[go: up one dir, main page]

SG10201506761XA - Deuterated analogs of pridopidine useful as dopaminergic stabilizers - Google Patents

Deuterated analogs of pridopidine useful as dopaminergic stabilizers

Info

Publication number
SG10201506761XA
SG10201506761XA SG10201506761XA SG10201506761XA SG10201506761XA SG 10201506761X A SG10201506761X A SG 10201506761XA SG 10201506761X A SG10201506761X A SG 10201506761XA SG 10201506761X A SG10201506761X A SG 10201506761XA SG 10201506761X A SG10201506761X A SG 10201506761XA
Authority
SG
Singapore
Prior art keywords
pridopidine
useful
deuterated analogs
dopaminergic stabilizers
dopaminergic
Prior art date
Application number
SG10201506761XA
Inventor
Clas Sonesson
Original Assignee
Teva Pharmaceuticals Int Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharmaceuticals Int Gmbh filed Critical Teva Pharmaceuticals Int Gmbh
Publication of SG10201506761XA publication Critical patent/SG10201506761XA/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/451Non condensed piperidines, e.g. piperocaine having a carbocyclic group directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B59/00Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
    • C07B59/002Heterocyclic compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/24Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by sulfur atoms to which a second hetero atom is attached
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/30Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom
    • C07D211/32Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by doubly bound oxygen or sulfur atoms or by two oxygen or sulfur atoms singly bound to the same carbon atom by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
SG10201506761XA 2010-09-03 2011-08-31 Deuterated analogs of pridopidine useful as dopaminergic stabilizers SG10201506761XA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA201070385 2010-09-03
US38085110P 2010-09-08 2010-09-08

Publications (1)

Publication Number Publication Date
SG10201506761XA true SG10201506761XA (en) 2015-10-29

Family

ID=44653278

Family Applications (2)

Application Number Title Priority Date Filing Date
SG2013014022A SG188298A1 (en) 2010-09-03 2011-08-31 Deuterated analogs of pridopidine useful as dopaminergic stabilizers
SG10201506761XA SG10201506761XA (en) 2010-09-03 2011-08-31 Deuterated analogs of pridopidine useful as dopaminergic stabilizers

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG2013014022A SG188298A1 (en) 2010-09-03 2011-08-31 Deuterated analogs of pridopidine useful as dopaminergic stabilizers

Country Status (18)

