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RU2001115829A - Дикетон в качестве промежуточного продукта при получении 3-галоген-1н-пиразолов - Google Patents

Дикетон в качестве промежуточного продукта при получении 3-галоген-1н-пиразолов

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Publication number
RU2001115829A
RU2001115829A RU2001115829/04A RU2001115829A RU2001115829A RU 2001115829 A RU2001115829 A RU 2001115829A RU 2001115829/04 A RU2001115829/04 A RU 2001115829/04A RU 2001115829 A RU2001115829 A RU 2001115829A RU 2001115829 A RU2001115829 A RU 2001115829A
Authority
RU
Russia
Prior art keywords
halogen
dicetone
pyrazoles
production
intermediate product
Prior art date
Application number
RU2001115829/04A
Other languages
English (en)
Other versions
RU2251543C2 (ru
Inventor
Бенксин ЗХИ
Мурад НЕВАЗ
Джон Дж. ТОЛИ
Стефен БЕРТЕНШО
Original Assignee
Джи. Ди. Сирл Энд Ко.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Джи. Ди. Сирл Энд Ко. filed Critical Джи. Ди. Сирл Энд Ко.
Publication of RU2001115829A publication Critical patent/RU2001115829A/ru
Application granted granted Critical
Publication of RU2251543C2 publication Critical patent/RU2251543C2/ru

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Claims (2)

1. Соединение общей формулы III
Figure 00000001
где R1 представляет собой галогеналкил;
R3 выбран из циклоалкила, циклоалкенила, арила и гетероарила, и R3 необязательно замещен в замещаемом положении одним или несколькими радикалами, выбранными из галогена, алкилтио, алкилсульфонила, циано, нитро, галогеналкила, алкила, гидроксила, алкенила, гидроксиалкила, карбоксила, циклоалкила, алкиламино, диалкиламино, алкоксикарбонила, аминокарбонила, алкокси, галогеналкокси, аминосульфонила, гетероцикло и амино.
2. Соединение по п.1, где R1 выбран из группы, включающей трифторметил, дифторметил, пентафторэтил и гептафторпропил, R3 представляет собой фенил, необязательно замещенный в замещаемом положении одним или несколькими радикалами, выбранными из фтора, хлора, брома, метила, этила, метокси, этокси и метилтио.
RU2001115829/04A 1995-05-25 1996-05-23 Дикетон в качестве промежуточного продукта при получении 3-галоген-1н-пиразолов RU2251543C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US44997595A 1995-05-25 1995-05-25
US08/449,975 1995-05-25

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
RU97121308/04A Division RU2169143C2 (ru) 1995-05-25 1996-05-23 Способ получения 3-галогеналкил-1н-пиразолов

Publications (2)

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RU2001115829A true RU2001115829A (ru) 2003-05-20
RU2251543C2 RU2251543C2 (ru) 2005-05-10

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RU97121308/04A RU2169143C2 (ru) 1995-05-25 1996-05-23 Способ получения 3-галогеналкил-1н-пиразолов
RU2001115829/04A RU2251543C2 (ru) 1995-05-25 1996-05-23 Дикетон в качестве промежуточного продукта при получении 3-галоген-1н-пиразолов

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US (2) US5892053A (ru)
EP (1) EP0828717B1 (ru)
JP (1) JP3996638B2 (ru)
KR (1) KR100444802B1 (ru)
CN (1) CN1174970C (ru)
AT (1) ATE223383T1 (ru)
AU (1) AU708964B2 (ru)
BR (1) BR9609043A (ru)
CA (1) CA2222138C (ru)
CZ (1) CZ292320B6 (ru)
DE (1) DE69623460T2 (ru)
DK (1) DK0828717T3 (ru)
ES (1) ES2182991T3 (ru)
NO (1) NO311130B1 (ru)
NZ (1) NZ308875A (ru)
PL (1) PL187410B1 (ru)
PT (1) PT828717E (ru)
RO (1) RO118200B1 (ru)
RU (2) RU2169143C2 (ru)
WO (1) WO1996037476A1 (ru)

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US20050009931A1 (en) * 2003-03-20 2005-01-13 Britten Nancy Jean Dispersible pharmaceutical composition for treatment of mastitis and otic disorders
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US20050004098A1 (en) * 2003-03-20 2005-01-06 Britten Nancy Jean Dispersible formulation of an anti-inflammatory agent
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