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RO77921A - PROCESS FOR THE PREPARATION OF DERIVATIVES OF INDOLIDIHYDROINDOL-3-CARBOXAMIDE - Google Patents

PROCESS FOR THE PREPARATION OF DERIVATIVES OF INDOLIDIHYDROINDOL-3-CARBOXAMIDE

Info

Publication number
RO77921A
RO77921A RO7798856A RO9885677A RO77921A RO 77921 A RO77921 A RO 77921A RO 7798856 A RO7798856 A RO 7798856A RO 9885677 A RO9885677 A RO 9885677A RO 77921 A RO77921 A RO 77921A
Authority
RO
Romania
Prior art keywords
indolidihydroindol
carboxamide
derivatives
preparation
Prior art date
Application number
RO7798856A
Other languages
French (fr)
Romanian (ro)
Inventor
George J Cullinan
Koert Gerzon
Original Assignee
Eli Lilly And Co,Us
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Co,Us filed Critical Eli Lilly And Co,Us
Publication of RO77921A publication Critical patent/RO77921A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C07D519/04Dimeric indole alkaloids, e.g. vincaleucoblastine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
RO7798856A 1976-09-08 1977-09-06 PROCESS FOR THE PREPARATION OF DERIVATIVES OF INDOLIDIHYDROINDOL-3-CARBOXAMIDE RO77921A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US72165076A 1976-09-08 1976-09-08

Publications (1)

Publication Number Publication Date
RO77921A true RO77921A (en) 1981-12-25

Family

ID=24898757

Family Applications (3)

Application Number Title Priority Date Filing Date
RO7798857A RO77922A (en) 1976-09-08 1977-09-06 PROCESS FOR THE PREPARATION OF DERIVATIVES OF INDOLIDIHYDROINDOL-3-CARBOXAMIDE
RO7798856A RO77921A (en) 1976-09-08 1977-09-06 PROCESS FOR THE PREPARATION OF DERIVATIVES OF INDOLIDIHYDROINDOL-3-CARBOXAMIDE
RO7791544A RO72474A (en) 1976-09-08 1977-09-07 PROCESS FOR PREPARING INDOLDIHYDROINDOL-3-CARBOXAMIDE DIMERES

Family Applications Before (1)

Application Number Title Priority Date Filing Date
RO7798857A RO77922A (en) 1976-09-08 1977-09-06 PROCESS FOR THE PREPARATION OF DERIVATIVES OF INDOLIDIHYDROINDOL-3-CARBOXAMIDE

Family Applications After (1)

Application Number Title Priority Date Filing Date
RO7791544A RO72474A (en) 1976-09-08 1977-09-07 PROCESS FOR PREPARING INDOLDIHYDROINDOL-3-CARBOXAMIDE DIMERES

Country Status (27)

Country Link
JP (1) JPS5340799A (en)
AR (3) AR226411A1 (en)
AT (1) AT360513B (en)
AU (1) AU511055B2 (en)
BE (1) BE858451A (en)
CA (1) CA1082179A (en)
CH (1) CH631990A5 (en)
DD (1) DD133055A5 (en)
DE (1) DE2739443A1 (en)
DK (1) DK146822C (en)
ES (1) ES462229A1 (en)
FR (1) FR2364220A1 (en)
GB (1) GB1586709A (en)
GR (1) GR69783B (en)
HU (1) HU180722B (en)
IE (1) IE45558B1 (en)
IL (1) IL52731A0 (en)
MX (1) MX4740E (en)
NL (1) NL7709806A (en)
NZ (1) NZ184932A (en)
PH (1) PH14771A (en)
PL (1) PL104309B1 (en)
PT (1) PT66984B (en)
RO (3) RO77922A (en)
SE (1) SE434953B (en)
YU (1) YU209777A (en)
ZA (1) ZA774988B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
USRE30561E (en) * 1976-12-06 1981-03-31 Eli Lilly And Company Vinca alkaloid intermediates
US4199504A (en) * 1978-05-15 1980-04-22 Eli Lilly And Company Bridged cathranthus alkaloid dimers
AR225153A1 (en) * 1978-10-10 1982-02-26 Lilly Co Eli A PROCEDURE FOR THE PREPARATION OF VINDESINE SULPHATE
US4357334A (en) 1980-03-20 1982-11-02 Eli Lilly And Company Use of VLB 3-(2-chloroethyl) carboxamide in treating neoplasms
OA06421A (en) * 1980-06-10 1981-09-30 Omnium Chimique Sa Process for the preparation of N- (vinblastinoyl-23) derivatives of amino acids and peptides.
US4362664A (en) * 1980-12-29 1982-12-07 Eli Lilly And Company Vinblastine oxazolidinedione disulfides and related compounds
US4831038A (en) * 1986-01-13 1989-05-16 Ire-Celltarg S.A. Vinblastine derivatives and pharmaceutical composition containing them

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR204004A1 (en) * 1973-04-02 1975-11-12 Lilly Co Eli PROCEDURES FOR PREPARING VINBLASTIN LEUROSIDINE AND LEUROCRISTINE DERIVATIVES
IL48685A (en) * 1975-01-09 1980-03-31 Lilly Co Eli Amides of vincadioline and vinblastine

Also Published As

Publication number Publication date
AR226411A1 (en) 1982-07-15
ZA774988B (en) 1979-03-28
AR231643A1 (en) 1985-01-31
IE45558B1 (en) 1982-09-22
DK398577A (en) 1978-03-09
RO72474A (en) 1982-05-10
GR69783B (en) 1982-07-07
FR2364220A1 (en) 1978-04-07
HU180722B (en) 1983-04-29
PH14771A (en) 1981-12-09
MX4740E (en) 1982-08-25
SE7710059L (en) 1978-03-09
ES462229A1 (en) 1978-07-16
NL7709806A (en) 1978-03-10
DE2739443A1 (en) 1978-03-09
YU209777A (en) 1982-08-31
BE858451A (en) 1978-03-07
DE2739443C2 (en) 1991-08-14
PL200607A1 (en) 1978-05-22
AU511055B2 (en) 1980-07-24
DD133055A5 (en) 1978-11-29
RO77922A (en) 1981-12-25
FR2364220B1 (en) 1980-04-25
PT66984B (en) 1979-02-13
ATA644277A (en) 1980-06-15
PT66984A (en) 1977-10-01
NZ184932A (en) 1979-11-01
AT360513B (en) 1981-01-12
GB1586709A (en) 1981-03-25
IL52731A0 (en) 1977-10-31
PL104309B1 (en) 1979-08-31
JPS624398B2 (en) 1987-01-30
SE434953B (en) 1984-08-27
AR230642A1 (en) 1984-05-31
CH631990A5 (en) 1982-09-15
AU2803977A (en) 1979-02-22
DK146822B (en) 1984-01-16
CA1082179A (en) 1980-07-22
JPS5340799A (en) 1978-04-13
IE771700L (en) 1978-03-08
DK146822C (en) 1984-06-25

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