Country Link
US (5) US20130197031A1 (en)
EP (1) EP2611759A1 (en)
JP (1) JP2013536825A (en)
KR (1) KR20140008297A (en)
CN (1) CN103249697B (en)
AU (2) AU2011298382A1 (en)
BR (1) BR112013005125A2 (en)
CA (1) CA2810092A1 (en)
CL (1) CL2013000604A1 (en)
EA (1) EA201390332A1 (en)
IL (1) IL224776A (en)
MX (1) MX2013002453A (en)
NZ (1) NZ608120A (en)
PE (1) PE20140105A1 (en)
PH (1) PH12013500406A1 (en)
SG (2) SG188298A1 (en)
WO (1) WO2012028635A1 (en)
ZA (1) ZA201301902B (en)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE46117E1 (en) 1999-12-22 2016-08-23 Teva Pharmaceuticals International Gmbh Modulators of dopamine neurotransmission
JP5393654B2 (en) * 2007-04-12 2014-01-22 イヴァックス インテルナツィオナール ゲゼルシャフト ミット ベシュレンクテル ハフツンク N-oxide and / or di-N-oxide derivatives of dopamine receptor stabilizers / modulators exhibiting an improved cardiovascular side effect profile
EP2611759A1 (en) 2010-09-03 2013-07-10 Ivax International Gmbh Deuterated analogs of pridopidine useful as dopaminergic stabilizers
CN103958469B (en) 2011-09-07 2016-04-20 梯瓦制药国际有限责任公司 A kind of new Puli many determines hydrochloride polymorph form
UY34503A (en) 2011-12-08 2013-07-31 Ivax Int Gmbh PRIDOPIDINE BROMHYDRATE SALT
US20130267552A1 (en) 2012-04-04 2013-10-10 IVAX International GmbH Pharmaceutical compositions for combination therapy
IN2015DN01662A (en) 2012-09-18 2015-07-03 Auspex Pharmaceuticals Inc
WO2014205229A1 (en) 2013-06-21 2014-12-24 IVAX International GmbH Use of high dose pridopidine for treating huntington's disease
US11090297B2 (en) 2013-06-21 2021-08-17 Prilenia Neurotherapeutics Ltd. Pridopidine for treating huntington's disease
US10166183B2 (en) 2014-02-07 2019-01-01 Auspex Pharmaceuticals, Inc. Pharmaceutical formulations
TW201613859A (en) 2014-06-30 2016-04-16 Teva Pharma Analogs of PRIDOPIDINE, their preparation and use
US9796673B2 (en) 2014-12-22 2017-10-24 Teva Pharmaceuticals International Gmbh L-tartrate salt of pridopidine
WO2016138130A1 (en) 2015-02-25 2016-09-01 Teva Pharmaceuticals International Gmbh Use of pridopidine to improve cognitive function and for treating alzheimer's disease
US11471449B2 (en) 2015-02-25 2022-10-18 Prilenia Neurotherapeutics Ltd. Use of pridopidine to improve cognitive function and for treating Alzheimer's disease
JP6932641B2 (en) 2015-03-06 2021-09-08 オースペックス ファーマシューティカルズ インコーポレイテッド Methods for the treatment of abnormal involuntary movement disorders
AR105434A1 (en) 2015-07-22 2017-10-04 Teva Pharmaceuticals Int Gmbh PROCESS TO PREPARE PRIDOPIDINE
CA3015512C (en) 2016-02-24 2024-01-16 Teva Pharmaceuticals International Gmbh Treatment of neurodegenerative eye disease using pridopidine
CA3035092C (en) 2016-08-24 2022-05-31 Prilenia Therapeutics Development Ltd. Use of pridopidine for treating functional decline
CA3035099C (en) 2016-08-24 2023-01-17 Prilenia Therapeutics Development Ltd. Use of pridopidine for treating dystonias
WO2018053287A1 (en) 2016-09-15 2018-03-22 Teva Pharmaceuticals International Gmbh Use of pridopidine for the treatment of anxiety and depression
US12102627B2 (en) 2016-09-16 2024-10-01 Prilenia Neurotherapeutics Ltd. Use of pridopidine for treating rett syndrome
DK4005570T3 (en) 2016-09-16 2024-08-19 Prilenia Neurotherapeutics Ltd PRIDOPIDINE FOR USE IN THE TREATMENT OF REET'S SYNDROME
AU2018210145B2 (en) 2017-01-20 2023-06-29 Agency For Science, Technology And Research Use of pridopidine for the treatment of fragile X syndrome
US10459055B2 (en) * 2017-04-07 2019-10-29 Case Western Reserve University System and method for reduced field of view MR fingerprinting for parametric mapping
BR112020003119A2 (en) 2017-08-14 2020-10-13 Prilenia Neurotherapeutics Ltd. method of treating amyotrophic lateral sclerosis with pridopidine
EP3675830A1 (en) 2017-08-30 2020-07-08 Prilenia Neurotherapeutics Ltd. High concentration dosage forms of pridopidine
US12036213B2 (en) 2017-09-08 2024-07-16 Prilenia Neurotherapeutics Ltd. Pridopidine for treating drug induced dyskinesias
EP3678664A1 (en) 2017-09-08 2020-07-15 Prilenia Neurotherapeutics Ltd. Pridopidine for treating drug induced dyskinesias
EP3920924A4 (en) 2019-02-04 2022-11-16 Prilenia Neurotherapeutics Ltd. Low dose pridopidine for parkinson's disease and other diseases associated with parkinsonism
MX2022010006A (en) 2020-02-13 2022-09-19 Prilenia Neurotherapeutics Ltd Combination therapy for treating amyotrophic lateral using pridopidine and another active agent.
JP7603713B2 (en) 2020-05-04 2024-12-20 プリレニア ニューロセラピューティクス リミテッド Treatment of viral infections, diseases, or disorders using selective S1R agonists
AU2021275863A1 (en) * 2020-05-20 2023-02-02 Certego Therapeutics Inc. Ring deuterated gaboxadol and its use for the treatment of psychiatric disorders
WO2021232096A1 (en) 2020-05-20 2021-11-25 Nthalmic Holding Pty Ltd Methods and apparatus to manage meibomian gland deficiencies

