PT1497290E - Processo para preparação de sais de ácido de gemifloxacina - Google Patents

Processo para preparação de sais de ácido de gemifloxacina Download PDF

Info

Publication number: PT1497290E
Authority: PT; Portugal
Prior art keywords: gemifloxacin; acid salts; preparing acid; preparing; salts
Prior art date: 2002-04-08

Application number

PT03715805T

Other languages

English (en)

Inventor

Hoon Choi

Sang-Chul Choi

Do-Hyun Nam

Bo-Seung Choi

Original Assignee

Lg Life Sciences Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-04-08

Filing date

2003-04-04

Publication date

2008-11-14

2003-04-04 Application filed by Lg Life Sciences Ltd filed Critical Lg Life Sciences Ltd

2008-11-14 Publication of PT1497290E publication Critical patent/PT1497290E/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Saccharide Compounds (AREA)

PT03715805T 2002-04-08 2003-04-04 Processo para preparação de sais de ácido de gemifloxacina PT1497290E (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
KR10-2002-0018847A KR100517638B1 (ko)	2002-04-08	2002-04-08	게미플록사신 산염의 새로운 제조방법

Publications (1)

Publication Number	Publication Date
PT1497290E true PT1497290E (pt)	2008-11-14

Family

ID=36241771

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT03715805T PT1497290E (pt)	2002-04-08	2003-04-04	Processo para preparação de sais de ácido de gemifloxacina

Country Status (31)

Country	Link
US (1)	US7361762B2 (pt)
EP (1)	EP1497290B1 (pt)
JP (1)	JP4315815B2 (pt)
KR (1)	KR100517638B1 (pt)
CN (1)	CN1291987C (pt)
AP (1)	AP1786A (pt)
AT (1)	ATE404559T1 (pt)
AU (1)	AU2003219581B2 (pt)
BR (1)	BRPI0309037B8 (pt)
CA (1)	CA2481217C (pt)
CO (1)	CO5611198A2 (pt)
CY (1)	CY1108469T1 (pt)
DE (1)	DE60322872D1 (pt)
DK (1)	DK1497290T3 (pt)
EA (1)	EA007222B1 (pt)
ES (1)	ES2311694T3 (pt)
GE (1)	GEP20074025B (pt)
HR (1)	HRP20040929B1 (pt)
IL (1)	IL164328A (pt)
IS (1)	IS2731B (pt)
MA (1)	MA26408A1 (pt)
MX (1)	MXPA04009777A (pt)
NO (1)	NO330042B1 (pt)
NZ (1)	NZ536174A (pt)
OA (1)	OA12801A (pt)
PL (1)	PL372815A1 (pt)
PT (1)	PT1497290E (pt)
SI (1)	SI1497290T1 (pt)
UA (1)	UA77070C2 (pt)
WO (1)	WO2003087100A1 (pt)
ZA (1)	ZA200408088B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PT1412078E (pt) *	2001-08-02	2009-01-08	Lg Life Sciences Ltd	Processos para a produção de derivados amino-protegidos da 4- aminometileno-pirrolidin-3-ona, gemifloxacina ou um seu sal
WO2006134431A1 (en) *	2005-05-03	2006-12-21	Ranbaxy Laboratories Limited	Formate salt of gemifloxacin
EP2159225A1 (en) *	2005-06-15	2010-03-03	Hetero Drugs Limited	Gemifloxacin process and polymorphs
KR20130128483A (ko) *	2006-03-07	2013-11-26	욱크하트 리미티드	벤조퀴놀리진-2-카르복실산의 프로드러그
US20100076193A1 (en) *	2006-10-31	2010-03-25	Chandrasekaran Ramasubbu	process for the preparation of gemifloxacin

