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SE8902076D0 - Derivatives of quinoline-3-carboxanilide - Google Patents

Derivatives of quinoline-3-carboxanilide

Info

Publication number
SE8902076D0
SE8902076D0 SE8902076A SE8902076A SE8902076D0 SE 8902076 D0 SE8902076 D0 SE 8902076D0 SE 8902076 A SE8902076 A SE 8902076A SE 8902076 A SE8902076 A SE 8902076A SE 8902076 D0 SE8902076 D0 SE 8902076D0
Authority
SE
Sweden
Prior art keywords
group
carboxanilide
quinoline
derivatives
methoxy
Prior art date
Application number
SE8902076A
Other languages
English (en)
Inventor
P-O Gunnarsson
K Strandgaarden
K Johansson
Original Assignee
Pharmacia Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Ab filed Critical Pharmacia Ab
Priority to SE8902076A priority Critical patent/SE8902076D0/sv
Publication of SE8902076D0 publication Critical patent/SE8902076D0/sv
Priority to NZ233860A priority patent/NZ233860A/en
Priority to JP2509778A priority patent/JPH04500373A/ja
Priority to DE69022368T priority patent/DE69022368T2/de
Priority to EP90909805A priority patent/EP0429627B1/en
Priority to PCT/SE1990/000375 priority patent/WO1990015052A1/en
Priority to AU59234/90A priority patent/AU648026B2/en
Priority to ES90909805T priority patent/ES2077071T3/es
Priority to AT90909805T priority patent/ATE127791T1/de
Priority to DK90909805.5T priority patent/DK0429627T3/da
Priority to CA002033211A priority patent/CA2033211A1/en
Priority to US08/102,393 priority patent/US5310913A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cosmetics (AREA)
  • Quinoline Compounds (AREA)
SE8902076A 1989-06-09 1989-06-09 Derivatives of quinoline-3-carboxanilide SE8902076D0 (sv)

Priority Applications (12)

Application Number Priority Date Filing Date Title
SE8902076A SE8902076D0 (sv) 1989-06-09 1989-06-09 Derivatives of quinoline-3-carboxanilide
NZ233860A NZ233860A (en) 1989-06-09 1990-05-30 Substituted quinoline derivatives
CA002033211A CA2033211A1 (en) 1989-06-09 1990-05-31 Derivatives of quinoline-3-carboxanilide
EP90909805A EP0429627B1 (en) 1989-06-09 1990-05-31 Derivatives of quinoline-3-carboxanilide
DE69022368T DE69022368T2 (de) 1989-06-09 1990-05-31 Quinolin-3-carboxanilid-derivate.
JP2509778A JPH04500373A (ja) 1989-06-09 1990-05-31 キノリン―3―カルボキシアニリドの誘導体
PCT/SE1990/000375 WO1990015052A1 (en) 1989-06-09 1990-05-31 Derivatives of quinoline-3-carboxanilide
AU59234/90A AU648026B2 (en) 1989-06-09 1990-05-31 Derivatives of quinoline-3-carboxanilide
ES90909805T ES2077071T3 (es) 1989-06-09 1990-05-31 Derivados de quinolin-3-carboxamida.
AT90909805T ATE127791T1 (de) 1989-06-09 1990-05-31 Quinolin-3-carboxanilid-derivate.
DK90909805.5T DK0429627T3 (da) 1989-06-09 1990-05-31 Derivater af quinolin-3-carboxanilider
US08/102,393 US5310913A (en) 1989-06-09 1993-08-05 Derivatives of quinoline-3-carboxanilide

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE8902076A SE8902076D0 (sv) 1989-06-09 1989-06-09 Derivatives of quinoline-3-carboxanilide

Publications (1)

Publication Number Publication Date
SE8902076D0 true SE8902076D0 (sv) 1989-06-09

Family

ID=20376220

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8902076A SE8902076D0 (sv) 1989-06-09 1989-06-09 Derivatives of quinoline-3-carboxanilide

Country Status (11)

