (zh) * 2020-10-27 2021-01-05 浙江诺得药业有限公司 一种布瑞哌唑片的制备方法
WO2022218358A1 (zh) * 2021-04-13 2022-10-20 上海博志研新药物技术有限公司 一种布瑞哌唑物口腔薄膜剂、其制备方法及应用
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JO3753B1 (ar) * 2011-10-14 2021-01-31 Otsuka Pharma Co Ltd قرص يتألف من 7-[4-(4-بينزو[بي]ثيوفين-4-ايل-ببرازين-1-1ايل)بوتكسيل]-1اتش-كوينولين-2-وان أو ملح منه

Also Published As

Publication number Publication date
EP2767285B2 (en) 2025-02-19
US20190240215A1 (en) 2019-08-08
UA114411C2 (uk) 2017-06-12
CY1122460T1 (el) 2021-01-27
JP2017088610A (ja) 2017-05-25
EA201490783A1 (ru) 2014-07-30
LT2767285T (lt) 2020-02-10
CA2851588A1 (en) 2013-04-18
US20210023078A1 (en) 2021-01-28
KR20140075754A (ko) 2014-06-19
HUE047493T2 (hu) 2020-04-28
ES2762479T5 (en) 2025-05-30
AP2014007564A0 (en) 2014-04-30
CN103889425A (zh) 2014-06-25
CN107397730A (zh) 2017-11-28
IN2014DN02055A (sl) 2015-05-15
PL2767285T3 (pl) 2020-04-30
IL231513B (en) 2020-01-30
MX2014004135A (es) 2014-07-24
CA2851588C (en) 2019-07-02
BR112014008603A2 (pt) 2017-04-18
FI2767285T4 (fi) 2025-05-08
AR088319A1 (es) 2014-05-28
ES2762479T3 (es) 2020-05-25
HRP20200037T1 (hr) 2020-03-20
PL2767285T5 (pl) 2025-06-02
ZA201402333B (en) 2015-07-29
MY173370A (en) 2020-01-21
SG10201608412SA (en) 2016-12-29
EP2767285A1 (en) 2014-08-20
US20140234417A1 (en) 2014-08-21
EP2767285B1 (en) 2019-11-27
TW201318651A (zh) 2013-05-16
DK2767285T4 (da) 2025-04-22
EP2767285A4 (en) 2015-03-11
US20160158227A1 (en) 2016-06-09
IL231513A0 (en) 2014-04-30
JP6084161B2 (ja) 2017-02-22
HRP20200037T4 (hr) 2025-05-23
KR102072371B1 (ko) 2020-02-03
PT2767285T (pt) 2020-01-21
US20240277703A1 (en) 2024-08-22
DK2767285T3 (da) 2020-01-27
SI2767285T2 (sl) 2025-06-30
US20180008600A1 (en) 2018-01-11
CL2014000909A1 (es) 2014-11-21
CO6950480A2 (es) 2014-05-20
AU2012321723C1 (en) 2017-11-02
JO3753B1 (ar) 2021-01-31
EA032930B1 (ru) 2019-08-30
PH12014500607A1 (en) 2014-04-21
TWI634908B (zh) 2018-09-11
AU2012321723A1 (en) 2014-05-15
SG2014013783A (en) 2014-06-27
US20170165258A1 (en) 2017-06-15
US20220331311A1 (en) 2022-10-20
NZ622639A (en) 2015-11-27
AU2012321723B2 (en) 2017-07-20
JPWO2013054872A1 (ja) 2015-03-30
WO2013054872A1 (ja) 2013-04-18
MX376092B (es) 2025-03-07
US10307419B2 (en) 2019-06-04
CN103889425B (zh) 2018-08-03

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