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RU2019125378A3 - - Google Patents

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Publication number
RU2019125378A3
RU2019125378A3 RU2019125378A RU2019125378A RU2019125378A3 RU 2019125378 A3 RU2019125378 A3 RU 2019125378A3 RU 2019125378 A RU2019125378 A RU 2019125378A RU 2019125378 A RU2019125378 A RU 2019125378A RU 2019125378 A3 RU2019125378 A3 RU 2019125378A3
Authority
RU
Russia
Application number
RU2019125378A
Other versions
RU2019125378A (ru
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP17156518.7A external-priority patent/EP3363802B1/en
Application filed filed Critical
Publication of RU2019125378A3 publication Critical patent/RU2019125378A3/ru
Publication of RU2019125378A publication Critical patent/RU2019125378A/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5365Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
RU2019125378A 2017-02-16 2018-01-25 Кристаллические формы каботегравира натрия RU2019125378A (ru)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP17156518.7 2017-02-16
EP17156518.7A EP3363802B1 (en) 2017-02-16 2017-02-16 Crystalline form of cabotegravir sodium
EP17161414.2 2017-03-16
EP17161414 2017-03-16
PCT/EP2018/051819 WO2018149608A1 (en) 2017-02-16 2018-01-25 Crystalline forms of cabotegravir sodium

Publications (2)

Publication Number Publication Date
RU2019125378A3 true RU2019125378A3 (ru) 2021-03-16
RU2019125378A RU2019125378A (ru) 2021-03-16

Family

ID=61168064

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2019125378A RU2019125378A (ru) 2017-02-16 2018-01-25 Кристаллические формы каботегравира натрия

Country Status (8)

Country Link
US (3) US11040986B2 (ru)
EP (1) EP3583107B1 (ru)
CN (1) CN110582504A (ru)
AU (2) AU2018221379B2 (ru)
CA (1) CA3053202C (ru)
MX (2) MX388699B (ru)
RU (1) RU2019125378A (ru)
WO (1) WO2018149608A1 (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110582504A (zh) * 2017-02-16 2019-12-17 桑多斯股份公司 卡博特韦钠的晶形
WO2023175386A2 (en) * 2021-10-08 2023-09-21 Laurus Labs Limited Processes for preparation of cabotegravir or its pharmaceutically acceptable salts thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20160757T1 (hr) 2004-04-19 2016-08-12 Krka, Tovarna Zdravil, D.D., Novo Mesto Postupak za proizvodnju polimorfnog oblika i od klopidogrel-vodik-sulfata
CN101212903B (zh) * 2005-04-28 2013-07-24 史密丝克莱恩比彻姆公司 具有hiv整合酶抑制活性的多环氨基甲酰基吡啶酮衍生物
JP4295353B2 (ja) 2005-04-28 2009-07-15 スミスクライン ビーチャム コーポレーション Hivインテグラーゼ阻害活性を有する多環性カルバモイルピリドン誘導体
EP3210603A1 (en) 2008-12-11 2017-08-30 Shionogi & Co., Ltd Synthesis of carbamoylpyridone hiv integrase inhibitors and intermediates
TWI582097B (zh) 2010-03-23 2017-05-11 Viiv醫療保健公司 製備胺甲醯吡啶酮衍生物及中間體之方法
WO2015139591A1 (zh) 2014-03-19 2015-09-24 杭州普晒医药科技有限公司 德罗格韦钠盐的晶型及其制备方法
ZA201503540B (en) 2014-05-20 2016-10-26 Cipla Ltd Process for preparing polycyclic carbamoyl pyridone derivatives
WO2018109786A1 (en) * 2016-12-16 2018-06-21 Cipla Limited Novel polymoprphs and salts of polycyclic carbamoyl pyridone derivatives
CN110582504A (zh) * 2017-02-16 2019-12-17 桑多斯股份公司 卡博特韦钠的晶形

Also Published As

Publication number Publication date
CA3053202C (en) 2022-10-04
US20200385401A1 (en) 2020-12-10
MX2019009810A (es) 2019-12-02
RU2019125378A (ru) 2021-03-16
AU2018221379A1 (en) 2019-08-29
US20210300945A1 (en) 2021-09-30
CA3053202A1 (en) 2018-08-23
AU2018221379B2 (en) 2021-11-04
EP3583107B1 (en) 2020-11-18
US11040986B2 (en) 2021-06-22
US20250236630A1 (en) 2025-07-24
AU2022200513A1 (en) 2022-02-17
EP3583107A1 (en) 2019-12-25
MX388699B (es) 2025-03-20
WO2018149608A1 (en) 2018-08-23
MX2021015441A (es) 2022-01-24
AU2022200513B2 (en) 2023-11-02
CN110582504A (zh) 2019-12-17

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HZ9A Changing address for correspondence with an applicant