PT100821A - Compostos amino terciario substituidos com triazolilo e seus sais, e processo para a sua preparacao - Google Patents

Compostos amino terciario substituidos com triazolilo e seus sais, e processo para a sua preparacao

Info

Publication number: PT100821A
Authority: PT; Portugal
Prior art keywords: triazolyl; heterocyclic group; salts; preparation; substituted amino
Prior art date: 1991-09-02

Application number

PT100821A

Other languages

English (en)

Other versions

PT100821B (pt

Inventor

Okada Minoru

Kawaminami Eiji

Yoden Toru

Kudo Masafumi

Isomura Yasuo

Original Assignee

Yamanouchi Pharma Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-09-02

Filing date

1992-08-28

Publication date

1993-11-30

1992-08-28 Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd

1993-11-30 Publication of PT100821A publication Critical patent/PT100821A/pt

1999-07-30 Publication of PT100821B publication Critical patent/PT100821B/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Medicinal Preparation (AREA)
Treatments Of Macromolecular Shaped Articles (AREA)
Processes Of Treating Macromolecular Substances (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
Cosmetics (AREA)

PT100821A 1991-09-02 1992-08-28 Compostos amino terciario substituidos com triazolilo e seus sais, e processo para a sua preparacao PT100821B (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP24826891		1991-09-02
JP34401191		1991-12-02

Publications (2)

Publication Number	Publication Date
PT100821A true PT100821A (pt)	1993-11-30
PT100821B PT100821B (pt)	1999-07-30

Family

ID=26538684

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT100821A PT100821B (pt)	1991-09-02	1992-08-28	Compostos amino terciario substituidos com triazolilo e seus sais, e processo para a sua preparacao

Country Status (20)

Country	Link
US (1)	US5674886A (pt)
EP (1)	EP0641785B1 (pt)
KR (1)	KR100204697B1 (pt)
CN (1)	CN1035817C (pt)
AT (1)	ATE186052T1 (pt)
AU (1)	AU665569B2 (pt)
BG (1)	BG61688B1 (pt)
CA (1)	CA2116773C (pt)
DE (1)	DE69230225T2 (pt)
ES (1)	ES2139605T3 (pt)
FI (1)	FI940988L (pt)
HU (1)	HU220863B1 (pt)
MX (1)	MX9204996A (pt)
NO (1)	NO305284B1 (pt)
PT (1)	PT100821B (pt)
RO (1)	RO114129B1 (pt)
RU (1)	RU2124010C1 (pt)
TW (1)	TW225526B (pt)
UA (1)	UA41295C2 (pt)
WO (1)	WO1993005027A1 (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5770616A (en)	1995-06-07	1998-06-23	The Procter & Gamble Company	Pharmaceutical composition for inhibiting the growth of cancers
RU2131422C1 (ru) *	1997-05-21	1999-06-10	Иван Антонович Мазур	Бромид 1-пентил-4-(п-метоксибензилиденамино)-1,2,4-триазолия, проявляющий спазмолитическую активность
US6420400B1 (en)	2000-04-07	2002-07-16	Kinetek Pharmaceuticals, Inc.	Antiproliferative 1,2,3-thiadiazole compounds
US7022702B2 (en) *	2000-04-07	2006-04-04	Qlt Inc.	Antiproliferative 1,2,3-thiadiazole compounds
CN100357278C (zh) *	2000-12-22	2007-12-26	奥索-麦克尼尔药品公司	作为激酶抑制剂的取代的三唑二胺衍生物
GB0120147D0 (en) *	2001-08-17	2001-10-10	Metris Therapeutics Ltd	Treatment method
MXPA04004802A (es) *	2001-11-21	2004-08-11	Sterix Ltd	Derivados del 1,2,4-triazol que contienen un grupo sulfamato como inhibidores de aromatasa.
GB0127923D0 (en) *	2001-11-21	2002-01-16	Sterix Ltd	Compound
JP2004196795A (ja) *	2002-12-16	2004-07-15	Wyeth	外部寄生虫駆除剤としてのｎ−フェニル−３−シクロプロピルピラゾール−４−カルボニトリル
EP1431292A1 (en) *	2002-12-16	2004-06-23	Laboratoire Theramex	1-N-phenylamino-1H-imidazole derivatives as aromatase inhibitors
AU2011226950B9 (en) *	2003-12-15	2013-04-11	Laboratoire Theramex	1-N-phenyl-amino-1H-imidazole derivatives and pharmaceutical compositions containing them
KR20060123186A (ko) *	2003-12-15	2006-12-01	라보라뚜와르 떼라멕스	1-엔-페닐-아미노-1에이치-이미다졸 유도체 및 이들을포함하는 약학적 조성물
EP1544195A1 (en) *	2003-12-15	2005-06-22	Laboratoire Theramex	1-N-phenyl-amino- 1H-imidazole derivatives and pharmaceutical compositions containing them
GB0411562D0 (en)	2004-05-24	2004-06-23	Sterix Ltd	Compound
EP2450354B1 (en) *	2009-07-03	2016-08-17	Riken	Labeling compound for pet
GB0914767D0 (en) *	2009-08-24	2009-09-30	Sterix Ltd	Compound
CN113387894B (zh) *	2021-06-22	2023-02-24	首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院)	1-n-苯乙腈基氨基-三氮唑和嘧啶衍生物及其制备方法和应用

