SI2217578T1 - (1,2,4)triazolo(1,5-a)piridinske in (1,2,4)triazolo(1,5-c)pirimidinske spojine in njihova uporaba - Google Patents
(1,2,4)triazolo(1,5-a)piridinske in (1,2,4)triazolo(1,5-c)pirimidinske spojine in njihova uporabaInfo
- Publication number
- SI2217578T1 SI2217578T1 SI200831148T SI200831148T SI2217578T1 SI 2217578 T1 SI2217578 T1 SI 2217578T1 SI 200831148 T SI200831148 T SI 200831148T SI 200831148 T SI200831148 T SI 200831148T SI 2217578 T1 SI2217578 T1 SI 2217578T1
- Authority
- SI
- Slovenia
- Prior art keywords
- cćpyrimidine
- aćpyridine
- compounds
- cćpyrimidine compounds
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US97879207P | 2007-10-10 | 2007-10-10 | |
| GBGB0719803.9A GB0719803D0 (en) | 2007-10-10 | 2007-10-10 | Therapeutic compounds and their use |
| EP08806565.1A EP2217578B9 (en) | 2007-10-10 | 2008-10-10 | [1,2,4]triazolo[1,5-a]pyridine and [1,2,4]triazolo[1,5-c]pyrimidine compounds and their use |
| PCT/GB2008/003428 WO2009047514A1 (en) | 2007-10-10 | 2008-10-10 | [1,2,4]triazolo[1,5-a]pyridine and [1,2,4]triazolo[1,5-c]pyrimidine compounds and their use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI2217578T1 true SI2217578T1 (sl) | 2014-03-31 |
Family
ID=38787938
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200831148T SI2217578T1 (sl) | 2007-10-10 | 2008-10-10 | (1,2,4)triazolo(1,5-a)piridinske in (1,2,4)triazolo(1,5-c)pirimidinske spojine in njihova uporaba |
Country Status (11)
| Country | Link |
|---|---|
| US (4) | US8431596B2 (sl) |
| EP (1) | EP2217578B9 (sl) |
| CY (1) | CY1114911T1 (sl) |
| DK (1) | DK2217578T5 (sl) |
| ES (1) | ES2446298T3 (sl) |
| GB (1) | GB0719803D0 (sl) |
| HR (1) | HRP20140191T1 (sl) |
| PL (1) | PL2217578T3 (sl) |
| PT (1) | PT2217578E (sl) |
| SI (1) | SI2217578T1 (sl) |
| WO (1) | WO2009047514A1 (sl) |
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| WO2010010188A1 (en) * | 2008-07-25 | 2010-01-28 | Galapagos Nv | Novel compounds useful for the treatment of degenerative and inflammatory diseases. |
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| JO3041B1 (ar) | 2008-07-25 | 2016-09-05 | Galapagos Nv | مركبات جديدة مفيدة لمعالجة الأمراض التنكسية والالتهابية |
| WO2010010184A1 (en) * | 2008-07-25 | 2010-01-28 | Galapagos Nv | [1, 2, 4] triazolo [1, 5-a] pyridines as jak inhibitors |
| EP2323978A1 (en) * | 2008-08-12 | 2011-05-25 | Takeda Pharmaceutical Company Limited | Amide compound |
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-
2007
- 2007-10-10 GB GBGB0719803.9A patent/GB0719803D0/en not_active Ceased
-
2008
- 2008-10-10 WO PCT/GB2008/003428 patent/WO2009047514A1/en not_active Ceased
- 2008-10-10 PT PT88065651T patent/PT2217578E/pt unknown
- 2008-10-10 HR HRP20140191AT patent/HRP20140191T1/hr unknown
- 2008-10-10 ES ES08806565.1T patent/ES2446298T3/es active Active
- 2008-10-10 SI SI200831148T patent/SI2217578T1/sl unknown
- 2008-10-10 US US12/679,871 patent/US8431596B2/en not_active Expired - Fee Related
- 2008-10-10 EP EP08806565.1A patent/EP2217578B9/en not_active Revoked
- 2008-10-10 DK DK08806565.1T patent/DK2217578T5/da active
- 2008-10-10 PL PL08806565T patent/PL2217578T3/pl unknown
-
2013
- 2013-04-24 US US13/869,374 patent/US9012633B2/en active Active
-
2014
- 2014-02-24 CY CY20141100147T patent/CY1114911T1/el unknown
-
2015
- 2015-03-16 US US14/658,437 patent/US9394301B2/en not_active Expired - Fee Related
-
2016
- 2016-06-20 US US15/186,689 patent/US9771362B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EP2217578B9 (en) | 2014-09-10 |
| DK2217578T3 (da) | 2014-02-03 |
| US9012633B2 (en) | 2015-04-21 |
| US8431596B2 (en) | 2013-04-30 |
| PT2217578E (pt) | 2014-02-17 |
| PL2217578T3 (pl) | 2014-05-30 |
| ES2446298T3 (es) | 2014-03-07 |
| US20100298339A1 (en) | 2010-11-25 |
| CY1114911T1 (el) | 2016-12-14 |
| US9771362B2 (en) | 2017-09-26 |
| EP2217578B1 (en) | 2013-12-04 |
| HRP20140191T1 (hr) | 2014-04-25 |
| US20150246915A1 (en) | 2015-09-03 |
| DK2217578T5 (da) | 2014-11-10 |
| US20170066762A1 (en) | 2017-03-09 |
| WO2009047514A1 (en) | 2009-04-16 |
| EP2217578A1 (en) | 2010-08-18 |
| ES2446298T9 (es) | 2014-09-29 |
| US20140155594A1 (en) | 2014-06-05 |
| GB0719803D0 (en) | 2007-11-21 |
| US9394301B2 (en) | 2016-07-19 |
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