SE0100374D0 - Novel compositions of potassium channel openers and protein kinase c inhibitors and use thereof - Google Patents
Novel compositions of potassium channel openers and protein kinase c inhibitors and use thereofInfo
- Publication number
- SE0100374D0 SE0100374D0 SE0100374A SE0100374A SE0100374D0 SE 0100374 D0 SE0100374 D0 SE 0100374D0 SE 0100374 A SE0100374 A SE 0100374A SE 0100374 A SE0100374 A SE 0100374A SE 0100374 D0 SE0100374 D0 SE 0100374D0
- Authority
- SE
- Sweden
- Prior art keywords
- novel compositions
- inhibitors
- protein kinase
- potassium channel
- channel openers
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 3
- 229940127315 Potassium Channel Openers Drugs 0.000 title abstract 2
- 229940123924 Protein kinase C inhibitor Drugs 0.000 title abstract 2
- 239000003881 protein kinase C inhibitor Substances 0.000 title abstract 2
- XFZJEEAOWLFHDH-NFJBMHMQSA-N procyanidin B2 Chemical compound C1([C@@H]2[C@H](O)[C@H](C3=C(O)C=C(O)C=C3O2)C=2C(O)=CC(O)=C3C[C@H]([C@H](OC3=2)C=2C=C(O)C(O)=CC=2)O)=CC=C(O)C(O)=C1 XFZJEEAOWLFHDH-NFJBMHMQSA-N 0.000 abstract 2
- XFZJEEAOWLFHDH-UHFFFAOYSA-N (2R,2'R,3R,3'R,4R)-3,3',4',5,7-Pentahydroxyflavan(48)-3,3',4',5,7-pentahydroxyflavan Natural products C=12OC(C=3C=C(O)C(O)=CC=3)C(O)CC2=C(O)C=C(O)C=1C(C1=C(O)C=C(O)C=C1O1)C(O)C1C1=CC=C(O)C(O)=C1 XFZJEEAOWLFHDH-UHFFFAOYSA-N 0.000 abstract 1
- ZFMITUMMTDLWHR-UHFFFAOYSA-N Minoxidil Chemical compound NC1=[N+]([O-])C(N)=CC(N2CCCCC2)=N1 ZFMITUMMTDLWHR-UHFFFAOYSA-N 0.000 abstract 1
- 229920002350 Procyanidin B2 Polymers 0.000 abstract 1
- 229960003632 minoxidil Drugs 0.000 abstract 1
- 230000003658 preventing hair loss Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q7/00—Preparations for affecting hair growth
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/4953—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom containing pyrimidine ring derivatives, e.g. minoxidil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/4973—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom
- A61K8/498—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom having 6-membered rings or their condensed derivatives, e.g. coumarin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/74—Biological properties of particular ingredients
- A61K2800/78—Enzyme modulators, e.g. Enzyme agonists
- A61K2800/782—Enzyme inhibitors; Enzyme antagonists
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Birds (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Cosmetics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0100374A SE0100374D0 (sv) | 2001-02-07 | 2001-02-07 | Novel compositions of potassium channel openers and protein kinase c inhibitors and use thereof |
| EP02715944A EP1357974A1 (fr) | 2001-02-07 | 2002-01-23 | Nouvelles compositions d'activateurs de canaux potassiques et inhibiteurs de la proteine kinase c et leur utilisation |
| JP2002562427A JP2004518701A (ja) | 2001-02-07 | 2002-01-23 | カリウムチャネル開口薬およびプロテインキナーゼｃ阻害薬の新規な組成物ならびにそれらの使用 |
| PCT/SE2002/000105 WO2002062422A1 (fr) | 2001-02-07 | 2002-01-23 | Nouvelles compositions d'activateurs de canaux potassiques et inhibiteurs de la proteine kinase c et leur utilisation |
| US10/059,658 US20020137692A1 (en) | 2001-02-07 | 2002-01-29 | Novel compositions of potassium channel openers and protein kinase C inhibitors and use thereof |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| SE0100374A SE0100374D0 (sv) | 2001-02-07 | 2001-02-07 | Novel compositions of potassium channel openers and protein kinase c inhibitors and use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SE0100374D0 true SE0100374D0 (sv) | 2001-02-07 |
Family
ID=20282870
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE0100374A SE0100374D0 (sv) | 2001-02-07 | 2001-02-07 | Novel compositions of potassium channel openers and protein kinase c inhibitors and use thereof |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP1357974A1 (fr) |
| JP (1) | JP2004518701A (fr) |
| SE (1) | SE0100374D0 (fr) |
| WO (1) | WO2002062422A1 (fr) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20070208087A1 (en) | 2001-11-02 | 2007-09-06 | Sanders Virginia J | Compounds, compositions and methods for the treatment of inflammatory diseases |
| CA2486869C (fr) | 2002-05-31 | 2011-09-13 | Proteotech, Inc. | Composes, compositions et procedes de traitement de maladies amyloides et de synucleinopathies, notamment de la maladie d'alzheimer, du diabete de type 2 et de la maladie de parkinson |
| EP1554270A2 (fr) * | 2002-10-11 | 2005-07-20 | Proteotech, Inc. | Isolation, purification et synthese de procyanidine b2, et ses utilisations |
| EP1921076A1 (fr) * | 2002-10-11 | 2008-05-14 | Proteotech Inc. | synthèse de procyanidine B2 |
| WO2010036947A2 (fr) * | 2008-09-27 | 2010-04-01 | Jina Pharmaceuticals, Inc. | Préparations pharmaceutiques à base de lipide(s) à usage oral et topique, leurs compositions, procédés et utilisations |
| CN117205216A (zh) * | 2022-05-06 | 2023-12-12 | 南京思聚生物医药有限公司 | 一种局部作用的雄激素受体拮抗剂与米诺地尔的组合物及其应用 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4596812A (en) * | 1976-05-24 | 1986-06-24 | The Upjohn Company | Methods and solutions for treating male pattern alopecia |
| JP3004718B2 (ja) * | 1990-08-10 | 2000-01-31 | ファルマシア・アンド・アップジョン・カンパニー | カリウムチャネルオープナーおよび５α―レダクターゼ抑制剤を用いる育毛刺激 |
| AU686691B2 (en) * | 1994-01-12 | 1998-02-12 | F. Hoffmann-La Roche Ag | Novel azepanes and homologs thereof |
| WO1996000561A1 (fr) * | 1994-06-30 | 1996-01-11 | Kyowa Hakko Kogyo Co., Ltd. | Produit stimulant la pousse des cheveux |
| TW339325B (en) * | 1995-07-05 | 1998-09-01 | Hoffmann La Roche | Novel azepane derivatives, process for the preparation thereof and pharmaceutical composition containing the same |
| KR100499190B1 (ko) * | 1996-03-29 | 2006-04-17 | 교와 핫꼬 고교 가부시끼가이샤 | 육모제 |
-
2001
- 2001-02-07 SE SE0100374A patent/SE0100374D0/xx unknown
-
2002
- 2002-01-23 EP EP02715944A patent/EP1357974A1/fr not_active Withdrawn
- 2002-01-23 JP JP2002562427A patent/JP2004518701A/ja not_active Withdrawn
- 2002-01-23 WO PCT/SE2002/000105 patent/WO2002062422A1/fr not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002062422A1 (fr) | 2002-08-15 |
| EP1357974A1 (fr) | 2003-11-05 |
| JP2004518701A (ja) | 2004-06-24 |
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