PT99238A - Processo para a preparacao de composicoes farmaceuticas contendo um inibidor da enzima conversora da angiotensina e um inibidor da actividade do tromboxano a2, utilizadas no tratamento de nefropatias - Google Patents
Processo para a preparacao de composicoes farmaceuticas contendo um inibidor da enzima conversora da angiotensina e um inibidor da actividade do tromboxano a2, utilizadas no tratamento de nefropatiasInfo
- Publication number
- PT99238A PT99238A PT99238A PT9923891A PT99238A PT 99238 A PT99238 A PT 99238A PT 99238 A PT99238 A PT 99238A PT 9923891 A PT9923891 A PT 9923891A PT 99238 A PT99238 A PT 99238A
- Authority
- PT
- Portugal
- Prior art keywords
- inhibitor
- nephropathes
- thomboxane
- activity
- preparation
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 2
- UUUHXMGGBIUAPW-UHFFFAOYSA-N 1-[1-[2-[[5-amino-2-[[1-[5-(diaminomethylideneamino)-2-[[1-[3-(1h-indol-3-yl)-2-[(5-oxopyrrolidine-2-carbonyl)amino]propanoyl]pyrrolidine-2-carbonyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]pyrrolidine-2-carbon Chemical compound C1CCC(C(=O)N2C(CCC2)C(O)=O)N1C(=O)C(C(C)CC)NC(=O)C(CCC(N)=O)NC(=O)C1CCCN1C(=O)C(CCCN=C(N)N)NC(=O)C1CCCN1C(=O)C(CC=1C2=CC=CC=C2NC=1)NC(=O)C1CCC(=O)N1 UUUHXMGGBIUAPW-UHFFFAOYSA-N 0.000 title 1
- 102000004270 Peptidyl-Dipeptidase A Human genes 0.000 title 1
- 108090000882 Peptidyl-Dipeptidase A Proteins 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/55—Protease inhibitors
- A61K38/556—Angiotensin converting enzyme inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Vascular Medicine (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Gastroenterology & Hepatology (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT021757A IT9021757A1 (it) | 1990-10-16 | 1990-10-16 | Prodotto per il trattamento delle nefropatie |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT99238A true PT99238A (pt) | 1992-09-30 |
Family
ID=11186438
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT99238A PT99238A (pt) | 1990-10-16 | 1991-10-15 | Processo para a preparacao de composicoes farmaceuticas contendo um inibidor da enzima conversora da angiotensina e um inibidor da actividade do tromboxano a2, utilizadas no tratamento de nefropatias |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0556204A1 (pt) |
| JP (1) | JPH06501943A (pt) |
| AU (1) | AU8725191A (pt) |
| IE (1) | IE913585A1 (pt) |
| IL (1) | IL99667A0 (pt) |
| IT (1) | IT9021757A1 (pt) |
| PT (1) | PT99238A (pt) |
| WO (1) | WO1992006713A1 (pt) |
| ZA (1) | ZA918038B (pt) |
-
1990
- 1990-10-16 IT IT021757A patent/IT9021757A1/it unknown
-
1991
- 1991-10-08 IL IL99667A patent/IL99667A0/xx unknown
- 1991-10-08 ZA ZA918038A patent/ZA918038B/xx unknown
- 1991-10-15 PT PT99238A patent/PT99238A/pt not_active Application Discontinuation
- 1991-10-16 WO PCT/EP1991/001972 patent/WO1992006713A1/en not_active Ceased
- 1991-10-16 AU AU87251/91A patent/AU8725191A/en not_active Abandoned
- 1991-10-16 JP JP3516412A patent/JPH06501943A/ja active Pending
- 1991-10-16 EP EP91918149A patent/EP0556204A1/en not_active Withdrawn
- 1991-10-16 IE IE358591A patent/IE913585A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA918038B (en) | 1992-06-24 |
| AU8725191A (en) | 1992-05-20 |
| IL99667A0 (en) | 1992-08-18 |
| IT9021757A0 (it) | 1990-10-16 |
| IE913585A1 (en) | 1992-04-22 |
| WO1992006713A1 (en) | 1992-04-30 |
| EP0556204A1 (en) | 1993-08-25 |
| IT9021757A1 (it) | 1992-04-16 |
| JPH06501943A (ja) | 1994-03-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB1A | Laying open of patent application |
Effective date: 19920422 |
|
| FC3A | Refusal |
Effective date: 19931015 |