Country Link
EP (1) EP0429627B1 (sv)
JP (1) JPH04500373A (sv)
AT (1) ATE127791T1 (sv)
AU (1) AU648026B2 (sv)
CA (1) CA2033211A1 (sv)
DE (1) DE69022368T2 (sv)
DK (1) DK0429627T3 (sv)
ES (1) ES2077071T3 (sv)
NZ (1) NZ233860A (sv)
SE (1) SE8902076D0 (sv)
WO (1) WO1990015052A1 (sv)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5310913A (en) * 1989-06-09 1994-05-10 Kabi Pharmacia Aktiebolag Derivatives of quinoline-3-carboxanilide
US5268378A (en) * 1990-05-31 1993-12-07 Merck Sharp & Dohme, Limited Dioxo-tetrahydroquinoline derivatives
GB9108547D0 (en) * 1991-04-22 1991-06-05 Fujisawa Pharmaceutical Co Quinoline derivatives
DE4138820A1 (de) * 1991-11-26 1993-05-27 Basf Ag Chinolin-3-carbonsaeureamide, deren herstellung und verwendung
GB9311562D0 (en) * 1993-06-04 1993-07-21 Fujisawa Pharmaceutical Co Heterocyclic derivatives
GB9404378D0 (en) * 1994-03-07 1994-04-20 Fujisawa Pharmaceutical Co Quinoline derivatives
SE9400809D0 (sv) * 1994-03-10 1994-03-10 Pharmacia Ab New use of quinoline-3-carboxamide compounds
SE9400810D0 (sv) * 1994-03-10 1994-03-10 Pharmacia Ab New use of Quinoline-3-carboxamide compounds
KR20000022040A (ko) * 1996-06-20 2000-04-25 보오드 오브 리젠츠, 더 유니버시티 오브 텍사스 시스템 약학적 활성 제제를 제공하기 위한 화합물, 방법 및 그의 용도
JP2000256323A (ja) 1999-01-08 2000-09-19 Japan Tobacco Inc 2−オキソキノリン化合物及びその医薬用途
RU2162326C1 (ru) * 1999-11-12 2001-01-27 Научно-исследовательский институт психического здоровья Томского научного центра СО РАМН Средство, стимулирующее фагоцитоз
US8314124B2 (en) 2004-02-06 2012-11-20 Active Biotech Ab Crystalline salts of quinoline compounds and methods for preparing them
SE0400235D0 (sv) 2004-02-06 2004-02-06 Active Biotech Ab New composition containing quinoline compounds
KR101440982B1 (ko) 2005-10-19 2014-09-17 테바 파마슈티컬 인더스트리즈 리미티드 라퀴니모드 나트륨의 결정 및 이의 제조방법
US7989473B2 (en) 2006-06-12 2011-08-02 Teva Pharmaceutical Industries, Ltd. Stable laquinimod preparations
US8178127B2 (en) 2007-12-20 2012-05-15 Teva Pharmaceuticals Industries, Ltd. Stable laquinimod preparations
JP2012502038A (ja) 2008-09-03 2012-01-26 テバ ファーマシューティカル インダストリーズ リミティド 免疫機能の2−オキソ−1,2−ジヒドロ−キノリンモジュレーター
JP6215238B2 (ja) * 2012-02-16 2017-10-18 テバ ファーマシューティカル インダストリーズ リミティド N−エチル−n−フェニル−1,2−ジヒドロ−4,5−ジ−ヒドロキシ−1−メチル−2−オキソ−3−キノリンカルボキサミド、その製剤、および使用
TW201350467A (zh) 2012-05-08 2013-12-16 Teva Pharma N-乙基-4-羥基-1-甲基-5-(甲基(2,3,4,5,6-五羥基己基)胺基)-2-側氧-n-苯基-1,2-二氫喹啉-3-甲醯胺
HK1215210A1 (zh) 2012-11-07 2016-08-19 Teva Pharmaceutical Industries Ltd. 拉喹莫德胺盐
US9233927B2 (en) 2013-03-14 2016-01-12 Teva Pharmaceutical Industries, Ltd. Crystals of laquinimod sodium and improved process for the manufacture thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE52670B1 (en) * 1981-03-03 1988-01-20 Leo Ab Heterocyclic carboxamides,compositions containing such compounds,and processes for their preparation
DE3420116A1 (de) * 1984-05-30 1985-12-05 Bayer Ag, 5090 Leverkusen Immunstimulierende mittel
DE3906365A1 (de) * 1988-07-15 1990-01-18 Bayer Ag 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe

Also Published As

Publication number Publication date
JPH04500373A (ja) 1992-01-23
ES2077071T3 (es) 1995-11-16
CA2033211A1 (en) 1990-12-10
EP0429627B1 (en) 1995-09-13
AU5923490A (en) 1991-01-07
AU648026B2 (en) 1994-04-14
WO1990015052A1 (en) 1990-12-13
EP0429627A1 (en) 1991-06-05
NZ233860A (en) 1991-04-26
DE69022368D1 (de) 1995-10-19
DE69022368T2 (de) 1996-05-02
DK0429627T3 (da) 1995-11-20
ATE127791T1 (de) 1995-09-15

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