PT92539A - Processo para a preparacao de derivados de anfotericina b - Google Patents
Processo para a preparacao de derivados de anfotericina bInfo
- Publication number
- PT92539A PT92539A PT92539A PT9253989A PT92539A PT 92539 A PT92539 A PT 92539A PT 92539 A PT92539 A PT 92539A PT 9253989 A PT9253989 A PT 9253989A PT 92539 A PT92539 A PT 92539A
- Authority
- PT
- Portugal
- Prior art keywords
- anfotericin
- derivatives
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
- C07H15/08—Polyoxyalkylene derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Crystallography & Structural Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB888829592A GB8829592D0 (en) | 1988-12-19 | 1988-12-19 | Novel compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT92539A true PT92539A (pt) | 1990-06-29 |
| PT92539B PT92539B (pt) | 1995-08-09 |
Family
ID=10648736
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT92539A PT92539B (pt) | 1988-12-19 | 1989-12-11 | Processo para a preparacao de derivados de anfotericina b |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US5066646A (pt) |
| EP (1) | EP0375223A3 (pt) |
| JP (1) | JPH02207094A (pt) |
| KR (1) | KR900009678A (pt) |
| AU (1) | AU614205B2 (pt) |
| CA (1) | CA2005133A1 (pt) |
| DK (1) | DK625389A (pt) |
| GB (1) | GB8829592D0 (pt) |
| NZ (1) | NZ231723A (pt) |
| PT (1) | PT92539B (pt) |
| ZA (1) | ZA899505B (pt) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0350164A3 (en) * | 1988-06-13 | 1991-07-24 | Beecham Group Plc | Amphotericin derivatives |
| GB8829593D0 (en) * | 1988-12-19 | 1989-02-08 | Beecham Group Plc | Novel compounds |
| WO1991009047A1 (en) * | 1989-12-08 | 1991-06-27 | Beecham Group Plc | Amphotericin b derivatives, their production and use |
| GB9114949D0 (en) * | 1991-07-11 | 1991-08-28 | Smithkline Beecham Plc | Novel compounds |
| FR2683723B1 (fr) * | 1991-11-14 | 1995-05-19 | Mayoly Spindler Laboratoires | Nouveaux medicaments antiviraux actifs sur le virus vih. |
| GB9200713D0 (en) * | 1992-01-14 | 1992-03-11 | Smithkline Beecham Plc | Novel compounds |
| GB9203476D0 (en) * | 1992-02-19 | 1992-04-08 | Smithkline Beecham Plc | Novel compounds |
| WO2001051061A1 (en) | 2000-01-14 | 2001-07-19 | Intrabiotics Pharmaceuticals, Inc. | Derivatives of polyene macrolides and preparation and use thereof |
| CN102115484B (zh) * | 2009-12-31 | 2013-03-13 | 中国药品生物制品检定所 | 一种两性霉素b降解产物、其制备方法及其应用 |
| US9447136B2 (en) | 2012-03-09 | 2016-09-20 | Blirt S.A. | Semisynthetic derivatives of Nystatin A1 |
| KR20150027217A (ko) | 2012-06-15 | 2015-03-11 | 블러트 에스.에이. | 항진균성 항생 암포테리신 b의 n-치환된 제2 세대 유도체, 및 이의 제조 및 응용 방법 |
| JP7240811B2 (ja) | 2015-04-15 | 2023-03-16 | スファンガ セラピューティクス インコーポレイテッド | アムホテリシンbの誘導体 |
| TWI637980B (zh) * | 2017-01-11 | 2018-10-11 | 長興材料工業股份有限公司 | 聚醯亞胺前驅物及其應用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2173632A1 (en) * | 1971-02-04 | 1973-10-12 | Le N Iss | Purificn of amfotericin b - in dmf soln by adding water acidifying filtering adding water,making alkaline and washing |
| US4041232A (en) * | 1976-02-23 | 1977-08-09 | E. R. Squibb & Sons, Inc. | Amphotericin B methyl ester salts |
| US4235993A (en) * | 1979-02-21 | 1980-11-25 | E. R. Squibb & Sons, Inc. | N-Benzylideneamphotericin B, its methyl ester and process for making water-soluble salts thereof |
| EP0350164A3 (en) * | 1988-06-13 | 1991-07-24 | Beecham Group Plc | Amphotericin derivatives |
| GB8829593D0 (en) * | 1988-12-19 | 1989-02-08 | Beecham Group Plc | Novel compounds |
-
1988
- 1988-12-19 GB GB888829592A patent/GB8829592D0/en active Pending
-
1989
- 1989-12-08 EP EP19890312825 patent/EP0375223A3/en not_active Withdrawn
- 1989-12-11 CA CA002005133A patent/CA2005133A1/en not_active Abandoned
- 1989-12-11 US US07/448,698 patent/US5066646A/en not_active Expired - Fee Related
- 1989-12-11 DK DK625389A patent/DK625389A/da not_active Application Discontinuation
- 1989-12-11 AU AU46171/89A patent/AU614205B2/en not_active Ceased
- 1989-12-11 PT PT92539A patent/PT92539B/pt not_active IP Right Cessation
- 1989-12-12 NZ NZ231723A patent/NZ231723A/en unknown
- 1989-12-12 KR KR1019890018428A patent/KR900009678A/ko not_active Withdrawn
- 1989-12-12 JP JP1320750A patent/JPH02207094A/ja active Pending
- 1989-12-13 ZA ZA899505A patent/ZA899505B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK625389A (da) | 1990-06-20 |
| AU614205B2 (en) | 1991-08-22 |
| AU4617189A (en) | 1990-06-21 |
| PT92539B (pt) | 1995-08-09 |
| EP0375223A2 (en) | 1990-06-27 |
| CA2005133A1 (en) | 1990-06-19 |
| US5066646A (en) | 1991-11-19 |
| NZ231723A (en) | 1992-03-26 |
| KR900009678A (ko) | 1990-07-05 |
| GB8829592D0 (en) | 1989-02-08 |
| DK625389D0 (da) | 1989-12-11 |
| JPH02207094A (ja) | 1990-08-16 |
| ZA899505B (en) | 1990-12-28 |
| EP0375223A3 (en) | 1991-07-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG3A | Patent granted, date of granting |
Effective date: 19950412 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19961031 |