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PL376659A1 - Skondensowane związki heterocykliczne - Google Patents

Skondensowane związki heterocykliczne

Info

Publication number
PL376659A1
PL376659A1 PL376659A PL37665903A PL376659A1 PL 376659 A1 PL376659 A1 PL 376659A1 PL 376659 A PL376659 A PL 376659A PL 37665903 A PL37665903 A PL 37665903A PL 376659 A1 PL376659 A1 PL 376659A1
Authority
PL
Poland
Prior art keywords
heterocyclic compounds
fused heterocyclic
fused
compounds
heterocyclic
Prior art date
Application number
PL376659A
Other languages
English (en)
Inventor
Xi Chen
Xiaoqi Chen
Pingchen Fan
Juan Jaen
Leping Li
Jeffrey T. Mihalic
Original Assignee
Tularik Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tularik Inc. filed Critical Tularik Inc.
Publication of PL376659A1 publication Critical patent/PL376659A1/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL376659A 2002-11-06 2003-11-06 Skondensowane związki heterocykliczne PL376659A1 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42445602P 2002-11-06 2002-11-06

Publications (1)

Publication Number Publication Date
PL376659A1 true PL376659A1 (pl) 2006-01-09

Family

ID=32312811

Family Applications (1)

Application Number Title Priority Date Filing Date
PL376659A PL376659A1 (pl) 2002-11-06 2003-11-06 Skondensowane związki heterocykliczne

Country Status (16)

Country Link
US (2) US7253179B2 (pl)
EP (1) EP1562943A1 (pl)
JP (1) JP4547266B2 (pl)
KR (1) KR20050103184A (pl)
CN (2) CN101134757A (pl)
AU (1) AU2003285160B2 (pl)
BR (1) BR0316070A (pl)
CA (1) CA2505372A1 (pl)
EA (1) EA009421B1 (pl)
IS (1) IS7833A (pl)
MX (1) MXPA05004739A (pl)
NO (1) NO20052655L (pl)
NZ (1) NZ540328A (pl)
PL (1) PL376659A1 (pl)
WO (1) WO2004043958A1 (pl)
ZA (1) ZA200503654B (pl)

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US6809104B2 (en) * 2001-05-04 2004-10-26 Tularik Inc. Fused heterocyclic compounds
US20070135425A1 (en) * 2001-05-04 2007-06-14 Amgen Inc. Fused heterocyclic compounds
PL376659A1 (pl) * 2002-11-06 2006-01-09 Tularik Inc. Skondensowane związki heterocykliczne
AU2004209505B2 (en) 2003-02-10 2009-07-23 Banyu Pharmaceutical Co., Ltd. Melanin-concentrating hormone receptor antagonists containing piperidine derivatives as the active ingredient
DE102010025663A1 (de) * 2010-06-30 2012-01-05 Karl-Heinz Glüsenkamp Neue beta-Aminoaldehyd-Derivate, Verfahren zu ihrer Herstellung und ihre chemische Verwendung als reaktive Intermediate
MX2013001612A (es) * 2010-08-10 2013-07-05 Abbvie Inc Moduladores de trpv3 novedosos.
WO2012129491A1 (en) 2011-03-24 2012-09-27 Abbott Laboratories Trpv3 modulators
CA2853097A1 (en) * 2011-10-24 2013-05-02 Abbvie Inc. Novel trpv3 modulators
CN106588812B (zh) * 2016-12-07 2019-02-22 烟台大学 一种酰氯制备2,4-二取代噻唑啉类化合物的方法
HRP20250104T1 (hr) 2019-01-14 2025-03-28 Zydus Lifesciences Limited Novi supstituirani derivati sulfonilureje
HUP2200222A1 (hu) 2022-06-17 2023-12-28 Richter Gedeon Nyrt MCHR1 antagonisták a Prader-Willi szindróma kezelésére

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JP3160941B2 (ja) 1991-06-17 2001-04-25 東レ株式会社 カルバゾール誘導体および免疫抑制剤
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JP2001525178A (ja) 1997-12-03 2001-12-11 スミスクライン ビーチャム コーポレーション ヒト11cbスプライス変異体に対するアゴニストおよびアンタゴニストの探索方法
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ATE460163T1 (de) * 2001-04-12 2010-03-15 Pharmacopeia Llc Arly und diaryl piperidinderivate verwendbar als mch-hemmer
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BR0209932A (pt) 2001-05-22 2004-10-13 Neurogen Corp Composto ou sal farmaceuticamente aceitável do mesmo, composição farmacêutica, preparação farmacêutica embalada, métodos para modular ligação de mch a um receptor de mch e de mvc, para alterar a atividade de transdução de sinal de um receptor de mch em uma célula, para tratar uma doença ou distúrbio associado com a ativação de receptor de mch patogênico obesidade e para determinar a presença ou ausência de receptor de mch em uma amostra, e, uso de um composto
US6664273B2 (en) * 2001-11-26 2003-12-16 Schering Corporation Piperidine based MCH antagonists for treatment of obesity and CNS disorders
JP2005532991A (ja) * 2002-01-10 2005-11-04 ニューロジェン・コーポレーション メラニン凝集ホルモン受容体リガンド:置換2−(4−ベンジル−ピペラジン−1−イルメチル)−及び2−(4−ベンジル−ジアゼパン−1−イルメチル)−1h−ベンゾイミダゾールアナログ
PL376659A1 (pl) * 2002-11-06 2006-01-09 Tularik Inc. Skondensowane związki heterocykliczne

Also Published As

Publication number Publication date
CN101134757A (zh) 2008-03-05
AU2003285160A1 (en) 2004-06-03
EA009421B1 (ru) 2007-12-28
US20040147538A1 (en) 2004-07-29
CA2505372A1 (en) 2004-05-27
EA200500770A1 (ru) 2005-12-29
AU2003285160B2 (en) 2009-06-04
JP4547266B2 (ja) 2010-09-22
IS7833A (is) 2005-05-02
EP1562943A1 (en) 2005-08-17
JP2006508130A (ja) 2006-03-09
CN1330651C (zh) 2007-08-08
ZA200503654B (en) 2006-09-27
US7253179B2 (en) 2007-08-07
NO20052655D0 (no) 2005-06-02
KR20050103184A (ko) 2005-10-27
NZ540328A (en) 2008-02-29
MXPA05004739A (es) 2005-08-02
US20080058365A1 (en) 2008-03-06
CN1735613A (zh) 2006-02-15
NO20052655L (no) 2005-07-26
WO2004043958A1 (en) 2004-05-27
BR0316070A (pt) 2005-09-27

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Legal Events

Date Code Title Description
REFS Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)