Family Cites Families (46)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6221335B1 (en) * 1994-03-25 2001-04-24 Isotechnika, Inc. Method of using deuterated calcium channel blockers
US6440710B1 (en) * 1998-12-10 2002-08-27 The Scripps Research Institute Antibody-catalyzed deuteration, tritiation, dedeuteration or detritiation of carbonyl compounds
PT1104760E (en) * 1999-12-03 2003-06-30 Pfizer Prod Inc SULFAMOYL-HETEROARILPIRAZOLE COMPOUNDS AS ANALGESIC AND ANTI-INFLAMMATORY AGENTS
SE9904724D0 (en) 1999-12-22 1999-12-22 Carlsson A Research Ab New modulators of dopamine neurotransmission I
USRE46117E1 (en) 1999-12-22 2016-08-23 Teva Pharmaceuticals International Gmbh Modulators of dopamine neurotransmission
SE9904723D0 (en) 1999-12-22 1999-12-22 Carlsson A Research Ab New modulators of dopamine neurotransmission II
DE10123129A1 (en) * 2001-05-02 2002-11-14 Berolina Drug Dev Ab Svedala Deuterated 3-piperidinopropiophenones and medicinal products containing these compounds
TW200413273A (en) * 2002-11-15 2004-08-01 Wako Pure Chem Ind Ltd Heavy hydrogenation method of heterocyclic rings
US7004629B2 (en) 2003-07-26 2006-02-28 Arthur Joseph Shrader Method and apparatus for hanging a resealable bag
ES2346452T3 (en) 2004-06-08 2010-10-15 Nsab, Filial Af Neurosearch Sweden Ab, Sverige NEW DISABLED PHENYLPIPERIDINS / PIPERAZINS USED AS MODULATORS OF THE DOPAMINE NEUROTRANSMISSION.
ES2659577T3 (en) 2004-10-13 2018-03-16 Teva Pharmaceuticals International Gmbh Process for the synthesis of 4- (3-methanesulfonylphenyl) -1-N-propyl-piperidine
CN101309917B (en) * 2005-10-06 2013-09-11 奥斯拜客斯制药有限公司 Deuterated inhibitor of gastric H+, K+-ATPase with enhanced therapeutic properties
SE529246C2 (en) 2005-10-13 2007-06-12 Neurosearch Sweden Ab New disubstituted phenyl-piperidines as modulators of dopamine neurotransmission
CN101360742A (en) * 2005-11-14 2009-02-04 奥斯拜客斯制药有限公司 Substituted phenylpiperidines with serotonin-derived activity and enhanced therapeutic properties
CA2629514A1 (en) 2005-11-14 2007-05-24 Auspex Pharmaceuticals, Inc. Substituted phenylpiperidines with serotoninergic activity and enhanced therapeutic properties
US7750168B2 (en) * 2006-02-10 2010-07-06 Sigma-Aldrich Co. Stabilized deuteroborane-tetrahydrofuran complex
JP5393654B2 (en) 2007-04-12 2014-01-22 イヴァックス インテルナツィオナール ゲゼルシャフト ミット ベシュレンクテル ハフツンク N-oxide and / or di-N-oxide derivatives of dopamine receptor stabilizers / modulators exhibiting an improved cardiovascular side effect profile
US20100197712A1 (en) * 2007-06-18 2010-08-05 Arvid Carlsson Use of dopamine stabilizers
US8288414B2 (en) * 2007-09-12 2012-10-16 Deuteria Pharmaceuticals, Inc. Deuterium-enriched lenalidomide
US20110206782A1 (en) * 2010-02-24 2011-08-25 Auspex Pharmaceuticals, Inc. Piperidine modulators of dopamine receptor
WO2011107583A1 (en) * 2010-03-04 2011-09-09 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Substituted 4-phenyl-n-alkyl-piperidines for preventing onset or slowing progression of neurodegenerative disorders
EP2611759A1 (en) * 2010-09-03 2013-07-10 Ivax International Gmbh Deuterated analogs of pridopidine useful as dopaminergic stabilizers
CN103958469B (en) 2011-09-07 2016-04-20 梯瓦制药国际有限责任公司 A kind of new Puli many determines hydrochloride polymorph form
UY34503A (en) 2011-12-08 2013-07-31 Ivax Int Gmbh PRIDOPIDINE BROMHYDRATE SALT
US20130267552A1 (en) 2012-04-04 2013-10-10 IVAX International GmbH Pharmaceutical compositions for combination therapy
WO2014052935A2 (en) 2012-09-27 2014-04-03 Teva Pharmaceutical Industries Ltd. Combination of rasagiline and pridopidine for treating neurodegenerative disorders, in particular huntington's disease
BR112015006623A2 (en) 2012-09-27 2017-07-04 Teva Pharma laquinimod and pridopidine for the treatment of neurodegenerative diseases
WO2014205229A1 (en) 2013-06-21 2014-12-24 IVAX International GmbH Use of high dose pridopidine for treating huntington's disease
US11090297B2 (en) 2013-06-21 2021-08-17 Prilenia Neurotherapeutics Ltd. Pridopidine for treating huntington's disease
MX377576B (en) 2014-01-22 2025-03-04 Prilenia Neurotherapeutics Ltd MODIFIED-RELEASE PRIDOPIDINE FORMULATIONS.
TW201613859A (en) 2014-06-30 2016-04-16 Teva Pharma Analogs of PRIDOPIDINE, their preparation and use
US9796673B2 (en) 2014-12-22 2017-10-24 Teva Pharmaceuticals International Gmbh L-tartrate salt of pridopidine
WO2016138130A1 (en) 2015-02-25 2016-09-01 Teva Pharmaceuticals International Gmbh Use of pridopidine to improve cognitive function and for treating alzheimer's disease
AR105434A1 (en) 2015-07-22 2017-10-04 Teva Pharmaceuticals Int Gmbh PROCESS TO PREPARE PRIDOPIDINE
WO2017015615A1 (en) 2015-07-22 2017-01-26 Teva Pharmaceuticals International Gmbh Pridopidine base formulations and their use
US20170026730A1 (en) 2015-07-23 2017-01-26 Knowles Electronics, Llc Microphone with temperature sensor
CA3015512C (en) 2016-02-24 2024-01-16 Teva Pharmaceuticals International Gmbh Treatment of neurodegenerative eye disease using pridopidine
CA3035099C (en) 2016-08-24 2023-01-17 Prilenia Therapeutics Development Ltd. Use of pridopidine for treating dystonias
CA3035092C (en) 2016-08-24 2022-05-31 Prilenia Therapeutics Development Ltd. Use of pridopidine for treating functional decline
WO2018053287A1 (en) 2016-09-15 2018-03-22 Teva Pharmaceuticals International Gmbh Use of pridopidine for the treatment of anxiety and depression
WO2018053230A1 (en) 2016-09-16 2018-03-22 Cargill, Incorporated Genetically modified lactate-consuming yeasts and fermentation processes using such genetically modified yeasts
WO2018053275A1 (en) 2016-09-16 2018-03-22 Teva Pharmaceuticals International Gmbh Use of pridopidine for the treatment of familial dysautonomia
AU2018210145B2 (en) 2017-01-20 2023-06-29 Agency For Science, Technology And Research Use of pridopidine for the treatment of fragile X syndrome
BR112020003119A2 (en) 2017-08-14 2020-10-13 Prilenia Neurotherapeutics Ltd. method of treating amyotrophic lateral sclerosis with pridopidine
NL2019473B1 (en) 2017-09-01 2019-03-11 Isobionics B V Terpene Synthase producing patchoulol and elemol, and preferably also pogostol
EP3678664A1 (en) 2017-09-08 2020-07-15 Prilenia Neurotherapeutics Ltd. Pridopidine for treating drug induced dyskinesias

