SI2004654T1 - Pirazolopirimidinski derivati za uporabo kot kinazni antagonisti - Google Patents
Pirazolopirimidinski derivati za uporabo kot kinazni antagonistiInfo
- Publication number
- SI2004654T1 SI2004654T1 SI200731298T SI200731298T SI2004654T1 SI 2004654 T1 SI2004654 T1 SI 2004654T1 SI 200731298 T SI200731298 T SI 200731298T SI 200731298 T SI200731298 T SI 200731298T SI 2004654 T1 SI2004654 T1 SI 2004654T1
- Authority
- SI
- Slovenia
- Prior art keywords
- pyrazolopyrimidine derivatives
- kinase antagonists
- antagonists
- kinase
- pyrazolopyrimidine
- Prior art date
Links
- 108091000080 Phosphotransferase Proteins 0.000 title 1
- 239000005557 antagonist Substances 0.000 title 1
- OGEBRHQLRGFBNV-RZDIXWSQSA-N chembl2036808 Chemical class C12=NC(NCCCC)=NC=C2C(C=2C=CC(F)=CC=2)=NN1C[C@H]1CC[C@H](N)CC1 OGEBRHQLRGFBNV-RZDIXWSQSA-N 0.000 title 1
- 102000020233 phosphotransferase Human genes 0.000 title 1
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74427006P | 2006-04-04 | 2006-04-04 | |
| US74426906P | 2006-04-04 | 2006-04-04 | |
| EP07754845.1A EP2004654B1 (en) | 2006-04-04 | 2007-04-04 | Pyrazolopyrimidine derivatives for use as kinase antagonists |
| PCT/US2007/008395 WO2007114926A2 (en) | 2006-04-04 | 2007-04-04 | Kinase antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI2004654T1 true SI2004654T1 (sl) | 2013-11-29 |
Family
ID=40743701
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI200731298T SI2004654T1 (sl) | 2006-04-04 | 2007-04-04 | Pirazolopirimidinski derivati za uporabo kot kinazni antagonisti |
Country Status (2)
| Country | Link |
|---|---|
| CN (2) | CN101448505A (sl) |
| SI (1) | SI2004654T1 (sl) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0918249D0 (en) * | 2009-10-19 | 2009-12-02 | Respivert Ltd | Compounds |
| US8399460B2 (en) * | 2009-10-27 | 2013-03-19 | Astrazeneca Ab | Chromenone derivatives |
| DE102010049595A1 (de) * | 2010-10-26 | 2012-04-26 | Merck Patent Gmbh | Chinazolinderivate |
| KR20140131971A (ko) | 2012-03-13 | 2014-11-14 | 레스피버트 리미티드 | 신규 약학 제제 |
| JO3279B1 (ar) * | 2013-03-15 | 2018-09-16 | Respivert Ltd | مشتقات 2-((4- امينو -3- (3- فلورو-5- هيدروكسي فينيل)-h1- بيرازولو [d-3,4] بيرمدين-1-يل )ميثيل )- 3- (2- تراي فلورو ميثيل ) بينزيل ) كوينازولين -4 (h3)- واحد واستخدامها كمثبطات فوسفواينوسيتايد 3- كاينيز |
| EP3236983B1 (en) * | 2014-12-24 | 2019-04-17 | Kither Biotech S.r.l. | Novel pi3k gamma inhibitor peptide for treatment of respiratory system diseases |
| CN106518809A (zh) * | 2015-09-15 | 2017-03-22 | 中国科学院上海药物研究所 | 丙酮酸脱氢酶激酶抑制剂及其应用 |
| CN111269231B (zh) * | 2018-12-04 | 2023-06-09 | 安徽中科拓苒药物科学研究有限公司 | 一种选择性PI3Kδ抑制剂及其用途 |
| CN114591335B (zh) * | 2021-03-29 | 2023-06-27 | 浙江大学 | 吲唑类化合物及其制备方法和应用 |
| CN115260164B (zh) * | 2021-05-01 | 2024-03-26 | 杭州星鳌生物科技有限公司 | 新型4(3h)-喹唑啉酮类似物的制备方法、结构组成及其在抗肿瘤药物中的应用 |
| WO2023206655A1 (zh) * | 2022-04-26 | 2023-11-02 | 安徽中科拓苒药物科学研究有限公司 | 一种PI3Kδ抑制剂及其用途 |
-
2007
- 2007-04-04 CN CNA2007800123688A patent/CN101448505A/zh active Pending
- 2007-04-04 CN CN200780012040.6A patent/CN101506211B/zh active Active
- 2007-04-04 SI SI200731298T patent/SI2004654T1/sl unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101506211A (zh) | 2009-08-12 |
| CN101448505A (zh) | 2009-06-03 |
| CN101506211B (zh) | 2013-05-22 |
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