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PT840609E - Utilizacao de n-(pirrol-1-il)-pirimidinas insubstituidas e substituidas como agentes anticonvulsivos - Google Patents

Utilizacao de n-(pirrol-1-il)-pirimidinas insubstituidas e substituidas como agentes anticonvulsivos

Info

Publication number
PT840609E
PT840609E PT96923693T PT96923693T PT840609E PT 840609 E PT840609 E PT 840609E PT 96923693 T PT96923693 T PT 96923693T PT 96923693 T PT96923693 T PT 96923693T PT 840609 E PT840609 E PT 840609E
Authority
PT
Portugal
Prior art keywords
insubstituted
pyrrol
pyridines
replaced
anticonvulsive agents
Prior art date
Application number
PT96923693T
Other languages
English (en)
Inventor
Francis P Huger
Sathapana Kongsamut
Craig Paul Smith
Lei Tang
Original Assignee
Aventis Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Inc filed Critical Aventis Pharma Inc
Publication of PT840609E publication Critical patent/PT840609E/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT96923693T 1995-07-27 1996-07-08 Utilizacao de n-(pirrol-1-il)-pirimidinas insubstituidas e substituidas como agentes anticonvulsivos PT840609E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US50807195A 1995-07-27 1995-07-27

Publications (1)

Publication Number Publication Date
PT840609E true PT840609E (pt) 2002-10-31

Family

ID=24021262

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96923693T PT840609E (pt) 1995-07-27 1996-07-08 Utilizacao de n-(pirrol-1-il)-pirimidinas insubstituidas e substituidas como agentes anticonvulsivos

Country Status (19)

Country Link
EP (1) EP0840609B1 (pt)
JP (1) JP4189029B2 (pt)
KR (1) KR100445629B1 (pt)
CN (1) CN1184969C (pt)
AR (1) AR003471A1 (pt)
AT (1) ATE218343T1 (pt)
AU (1) AU696007B2 (pt)
CA (1) CA2225156C (pt)
DE (1) DE69621617T2 (pt)
DK (1) DK0840609T3 (pt)
ES (1) ES2174081T3 (pt)
IL (1) IL122845A0 (pt)
MX (1) MX9800774A (pt)
NO (1) NO315148B1 (pt)
NZ (1) NZ312577A (pt)
PT (1) PT840609E (pt)
TW (1) TW464497B (pt)
WO (1) WO1997004777A1 (pt)
ZA (1) ZA966254B (pt)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GT200500063A (es) * 2004-04-01 2005-10-14 Metodo para tratar la esquizofrenia y/o anormalidades glucoregulatorias
FR2897614B1 (fr) * 2006-02-20 2008-05-23 Urogene Forme cristalline du chlorhydrate de la besipirdine, procedes de preparation et utilisations

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5032599A (en) * 1986-11-12 1991-07-16 Hoechst-Roussel Pharmaceuticals Inc. N-(pyrrol-l-yl)pyridinamines
ATE115143T1 (de) * 1987-04-24 1994-12-15 Hoechst Roussel Pharma N-(pyridinyl)-1h-indol-1-amine, verfahren zu deren herstellung und ihre verwendung als arzneimittel.
US4868190A (en) * 1988-12-27 1989-09-19 Hoechst-Roussel Pharmaceuticals, Inc. N-pyridinyl-9H-carbazol-9-amines
US5179099A (en) * 1989-08-02 1993-01-12 Hoechst-Roussel Pharmaceuticals Incorporated 2,3-dihydro-1-(pyridinylamino)-indoles
US5356910A (en) * 1993-07-19 1994-10-18 Hoechst-Roussel Pharmaceuticals Inc. Use of N-(pyridinyl)-1H-indol-1-amines for the treatment of obsessive-compulsive disorder

Also Published As

Publication number Publication date
DK0840609T3 (da) 2002-09-30
EP0840609A1 (en) 1998-05-13
NO980334L (no) 1998-03-26
KR100445629B1 (ko) 2004-10-14
AU6454796A (en) 1997-02-26
CA2225156C (en) 2003-06-10
AU696007B2 (en) 1998-08-27
KR19990035973A (ko) 1999-05-25
AR003471A1 (es) 1998-08-05
JPH11510159A (ja) 1999-09-07
HK1015687A1 (en) 1999-10-22
NZ312577A (en) 1999-08-30
ES2174081T3 (es) 2002-11-01
ATE218343T1 (de) 2002-06-15
NO980334D0 (no) 1998-01-26
MX9800774A (es) 1998-04-30
EP0840609B1 (en) 2002-06-05
NO315148B1 (no) 2003-07-21
IL122845A0 (en) 1998-08-16
ZA966254B (en) 1997-02-11
WO1997004777A1 (en) 1997-02-13
DE69621617T2 (de) 2003-01-02
CN1191486A (zh) 1998-08-26
JP4189029B2 (ja) 2008-12-03
CA2225156A1 (en) 1997-02-13
CN1184969C (zh) 2005-01-19
TW464497B (en) 2001-11-21
DE69621617D1 (de) 2002-07-11

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