RU2011100552A - RECTAL OINTMENT CONTAINING INSULIN AND LIPOSOMES - Google Patents
RECTAL OINTMENT CONTAINING INSULIN AND LIPOSOMES Download PDFInfo
- Publication number
- RU2011100552A RU2011100552A RU2011100552/15A RU2011100552A RU2011100552A RU 2011100552 A RU2011100552 A RU 2011100552A RU 2011100552/15 A RU2011100552/15 A RU 2011100552/15A RU 2011100552 A RU2011100552 A RU 2011100552A RU 2011100552 A RU2011100552 A RU 2011100552A
- Authority
- RU
- Russia
- Prior art keywords
- liposomes
- ointment containing
- containing insulin
- rectal ointment
- rectal
- Prior art date
Links
- NOESYZHRGYRDHS-UHFFFAOYSA-N insulin Chemical compound N1C(=O)C(NC(=O)C(CCC(N)=O)NC(=O)C(CCC(O)=O)NC(=O)C(C(C)C)NC(=O)C(NC(=O)CN)C(C)CC)CSSCC(C(NC(CO)C(=O)NC(CC(C)C)C(=O)NC(CC=2C=CC(O)=CC=2)C(=O)NC(CCC(N)=O)C(=O)NC(CC(C)C)C(=O)NC(CCC(O)=O)C(=O)NC(CC(N)=O)C(=O)NC(CC=2C=CC(O)=CC=2)C(=O)NC(CSSCC(NC(=O)C(C(C)C)NC(=O)C(CC(C)C)NC(=O)C(CC=2C=CC(O)=CC=2)NC(=O)C(CC(C)C)NC(=O)C(C)NC(=O)C(CCC(O)=O)NC(=O)C(C(C)C)NC(=O)C(CC(C)C)NC(=O)C(CC=2NC=NC=2)NC(=O)C(CO)NC(=O)CNC2=O)C(=O)NCC(=O)NC(CCC(O)=O)C(=O)NC(CCCNC(N)=N)C(=O)NCC(=O)NC(CC=3C=CC=CC=3)C(=O)NC(CC=3C=CC=CC=3)C(=O)NC(CC=3C=CC(O)=CC=3)C(=O)NC(C(C)O)C(=O)N3C(CCC3)C(=O)NC(CCCCN)C(=O)NC(C)C(O)=O)C(=O)NC(CC(N)=O)C(O)=O)=O)NC(=O)C(C(C)CC)NC(=O)C(CO)NC(=O)C(C(C)O)NC(=O)C1CSSCC2NC(=O)C(CC(C)C)NC(=O)C(NC(=O)C(CCC(N)=O)NC(=O)C(CC(N)=O)NC(=O)C(NC(=O)C(N)CC=1C=CC=CC=1)C(C)C)CC1=CN=CN1 NOESYZHRGYRDHS-UHFFFAOYSA-N 0.000 title claims abstract 10
- 102000004877 Insulin Human genes 0.000 title claims abstract 5
- 108090001061 Insulin Proteins 0.000 title claims abstract 5
- 229940125396 insulin Drugs 0.000 title claims abstract 5
- 239000002502 liposome Substances 0.000 title claims abstract 5
- 229940098468 rectal ointment Drugs 0.000 title claims abstract 5
- 239000003937 drug carrier Substances 0.000 claims abstract 2
- 239000003995 emulsifying agent Substances 0.000 claims abstract 2
- 230000002209 hydrophobic effect Effects 0.000 claims abstract 2
- 239000000203 mixture Substances 0.000 claims abstract 2
- 239000000546 pharmaceutical excipient Substances 0.000 claims abstract 2
Landscapes
- Medicinal Preparation (AREA)
Abstract
1. Ректальная мазь, содержащая инсулин и фармацевтически приемлемые носители или эксципиенты, отличающаяся тем, что она дополнительно включает в себя липосомы. ! 2. Ректальная мазь по п.1, отличающаяся тем, что они имеют следующий состав, мас.%: ! инсулин 0,004-0,04 липосомы 0,01-20,0 эмульгатор 0,5-10,0 гидрофильная или гидрофобная основа 68,96-99,486 1. A rectal ointment containing insulin and pharmaceutically acceptable carriers or excipients, characterized in that it further includes liposomes. ! 2. Rectal ointment according to claim 1, characterized in that they have the following composition, wt.%:! insulin 0.004-0.04 liposomes 0.01-20.0 emulsifier 0.5-10.0 hydrophilic or hydrophobic base 68.96-99.486
Claims (2)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2011100552/15A RU2011100552A (en) | 2011-01-11 | 2011-01-11 | RECTAL OINTMENT CONTAINING INSULIN AND LIPOSOMES |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2011100552/15A RU2011100552A (en) | 2011-01-11 | 2011-01-11 | RECTAL OINTMENT CONTAINING INSULIN AND LIPOSOMES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RU2011100552A true RU2011100552A (en) | 2012-07-20 |
Family
ID=46846968
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2011100552/15A RU2011100552A (en) | 2011-01-11 | 2011-01-11 | RECTAL OINTMENT CONTAINING INSULIN AND LIPOSOMES |
Country Status (1)
| Country | Link |
|---|---|
| RU (1) | RU2011100552A (en) |
-
2011
- 2011-01-11 RU RU2011100552/15A patent/RU2011100552A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA92 | Acknowledgement of application withdrawn (lack of supplementary materials submitted) |
Effective date: 20121123 |
|
| FZ9A | Application not withdrawn (correction of the notice of withdrawal) |
Effective date: 20130115 |