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RU2018119359A - Способ индукции пролиферации кардиомиоцитов и лечения заболеваний сердца - Google Patents

Способ индукции пролиферации кардиомиоцитов и лечения заболеваний сердца Download PDF

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RU2018119359A
RU2018119359A RU2018119359A RU2018119359A RU2018119359A RU 2018119359 A RU2018119359 A RU 2018119359A RU 2018119359 A RU2018119359 A RU 2018119359A RU 2018119359 A RU2018119359 A RU 2018119359A RU 2018119359 A RU2018119359 A RU 2018119359A
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Prior art keywords
agrin
agrin peptide
domain
induces
peptide
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RU2018119359A
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RU2018119359A3 (ru
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Элдад ТЗАХОР
Элад БАССАТ
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Иеда Рисеч Энд Девелопмент Ко. Лтд.
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Publication of RU2018119359A publication Critical patent/RU2018119359A/ru
Publication of RU2018119359A3 publication Critical patent/RU2018119359A3/ru

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/1703Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • A61K38/1709Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61LMETHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
    • A61L27/00Materials for grafts or prostheses or for coating grafts or prostheses
    • A61L27/50Materials characterised by their function or physical properties, e.g. injectable or lubricating compositions, shape-memory materials, surface modified materials
    • A61L27/54Biologically active materials, e.g. therapeutic substances
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/46Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • C07K14/47Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
    • C07K14/4701Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals not used
    • C07K14/4725Proteoglycans, e.g. aggreccan
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N5/00Undifferentiated human, animal or plant cells, e.g. cell lines; Tissues; Cultivation or maintenance thereof; Culture media therefor
    • C12N5/06Animal cells or tissues; Human cells or tissues
    • C12N5/0602Vertebrate cells
    • C12N5/0652Cells of skeletal and connective tissues; Mesenchyme
    • C12N5/0657Cardiomyocytes; Heart cells
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61LMETHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
    • A61L2300/00Biologically active materials used in bandages, wound dressings, absorbent pads or medical devices
    • A61L2300/20Biologically active materials used in bandages, wound dressings, absorbent pads or medical devices containing or releasing organic materials
    • A61L2300/252Polypeptides, proteins, e.g. glycoproteins, lipoproteins, cytokines
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N2501/00Active agents used in cell culture processes, e.g. differentation
    • C12N2501/998Proteins not provided for elsewhere

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Zoology (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Wood Science & Technology (AREA)
  • Biotechnology (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • General Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Microbiology (AREA)
  • Cell Biology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Transplantation (AREA)
  • Marine Sciences & Fisheries (AREA)
  • Dermatology (AREA)
  • Oral & Maxillofacial Surgery (AREA)
  • Immunology (AREA)
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Claims (10)

1. Применение терапевтически эффективного количества агринового пептида, который индуцирует пролиферацию кардиомиоцитов, в изготовлении лекарственного препарата для лечения заболевания сердца, причем указанный агриновый пептид не является частью слитого полипептида, и причем указанный агриновый пептид содержит ламинин-G-подобный домен 1 (G1) и ламинин-G-подобный домен 2 (G2).
2. Применение средства, которое ингибирует дистрогликановый комплекс на кардиомиоцитах, в изготовлении лекарственного препарата для лечения заболевания сердца, причем указанное средство содержит агриновый пептид, который индуцирует пролиферацию кардиомиоцитов, указанный агриновый пептид не является частью слитого полипептида, и причем указанный агриновый пептид содержит ламинин-G-подобный домен 1 (G1) и ламинин-G-подобный домен 2 (G2).
3. Применение по п. 2, причем указанное средство содержит указанный агриновый пептид, который индуцирует иммуномодуляцию.
4. Применение по любому из пп. 2-3, причем указанное средство индуцирует активацию Erk.
5. Применение по любому из пп. 2-4, причем указанное средство ингибирует саркомерогенез.
6. Имплантируемое устройство, содержащее агриновый пептид, который индуцирует пролиферацию кардиомиоцитов, причем указанный агриновый пептид не является частью слитого полипептида, и причем указанный агриновый пептид содержит ламинин-G-подобный домен 1 (G1) и ламинин-G-подобный домен 2 (G2).
7. Устройство по п. 6, причем указанный агриновый пептид индуцирует иммуномодуляцию.
8. Применение по любому из пп. 1-5, причем указанный агриновый пептид имеет растворимую форму.
9. Применение по любому из пп. 1-5 и 8, причем указанный агриновый пептид содержит фрагмент агрина человека.
10. Применение по любому из пп. 1-5 и 8-9, причем указанное заболевание сердца является ишемической болезнью сердца.
RU2018119359A 2015-10-29 2016-10-27 Способ индукции пролиферации кардиомиоцитов и лечения заболеваний сердца RU2018119359A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IL242380 2015-10-29
IL242380A IL242380A0 (en) 2015-10-29 2015-10-29 A method for inducing the division of cardiomyocytes and treating heart diseases
PCT/IL2016/051165 WO2017072772A1 (en) 2015-10-29 2016-10-27 A method of inducing cardiomyocytes proliferation and treating heart diseases

Publications (2)

Publication Number Publication Date
RU2018119359A true RU2018119359A (ru) 2019-11-29
RU2018119359A3 RU2018119359A3 (ru) 2020-02-13

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RU2018119359A RU2018119359A (ru) 2015-10-29 2016-10-27 Способ индукции пролиферации кардиомиоцитов и лечения заболеваний сердца

Country Status (9)

Country Link
US (3) US10589132B2 (ru)
EP (2) EP3368058B1 (ru)
CN (1) CN108495647B (ru)
AU (2) AU2016347661B2 (ru)
DK (1) DK3368058T5 (ru)
ES (1) ES2949348T3 (ru)
IL (1) IL242380A0 (ru)
RU (1) RU2018119359A (ru)
WO (1) WO2017072772A1 (ru)

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IL292957A (en) 2022-05-11 2023-12-01 Yeda res & development co ltd Treatment of heart disease

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Also Published As

Publication number Publication date
US20180318612A1 (en) 2018-11-08
US11786640B2 (en) 2023-10-17
DK3368058T3 (da) 2023-07-24
ES2949348T3 (es) 2023-09-27
DK3368058T5 (da) 2024-09-30
AU2016347661A1 (en) 2018-06-14
EP3368058A1 (en) 2018-09-05
US10589132B2 (en) 2020-03-17
US20240042104A1 (en) 2024-02-08
EP4400164A2 (en) 2024-07-17
AU2023208156A1 (en) 2023-08-17
CN108495647B (zh) 2022-04-12
RU2018119359A3 (ru) 2020-02-13
EP3368058B1 (en) 2023-05-03
IL242380A0 (en) 2016-02-01
EP4400164A3 (en) 2024-09-11
AU2016347661B2 (en) 2023-08-17
CN108495647A (zh) 2018-09-04
US20200139162A1 (en) 2020-05-07
WO2017072772A1 (en) 2017-05-04

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