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SG11201405918XA - Estrogen receptor modulators and uses thereof - Google Patents

Estrogen receptor modulators and uses thereof

Info

Publication number
SG11201405918XA
SG11201405918XA SG11201405918XA SG11201405918XA SG11201405918XA SG 11201405918X A SG11201405918X A SG 11201405918XA SG 11201405918X A SG11201405918X A SG 11201405918XA SG 11201405918X A SG11201405918X A SG 11201405918XA SG 11201405918X A SG11201405918X A SG 11201405918XA
Authority
SG
Singapore
Prior art keywords
estrogen receptor
receptor modulators
modulators
estrogen
receptor
Prior art date
Application number
SG11201405918XA
Inventor
Nicholas D Smith
Steven P Govek
Mehmet Kahraman
Jackaline D Julien
Johnny Y Nagasawa
Karensa L Douglas
Celine Bonnefous
Andiliy G Lai
Original Assignee
Seragon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Seragon Pharmaceuticals Inc filed Critical Seragon Pharmaceuticals Inc
Publication of SG11201405918XA publication Critical patent/SG11201405918XA/en

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    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
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    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
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  • Psychiatry (AREA)
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  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
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SG11201405918XA 2012-03-20 2013-03-14 Estrogen receptor modulators and uses thereof SG11201405918XA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261613442P 2012-03-20 2012-03-20
PCT/US2013/031507 WO2013142266A1 (en) 2012-03-20 2013-03-14 Estrogen receptor modulators and uses thereof

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US (1) US9499538B2 (en)
EP (1) EP2828243B1 (en)
JP (1) JP6154887B2 (en)
KR (1) KR20140138296A (en)
CN (1) CN104220426B (en)
AU (1) AU2013235499A1 (en)
CA (1) CA2866891A1 (en)
CO (1) CO7170179A2 (en)
CR (1) CR20140479A (en)
EA (1) EA201491530A1 (en)
IL (1) IL234487A0 (en)
MX (1) MX2014011217A (en)
NZ (1) NZ630124A (en)
PE (1) PE20142461A1 (en)
PH (1) PH12014502095A1 (en)
SG (1) SG11201405918XA (en)
WO (1) WO2013142266A1 (en)

Families Citing this family (32)

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Publication number Priority date Publication date Assignee Title
JP6154887B2 (en) 2012-03-20 2017-06-28 セラゴン ファーマシューティカルズ,インク. Estrogen receptor modulators and uses thereof
US9586952B2 (en) 2013-03-14 2017-03-07 Genentech, Inc. Polycyclic estrogen receptor modulators and uses thereof
CN105142635B (en) 2013-03-15 2021-07-27 艾匹根生物技术有限公司 Heterocyclic compounds useful in the treatment of disease
MX2015016171A (en) 2013-06-19 2016-08-08 Seragon Pharmaceuticals Inc Azetidine estrogen receptor modulators and uses thereof.
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