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2488891A1 (fr) *	1980-08-22	1982-02-26	Roussel Uclaf	Nouveaux derives du 4h-1,2,4-triazole, leur procede de preparation et leur application comme medicament
DE3410700A1 (de) *	1984-03-23	1985-09-26	Basf Ag, 6700 Ludwigshafen	2,4,5-triphenyl-v-triazole und deren verwendung
US4609666A (en) *	1984-06-18	1986-09-02	Eli Lilly And Company	Aromatase inhibiting derivatives of α,α-bis(4-halophenyl)methyltetrazoles and triazoles
US4602025A (en) *	1984-06-18	1986-07-22	Eli Lilly And Company	Aromatase inhibitors
US4661508A (en) *	1984-06-18	1987-04-28	Eli Lilly And Company	Aromatase inhibiting α,α-diphenyl-4(5)imidazole-methanes or -ethanes
US4749713A (en)	1986-03-07	1988-06-07	Ciba-Geigy Corporation	Alpha-heterocycle substituted tolunitriles
CH677925A5 (pt) *	1986-12-03	1991-07-15	Sandoz Ag
US5041458A (en) *	1987-03-20	1991-08-20	E. I. Du Pont De Nemours And Company	Fungicidal aminotriazoles and aminoimidazoles
EP0283245A1 (en) *	1987-03-20	1988-09-21	E.I. Du Pont De Nemours And Company	Fungicidal aminotriazoles and aminoimidazoles
NZ224714A (en) *	1987-06-01	1990-03-27	Janssen Pharmaceutica Nv	Substituted benzotriazole derivatives and pharmaceutical compositions
US4806554A (en) *	1988-01-11	1989-02-21	Hoechst-Roussel Pharmaceuticals, Inc.	Pyrazol and indazolpyridinamines
GR900100380A (el) *	1989-05-20	1991-10-10	Fisons Plc	Μέ?οδος παρασκευής αντι-φλεγμονωδών παραγώγων αμινοφενόλης.

1992
- 1992-08-27 KR KR1019940700682A patent/KR100204697B1/ko not_active Expired - Fee Related
- 1992-08-27 EP EP92918529A patent/EP0641785B1/en not_active Expired - Lifetime
- 1992-08-27 FI FI940988A patent/FI940988L/fi unknown
- 1992-08-27 DE DE69230225T patent/DE69230225T2/de not_active Expired - Fee Related
- 1992-08-27 RU RU94016190/04A patent/RU2124010C1/ru not_active IP Right Cessation
- 1992-08-27 ES ES92918529T patent/ES2139605T3/es not_active Expired - Lifetime
- 1992-08-27 TW TW081106759A patent/TW225526B/zh active
- 1992-08-27 HU HU9400611A patent/HU220863B1/hu not_active IP Right Cessation
- 1992-08-27 US US08/199,180 patent/US5674886A/en not_active Expired - Fee Related
- 1992-08-27 AT AT92918529T patent/ATE186052T1/de not_active IP Right Cessation
- 1992-08-27 CA CA002116773A patent/CA2116773C/en not_active Expired - Fee Related
- 1992-08-27 UA UA94005459A patent/UA41295C2/uk unknown
- 1992-08-27 AU AU24874/92A patent/AU665569B2/en not_active Ceased
- 1992-08-27 WO PCT/JP1992/001089 patent/WO1993005027A1/ja not_active Ceased
- 1992-08-27 RO RO94-00319A patent/RO114129B1/ro unknown
- 1992-08-28 PT PT100821A patent/PT100821B/pt not_active IP Right Cessation
- 1992-08-31 MX MX9204996A patent/MX9204996A/es unknown
- 1992-09-02 CN CN92110016A patent/CN1035817C/zh not_active Expired - Fee Related
1994
- 1994-02-28 BG BG98618A patent/BG61688B1/bg unknown
- 1994-02-28 NO NO940686A patent/NO305284B1/no unknown

