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SG10201901676UA - Pyrazolothiazole compound and medicine comprising same - Google Patents

Pyrazolothiazole compound and medicine comprising same

Info

Publication number
SG10201901676UA
SG10201901676UA SG10201901676UA SG10201901676UA SG10201901676UA SG 10201901676U A SG10201901676U A SG 10201901676UA SG 10201901676U A SG10201901676U A SG 10201901676UA SG 10201901676U A SG10201901676U A SG 10201901676UA SG 10201901676U A SG10201901676U A SG 10201901676UA
Authority
SG
Singapore
Prior art keywords
compound
medicine
same
effect
pyrazolothiazole
Prior art date
Application number
SG10201901676UA
Inventor
Yoshinobu Shiba
Satoshi Akiyama
Original Assignee
Nippon Shinyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Shinyaku Co Ltd filed Critical Nippon Shinyaku Co Ltd
Publication of SG10201901676UA publication Critical patent/SG10201901676UA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/095Sulfur, selenium, or tellurium compounds, e.g. thiols
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/25Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids with polyoxyalkylated alcohols, e.g. esters of polyethylene glycol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

PYRAZOLOTHIAZOLE COMPOUND AND MEDICINE COMPRISING SAME The invention provides a pyrazolothiazolecompound compound of the formula [IJ, or a pharmaceutically 5 acceptable salt thereof: The compound of the invention has JAKI inhibitory activity, and thus, irr~unosuppressive effect, anti-inflammatory effect and anti-proliferative effect, and is useful in the 10 treatment of the diseases, for example, rheumatoid arthritis, inflammatory bowel disease, psoriasis and vasculitis, bronchial asthma, chronic obstructive pulmonary disease and eosinophilic sinusitis, nasal polyp. Figure for publication: None
SG10201901676UA 2014-09-02 2015-09-02 Pyrazolothiazole compound and medicine comprising same SG10201901676UA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2014177969 2014-09-02

Publications (1)

Publication Number Publication Date
SG10201901676UA true SG10201901676UA (en) 2019-03-28

Family

ID=55439874

Family Applications (2)

Application Number Title Priority Date Filing Date
SG10201901676UA SG10201901676UA (en) 2014-09-02 2015-09-02 Pyrazolothiazole compound and medicine comprising same
SG11201701447UA SG11201701447UA (en) 2014-09-02 2015-09-02 Pyrazolothiazole compound and medicine comprising same

Family Applications After (1)

Application Number Title Priority Date Filing Date
SG11201701447UA SG11201701447UA (en) 2014-09-02 2015-09-02 Pyrazolothiazole compound and medicine comprising same

Country Status (34)

Country Link
US (2) US9937176B2 (en)
EP (1) EP3190116B1 (en)
JP (1) JP6558372B2 (en)
KR (1) KR102294330B1 (en)
CN (1) CN107108653B (en)
AU (1) AU2015312886B2 (en)
BR (1) BR112017003800B1 (en)
CA (1) CA2959721C (en)
CL (1) CL2017000478A1 (en)
CO (1) CO2017002982A2 (en)
CY (1) CY1123320T1 (en)
DK (1) DK3190116T3 (en)
ES (1) ES2827243T3 (en)
HR (1) HRP20201382T1 (en)
HU (1) HUE050565T2 (en)
IL (1) IL250729B (en)
LT (1) LT3190116T (en)
MA (1) MA40605B1 (en)
MX (1) MX377926B (en)
MY (1) MY181814A (en)
NZ (1) NZ729494A (en)
PE (1) PE20170668A1 (en)
PH (1) PH12017500383B1 (en)
PL (1) PL3190116T3 (en)
PT (1) PT3190116T (en)
RS (1) RS60798B1 (en)
RU (1) RU2688660C2 (en)
SG (2) SG10201901676UA (en)
SI (1) SI3190116T1 (en)
SM (1) SMT202000503T1 (en)
TW (1) TWI679205B (en)
UA (1) UA121869C2 (en)
WO (1) WO2016035814A1 (en)
ZA (1) ZA201701492B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI679205B (en) * 2014-09-02 2019-12-11 日商日本新藥股份有限公司 Pyrazolothiazole compounds and medicine
TWI712604B (en) * 2016-03-01 2020-12-11 日商日本新藥股份有限公司 Crystal of compound with JAK inhibitory effect
WO2018225247A1 (en) 2017-06-09 2018-12-13 三菱電機株式会社 Passenger conveyor
EP4081199A4 (en) * 2019-12-23 2024-01-17 SRI International Lipoxygenase inhibitors
JP7742516B1 (en) * 2025-07-31 2025-09-19 日本新薬株式会社 Treatment for eosinophilic granulomatosis with polyangiitis

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PH25866A (en) * 1986-03-20 1991-12-02 Takeda Chemical Industries Ltd Sulfonylurea compounds and their herbicides
US5082847A (en) 1990-07-18 1992-01-21 Syntex (U.S.A.) Inc. Carbostyril compounds connected via an oxyalkyl group with a piperidine ring and having pharmaceutical utility
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Also Published As

Publication number Publication date
MX377926B (en) 2025-03-10
TW201613942A (en) 2016-04-16
KR20170044202A (en) 2017-04-24
US9937176B2 (en) 2018-04-10
SI3190116T1 (en) 2020-10-30
LT3190116T (en) 2020-11-10
EP3190116A1 (en) 2017-07-12
SG11201701447UA (en) 2017-03-30
PH12017500383A1 (en) 2017-07-17
IL250729A0 (en) 2017-04-30
US20170252341A1 (en) 2017-09-07
US20180092919A1 (en) 2018-04-05
SMT202000503T1 (en) 2020-11-10
US9999622B2 (en) 2018-06-19
WO2016035814A1 (en) 2016-03-10
DK3190116T3 (en) 2020-09-07
AU2015312886A1 (en) 2017-03-16
CN107108653B (en) 2019-04-09
UA121869C2 (en) 2020-08-10
JPWO2016035814A1 (en) 2017-06-22
CL2017000478A1 (en) 2017-11-10
CN107108653A (en) 2017-08-29
ES2827243T3 (en) 2021-05-20
RS60798B1 (en) 2020-10-30
MX2017002488A (en) 2017-05-23
CO2017002982A2 (en) 2017-07-11
AU2015312886B2 (en) 2020-02-06
PL3190116T3 (en) 2020-11-30
HRP20201382T1 (en) 2020-11-27
EP3190116A4 (en) 2018-04-04
BR112017003800A2 (en) 2017-11-28
KR102294330B1 (en) 2021-08-25
MY181814A (en) 2021-01-08
BR112017003800B1 (en) 2022-09-13
RU2688660C2 (en) 2019-05-22
CY1123320T1 (en) 2021-12-31
IL250729B (en) 2019-09-26
MA40605A (en) 2017-07-12
PE20170668A1 (en) 2017-06-06
EP3190116B1 (en) 2020-08-05
MA40605B1 (en) 2020-10-28
RU2017110535A3 (en) 2018-10-31
JP6558372B2 (en) 2019-08-14
CA2959721A1 (en) 2016-03-10
TWI679205B (en) 2019-12-11
PH12017500383B1 (en) 2019-11-20
NZ729494A (en) 2022-04-29
RU2017110535A (en) 2018-10-04
PT3190116T (en) 2020-09-04
HUE050565T2 (en) 2020-12-28
ZA201701492B (en) 2022-05-25
CA2959721C (en) 2022-10-25

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