Also Published As

Publication number Publication date
PE20140105A1 (en) 2014-02-14
EA201390332A1 (en) 2013-08-30
JP2013536825A (en) 2013-09-26
CA2810092A1 (en) 2012-03-08
US20130197031A1 (en) 2013-08-01
NZ608120A (en) 2014-12-24
US20190015401A1 (en) 2019-01-17
CN103249697A (en) 2013-08-14
PH12013500406A1 (en) 2019-07-17
SG188298A1 (en) 2013-04-30
IL224776A (en) 2017-07-31
CL2013000604A1 (en) 2013-11-15
US20180235950A1 (en) 2018-08-23
BR112013005125A2 (en) 2016-08-16
US10799492B2 (en) 2020-10-13
US20160095847A1 (en) 2016-04-07
CN103249697B (en) 2016-06-15
ZA201301902B (en) 2014-05-28
WO2012028635A1 (en) 2012-03-08
EP2611759A1 (en) 2013-07-10
AU2016250390A1 (en) 2016-11-10
AU2011298382A1 (en) 2013-05-02
KR20140008297A (en) 2014-01-21
MX2013002453A (en) 2013-08-01
US20160166559A1 (en) 2016-06-16

Similar Documents

Publication Publication Date Title
ZA201301902B (en) Deuterated analogs of pridopidine useful as dopaminergic stabilizers
EP2655392A4 (en) Cyclic nucleotide analogs
AP3584A (en) Substituted nucleotide analogs
HUE047354T2 (en) Deuterated derivatives of ivacaftor
PT2709986T (en) Deuterated derivatives of ivacaftor
IL227754A0 (en) 4-hydroxybutyric acid deuterated analogs
EP2828278A4 (en) Methods of preparing substituted nucleotide analogs
IL225617A0 (en) Cyclosporin analogs
ZA201309245B (en) Novel fluoroergoline analogs
IL216632A0 (en) Wearable utility instrument assembly
EP2611451A4 (en) Design of oligonucleotide analogs as therapeutic agents
PL2658531T3 (en) Use of glutamide stabilizers
GB201311220D0 (en) Improved structure of shoe
IL225616A0 (en) Cyclosporin analogs
ZA201404034B (en) Anhydrous antiperspirant compositions
TWM388611U (en) Improved structure of light-emitting device
IL228985A0 (en) Diazonamide analogs
HK1187036A (en) Deuterated analogs of pridopidine useful as dopaminergic stabilizers
TWM400766U (en) Improved structure of insole
TWM387196U (en) Improved structure of LED
TWM402983U (en) Improved structure of LED
TWM390954U (en) Structure of light-emitting yarn
TWM401317U (en) Improved multi-weave structure of socks
TWM400768U (en) High heel structure
TWM388315U (en) Improved structure of hemoclip