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JPS57134482A (en)	1981-02-13	1982-08-19	Dainippon Pharmaceut Co Ltd	1-ethyl-6-fluoro-1,4-dihydro-4-oxo-7-(1-piperazinyl)-1,8- naphthyridine-3-carboxylic acid-3/2 hydrate and its preparation
IN162769B (pt)	1984-11-13	1988-07-09	Kyorin Seiyaku Kk
NZ222047A (en)	1986-10-08	1991-01-29	Bristol Myers Co	Quinoline - or naphthyridine - carboxylic acid anti-bacterial agents
JPH01100165A (ja)	1987-10-13	1989-04-18	Shionogi & Co Ltd	オキシムまたはヒドロキシアミン誘導体系抗菌剤
US4920120A (en)	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents
JPH0356479A (ja)	1989-07-24	1991-03-12	Takeshi Yokota	水溶性キノロン誘導体のｐ‐トルエンスルホン酸塩
PL166381B1 (pl)	1989-08-16	1995-05-31	Pfizer	Sposób wytwarzania nowych podstawionych kwasów 7-azabicyklochinolonokarboksylowych PL PL PL PL
US5137892A (en)	1990-12-12	1992-08-11	Abbott Laboratories	Quinoline, naphthyridine and pyridobenzoxazine derivatives
EP0541086A1 (en)	1991-11-08	1993-05-12	Kaken Pharmaceutical Co., Ltd.	Antibacterial 6-fluoro-quinolones having an oxime group on the substituent in position 7
JPH0673056A (ja)	1992-08-26	1994-03-15	Kaken Pharmaceut Co Ltd	キノリンカルボン酸誘導体およびその塩
DE69509442T2 (de)	1994-06-16	1999-09-02	Lg Chemical Ltd.	Chinolincarbonsäurederivate mit 7-(4-Amino-methyl-3-oxim)-pyrrolidin-Substituenten und Verfahren zu ihrer Herstellung
US5776944A (en) *	1994-06-16	1998-07-07	Lg Chemical Ltd.	7-(4-aminomethyl-3-methyloxyiminopyrroplidin-1-yl)-1-cyclopropyl-6-flu oro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
JP3449658B2 (ja)	1994-12-21	2003-09-22	杏林製薬株式会社	安定性に優れた８−アルコキシキノロンカルボン酸水和物並びにその製造方法
ES2117426T3 (es)	1995-06-06	1998-08-01	Pfizer	Forma cristalina de la sal anhidra compuesta de los acidos 7-((1a,5a,6a)-6-amino-3-azabiciclo(3.1.0.)hex-3-il)-6-fluoro-1-(2,4-difluorofenil)-1,4-dihidro-4-oxo-1,8-naftiridina-3-carboxilico y metanosulfonico.
UA59341C2 (uk)	1995-08-11	2003-09-15	Пфайзер, Інк.	(1s,2s)-1-(4-гідроксифеніл)-2-(4-гідрокси-4-фенілпіперидин-1-іл)-1-пропанолметансульфонат тригідрат
JP4316013B2 (ja)	1996-03-29	2009-08-19	スミスクライン・ビーチャム・コーポレイション	エプロサルタン二水和物ならびにその製法および処方
MA24500A1 (fr) *	1997-03-21	1998-10-01	Lg Life Sciences Ltd	Derive du sel d'acide carboxylique de naphthyridine .
KR100286874B1 (ko)	1998-03-04	2001-04-16	성재갑	보호된 4-아미노메틸-피롤리딘-3-온의 제조방법
PT1082300E (pt)	1998-05-29	2004-02-27	Upjohn Co	Monometanossulfonato de 3-¬(1'-n-metilamino)etil-n-benzil\|pirrolidina
GB9820405D0 (en)	1998-09-18	1998-11-11	Smithkline Beecham Plc	Process
PT1223935E (pt)	1999-06-29	2008-04-03	Lg Life Sciences Ltd	Utilização de compostos de gemifloxacina contra bactérias
AU6947900A (en)	1999-09-01	2001-03-26	Smithkline Beecham Corporation	Methods of use of fluoroquinolone compounds against bacteria
GB9920917D0 (en) *	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel process
GB9920919D0 (en)	1999-09-03	1999-11-10	Sb Pharmco Inc	Novel compound
EP1242079A4 (en)	1999-09-22	2003-01-22	Smithkline Beecham	Methods of anti-bacterial use of fluoroquinolonic compounds
KR20010091379A (ko)	2000-03-15	2001-10-23	성재갑	7-(4-아미노메틸-3-옥심)피롤리딘 치환체를 갖는 퀴놀린카르복실산 유도체의 신규 제조방법
KR20020018560A (ko)	2000-09-01	2002-03-08	성재갑	3-아미노메틸-4-ｚ-메톡시이미노피롤리딘의 신규 제조방법