Also Published As

Publication number	Publication date
UA41295C2 (uk)	2001-09-17
US5674886A (en)	1997-10-07
PT100821B (pt)	1999-07-30
TW225526B (pt)	1994-06-21
FI940988A7 (fi)	1994-04-05
MX9204996A (es)	1993-08-01
NO305284B1 (no)	1999-05-03
AU2487492A (en)	1993-04-05
FI940988L (fi)	1994-04-05
CA2116773C (en)	2002-12-10
HU9400611D0 (en)	1994-09-28
EP0641785A4 (en)	1994-06-16
EP0641785B1 (en)	1999-10-27
ES2139605T3 (es)	2000-02-16
KR100204697B1 (ko)	1999-06-15
WO1993005027A1 (fr)	1993-03-18
RO114129B1 (ro)	1999-01-29
EP0641785A1 (en)	1995-03-08
BG61688B1 (bg)	1998-03-31
NO940686D0 (no)	1994-02-28
RU2124010C1 (ru)	1998-12-27
CN1069974A (zh)	1993-03-17
DE69230225T2 (de)	2000-05-31
ATE186052T1 (de)	1999-11-15
HUT67249A (en)	1995-03-28
FI940988A0 (fi)	1994-03-02
CA2116773A1 (en)	1993-03-18
CN1035817C (zh)	1997-09-10
AU665569B2 (en)	1996-01-11
BG98618A (bg)	1995-03-31
NO940686L (pt)	1994-04-29
HU220863B1 (en)	2002-06-29
DE69230225D1 (de)	1999-12-02

Publication	Publication Date	Title
PT100821A (pt)	1993-11-30	Compostos amino terciario substituidos com triazolilo e seus sais, e processo para a sua preparacao
MX9202947A (es)	1992-07-01	Compuesto antibacteriano de quinolina.
ATE214055T1 (de)	2002-03-15	Retinoid-potenzierende verbindungen
GB1355631A (en)	1974-06-05	Imidazole derivatives
RU94016190A (ru)	1995-12-10	Триазолилзамещенные третичные аминные соединения и их соли, способ их получения и содержащие их ингибитор ароматазы и фармацевтический состав
MX198902B (en)	2000-10-03	Azole compounds, their production and use
DE69215035D1 (de)	1996-12-12	Zusammensetzung, die Rhodacyanine-Farbstoffen enthält, zur Behandlung von Krebs
DE69324141D1 (de)	1999-04-29	Substituierte tertiäre amine und deren salze
DE69026311D1 (de)	1996-05-09	4-[4-[4-[4-[[2-(2,4-Difluorphenyl)-2-(1H-azolylmethyl)-1,3-dioxolan-4-yl]methoxy]phenyl]-1-piperazinyl]phenyl]triazolone und Imidazolone zur Bekämpfung von Pilzen
GB1264485A (pt)	1972-02-23
GR81836B (pt)	1984-12-12
BR8701541A (pt)	1988-01-26	Composto,composicao fungicida agricola,e processo para preparacao de tal composto
ATE104661T1 (de)	1994-05-15	Thioformamid-derivate.
ES2021476B3 (es)	1991-11-01	Azolilmetilciclopropano y su aplicacion como medio protector de plantas
JPS57106666A (en)	1982-07-02	N-substituted imidazoles
TH18465A (th)	1996-05-09	สารประกอบอาโซล การผลิต และการใช้สารเหล่านี้
BR8903043A (pt)	1990-02-06	Processo para preparacao de compostos
ES348123A1 (es)	1969-03-16	Un procedimiento para la preparacion de derivados de quina-zolina.
TH13545A (th)	1993-12-15	ไนโตรเอธิลีนและไนโตรกัวนิดีนที่เป็นสารฆ่าสัตว์ขาปล้อง
TH382A (th)	1982-06-04	อนุพันธ์ใหม่ของอิมิดาโซล
TH15500A (th)	1995-02-24	สารฆ่าเชื้อราประเภทแอริลพิแรโซล
TH13508A (th)	1993-12-15	สารประกอบสำหรับใช้รักษาโรคที่เกี่ยวข้องกับสิวโคไทรอีน
IT1143792B (it)	1986-10-22	Composizione fungicida

Legal Events

Date	Code	Title	Description
1999-07-30	FG3A	Patent granted, date of granting	Effective date: 19990413
2004-01-30	MM3A	Annulment or lapse	Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20031031

Date

Code

Title

Description

1999-07-30

FG3A

Patent granted, date of granting

Effective date: 19990413

2004-01-30

MM3A

Annulment or lapse

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20031031