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SG11202004231YA - Dopamine-β-hydroxylase inhibitors - Google Patents

Dopamine-β-hydroxylase inhibitors

Info

Publication number
SG11202004231YA
SG11202004231YA SG11202004231YA SG11202004231YA SG11202004231YA SG 11202004231Y A SG11202004231Y A SG 11202004231YA SG 11202004231Y A SG11202004231Y A SG 11202004231YA SG 11202004231Y A SG11202004231Y A SG 11202004231YA SG 11202004231Y A SG11202004231Y A SG 11202004231YA
Authority
SG
Singapore
Prior art keywords
dopamine
hydroxylase inhibitors
hydroxylase
inhibitors
Prior art date
Application number
SG11202004231YA
Inventor
Laszlo Erno Kiss
Alexander Beliaev
Tino Rossi
Pedro Nuno Leal Palma
Da Silva Patrício Manuel Vieira Araujo Soares
Rui Pinto
Francisco Cardona
Original Assignee
BIAL PORTELA & Cª S A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB1720189.8A external-priority patent/GB201720189D0/en
Priority claimed from GBGB1804439.6A external-priority patent/GB201804439D0/en
Application filed by BIAL PORTELA & Cª S A filed Critical BIAL PORTELA & Cª S A
Publication of SG11202004231YA publication Critical patent/SG11202004231YA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/05Isotopically modified compounds, e.g. labelled

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SG11202004231YA 2017-12-04 2018-11-30 Dopamine-β-hydroxylase inhibitors SG11202004231YA (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1720189.8A GB201720189D0 (en) 2017-12-04 2017-12-04 Dopamine-B-hydroxylase inhibitors
GBGB1804439.6A GB201804439D0 (en) 2018-03-20 2018-03-20 Dopamin-b-hydroxylase inhibitors
PCT/PT2018/050043 WO2019112457A1 (en) 2017-12-04 2018-11-30 Dopamine-β-hydroxylase inhibitors

Publications (1)

Publication Number Publication Date
SG11202004231YA true SG11202004231YA (en) 2020-06-29

Family

ID=65012066

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202004231YA SG11202004231YA (en) 2017-12-04 2018-11-30 Dopamine-β-hydroxylase inhibitors

Country Status (16)

Country Link
US (2) US11434242B2 (en)
EP (1) EP3720856A1 (en)
JP (1) JP7167155B2 (en)
KR (1) KR20200096584A (en)
CN (1) CN111479812A (en)
AU (1) AU2018379646A1 (en)
BR (1) BR112020010216A2 (en)
CA (1) CA3082337A1 (en)
CL (1) CL2020001461A1 (en)
IL (1) IL274550B2 (en)
MX (1) MX2020005864A (en)
PH (1) PH12020500542A1 (en)
RU (1) RU2020121820A (en)
SG (1) SG11202004231YA (en)
TW (1) TW201925193A (en)
WO (1) WO2019112457A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2020121820A (en) 2017-12-04 2022-01-10 БИАЛ - ПОРТЕЛА ЭНД Ка, С.А. DOPAMINE B-HYDROXYLASE INHIBITORS
GB201908044D0 (en) * 2019-06-05 2019-07-17 Bial Portela & Ca Sa Dopamine-B-Hydroxylase inhibitors
TW202528310A (en) * 2023-09-20 2025-07-16 美商深蘋果治療股份有限公司 Substituted amine compounds, compositions and methods of use
CN120383599A (en) * 2024-01-29 2025-07-29 上海深势唯思科技有限责任公司 Aryl heterocyclic Kv1.3 inhibitors and their preparation method and use

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3635982A (en) 1969-04-08 1972-01-18 American Home Prod Amino-substituted-quinoxalinyloxazolidines and -oxazines
FR2449689A1 (en) 1979-02-20 1980-09-19 Logeais Labor Jacques NOVEL CONDENSED PYRROLIDINE OR PIPERIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC APPLICATIONS
US4628059A (en) 1985-10-31 1986-12-09 Smithklein Beckman Corporation Dopamine-β-hydroxylase inhibitors
HUT76295A (en) 1994-04-26 1997-07-28 Syntex Inc Imidazolyl- and triazolyl-thion derivatives, pharmaceutical compositions containing them and process for producing them
US6482982B1 (en) 2001-03-09 2002-11-19 University Of Sciences Of Philadelphia Halogenated antituberculosis agents
IL143379A (en) * 2001-05-24 2013-11-28 Yissum Res Dev Co Antisense oligonucleotide against the r isophorm of human ache and uses thereof
US7125904B2 (en) * 2002-10-11 2006-10-24 Portela & C.A., S.A. Peripherally-selective inhibitors of dopamine-β-hydroxylase and method of their preparation
WO2008085008A1 (en) 2007-01-11 2008-07-17 Mogam Biotechnology Research Institute T-cell inhibiting compounds and their use for the treatment of t-cell-mediated diseases
GB0708818D0 (en) 2007-05-08 2007-06-13 Portela & Ca Sa Compounds
AU2008279091A1 (en) 2007-07-23 2009-01-29 Biotie Therapies, Inc Treatment of post-traumatic stress disorder
US8110578B2 (en) * 2008-10-27 2012-02-07 Signal Pharmaceuticals, Llc Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
CA2901577A1 (en) 2013-02-18 2014-08-21 The Scripps Research Institute Modulators of vasopressin receptors with therapeutic potential
JOP20190050A1 (en) * 2016-09-23 2019-03-20 Bial Portela & C? S A Blood-brain barrier-penetrant dopamine-?-hydroxylase inhibitors
RU2020121820A (en) 2017-12-04 2022-01-10 БИАЛ - ПОРТЕЛА ЭНД Ка, С.А. DOPAMINE B-HYDROXYLASE INHIBITORS

Also Published As

Publication number Publication date
RU2020121820A (en) 2022-01-10
KR20200096584A (en) 2020-08-12
US11434242B2 (en) 2022-09-06
US20230138795A1 (en) 2023-05-04
US20210171528A1 (en) 2021-06-10
TW201925193A (en) 2019-07-01
MX2020005864A (en) 2020-09-09
CL2020001461A1 (en) 2020-10-16
PH12020500542A1 (en) 2021-01-25
BR112020010216A2 (en) 2020-09-15
CN111479812A (en) 2020-07-31
JP7167155B2 (en) 2022-11-08
IL274550B2 (en) 2023-06-01
AU2018379646A1 (en) 2020-06-11
JP2021505568A (en) 2021-02-18
WO2019112457A1 (en) 2019-06-13
CA3082337A1 (en) 2019-06-13
IL274550A (en) 2020-06-30
EP3720856A1 (en) 2020-10-14

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