2002
- 2002-04-08 KR KR10-2002-0018847A patent/KR100517638B1/ko not_active Expired - Lifetime
2003
- 2003-04-04 JP JP2003584056A patent/JP4315815B2/ja not_active Expired - Fee Related
- 2003-04-04 AT AT03715805T patent/ATE404559T1/de active
- 2003-04-04 NZ NZ536174A patent/NZ536174A/en not_active IP Right Cessation
- 2003-04-04 US US10/510,514 patent/US7361762B2/en not_active Expired - Lifetime
- 2003-04-04 EA EA200401328A patent/EA007222B1/ru not_active IP Right Cessation
- 2003-04-04 MX MXPA04009777A patent/MXPA04009777A/es active IP Right Grant
- 2003-04-04 OA OA1200400271A patent/OA12801A/en unknown
- 2003-04-04 PT PT03715805T patent/PT1497290E/pt unknown
- 2003-04-04 SI SI200331341T patent/SI1497290T1/sl unknown
- 2003-04-04 AP APAP/P/2004/003148A patent/AP1786A/en active
- 2003-04-04 WO PCT/KR2003/000683 patent/WO2003087100A1/en not_active Ceased
- 2003-04-04 ES ES03715805T patent/ES2311694T3/es not_active Expired - Lifetime
- 2003-04-04 DK DK03715805T patent/DK1497290T3/da active
- 2003-04-04 AU AU2003219581A patent/AU2003219581B2/en not_active Ceased
- 2003-04-04 EP EP03715805A patent/EP1497290B1/en not_active Expired - Lifetime
- 2003-04-04 HR HRP20040929AA patent/HRP20040929B1/hr not_active IP Right Cessation
- 2003-04-04 UA UA20041008144A patent/UA77070C2/uk unknown
- 2003-04-04 PL PL03372815A patent/PL372815A1/xx not_active Application Discontinuation
- 2003-04-04 GE GEAP8436A patent/GEP20074025B/en unknown
- 2003-04-04 BR BRPI0309037A patent/BRPI0309037B8/pt not_active IP Right Cessation
- 2003-04-04 DE DE60322872T patent/DE60322872D1/de not_active Expired - Lifetime
- 2003-04-04 CN CNB038095483A patent/CN1291987C/zh not_active Expired - Lifetime
- 2003-04-04 CA CA2481217A patent/CA2481217C/en not_active Expired - Lifetime
2004
- 2004-09-30 IS IS7477A patent/IS2731B/is unknown
- 2004-10-05 CO CO04099283A patent/CO5611198A2/es active IP Right Grant
- 2004-10-07 MA MA27894A patent/MA26408A1/fr unknown
- 2004-10-07 ZA ZA200408088A patent/ZA200408088B/xx unknown
- 2004-10-21 IL IL164328A patent/IL164328A/en unknown
- 2004-10-27 NO NO20044629A patent/NO330042B1/no not_active IP Right Cessation
2008
- 2008-10-31 CY CY20081101234T patent/CY1108469T1/el unknown

Also Published As

Publication number	Publication date
ZA200408088B (en)	2006-05-31
DK1497290T3 (da)	2008-12-15
EA007222B1 (ru)	2006-08-25
HRP20040929A2 (en)	2005-02-28
EP1497290A4 (en)	2006-05-10
NO330042B1 (no)	2011-02-07
IS2731B (is)	2011-04-15
US20050148622A1 (en)	2005-07-07
AP2004003148A0 (en)	2004-12-31
KR100517638B1 (ko)	2005-09-28
BR0309037A (pt)	2005-02-01
CA2481217A1 (en)	2003-10-23
MA26408A1 (fr)	2004-12-01
UA77070C2 (uk)	2006-10-16
DE60322872D1 (de)	2008-09-25
KR20030080292A (ko)	2003-10-17
HRP20040929B1 (hr)	2013-12-06
EA200401328A1 (ru)	2005-06-30
CA2481217C (en)	2010-06-01
US7361762B2 (en)	2008-04-22
ATE404559T1 (de)	2008-08-15
AU2003219581A1 (en)	2003-10-27
NZ536174A (en)	2006-09-29
HK1074440A1 (en)	2005-11-11
BRPI0309037B1 (pt)	2018-07-31
MXPA04009777A (es)	2004-12-13
PL372815A1 (en)	2005-08-08
ES2311694T3 (es)	2009-02-16
IS7477A (is)	2004-09-30
EP1497290A1 (en)	2005-01-19
NO20044629L (no)	2004-10-27
BRPI0309037B8 (pt)	2021-05-25
CN1291987C (zh)	2006-12-27
IL164328A (en)	2009-08-03
SI1497290T1 (sl)	2008-12-31
IL164328A0 (en)	2005-12-18
CN1649868A (zh)	2005-08-03
AU2003219581B2 (en)	2006-08-24
OA12801A (en)	2006-07-11
CO5611198A2 (es)	2006-02-28
WO2003087100A1 (en)	2003-10-23
JP2005529112A (ja)	2005-09-29
GEP20074025B (en)	2007-01-25
JP4315815B2 (ja)	2009-08-19
AP1786A (en)	2007-10-04
EP1497290B1 (en)	2008-08-13
CY1108469T1 (el)	2014-04-09

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