[go: up one dir, main page]

PL2768807T3 - Sposoby wytwarzania 6-chloro-2,3,4,9-tetrahydro-1H-karbazolo-1-karboksyamidu oraz jego prekursorów - Google Patents

Sposoby wytwarzania 6-chloro-2,3,4,9-tetrahydro-1H-karbazolo-1-karboksyamidu oraz jego prekursorów

Info

Publication number
PL2768807T3
PL2768807T3 PL12783161T PL12783161T PL2768807T3 PL 2768807 T3 PL2768807 T3 PL 2768807T3 PL 12783161 T PL12783161 T PL 12783161T PL 12783161 T PL12783161 T PL 12783161T PL 2768807 T3 PL2768807 T3 PL 2768807T3
Authority
PL
Poland
Prior art keywords
carbazole
carboxamide
tetrahydro
precursors
chloro
Prior art date
Application number
PL12783161T
Other languages
English (en)
Inventor
Enrica Diodato
Katia Marcucci
Russell Thomas
Paul Wiedenau
Martin Rettig
Huw Roberts
Original Assignee
Siena Biotech S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Siena Biotech S.P.A. filed Critical Siena Biotech S.P.A.
Publication of PL2768807T3 publication Critical patent/PL2768807T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/88Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL12783161T 2011-10-20 2012-10-19 Sposoby wytwarzania 6-chloro-2,3,4,9-tetrahydro-1H-karbazolo-1-karboksyamidu oraz jego prekursorów PL2768807T3 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP11185959 2011-10-20

Publications (1)

Publication Number Publication Date
PL2768807T3 true PL2768807T3 (pl) 2017-03-31

Family

ID=47143859

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12783161T PL2768807T3 (pl) 2011-10-20 2012-10-19 Sposoby wytwarzania 6-chloro-2,3,4,9-tetrahydro-1H-karbazolo-1-karboksyamidu oraz jego prekursorów

Country Status (16)

Country Link
US (2) US20140303382A1 (pl)
EP (1) EP2768807B1 (pl)
JP (1) JP6142459B2 (pl)
CN (1) CN103958467B (pl)
AR (1) AR088377A1 (pl)
AU (1) AU2012324824B2 (pl)
BR (1) BR112014009297A2 (pl)
CA (1) CA2852797C (pl)
ES (1) ES2585077T3 (pl)
HR (1) HRP20160918T1 (pl)
HU (1) HUE029282T2 (pl)
IL (1) IL232058A (pl)
PL (1) PL2768807T3 (pl)
PT (1) PT2768807T (pl)
SI (1) SI2768807T1 (pl)
WO (1) WO2013057258A1 (pl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3248174B2 (ja) 1992-10-02 2002-01-21 日本電信電話株式会社 光通信方式
JP3252303B2 (ja) 1993-03-11 2002-02-04 日本電信電話株式会社 光通信方式
GB201312768D0 (en) * 2013-07-17 2013-08-28 Ge Healthcare Ltd Work-up procedure
CN121127455A (zh) 2023-05-16 2025-12-12 Aop奥尔芬知识产权公司 晶体形式的(s)-6-氯-2,3,4,9-四氢-1h-咔唑-1-甲酰胺的新型多晶型物
AR132691A1 (es) 2023-05-16 2025-07-23 Aop Orphan Ip Ag Preparación de (s)-6-cloro-2,3,4,9-tetrahidro-1h-carbazol-1-carboxamida en forma enantioméricamente enriquecida mediante proceso de resolución
CN120118019A (zh) * 2023-12-08 2025-06-10 苏州湃芮生物科技有限公司 一种RNA m6A调控剂的共晶形式及其制备方法与应用
CN120136769A (zh) * 2023-12-11 2025-06-13 苏州湃芮生物科技有限公司 一种RNA m6A调控剂的结晶形式及其制备方法与应用

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3769298A (en) * 1971-04-02 1973-10-30 Pfizer Substituted aminomethylcarbazoles
US4057640A (en) * 1973-07-18 1977-11-08 Schering Aktiengesellschaft 5,6,7,8:Tetrahydrocarbazole-1-carboxylic acid derivatives
DE2337154C2 (de) * 1973-07-18 1986-04-24 Schering AG, 1000 Berlin und 4709 Bergkamen Neue Carbazolderivate
BG25793A3 (bg) 1973-07-18 1978-12-12 Schering Aktiengesellschaft Метод за получаване на карбазолови деривати
DE2431292A1 (de) * 1974-06-27 1976-01-15 Schering Ag Neue carbazol-derivate
US3907054A (en) 1974-06-13 1975-09-23 Caterpillar Tractor Co Diagonal brace bearing for crawler-type tractors
GB1504707A (en) 1974-08-07 1978-03-22 Bellon Labor Sa Roger 1-aryl-2-oxo-2,4,5,6,7,7a-hexahydroindoles
DZ2769A1 (fr) 1998-04-17 2003-12-01 Lilly Co Eli Composés tricycliques substitués.
DZ2770A1 (fr) 1998-04-17 2003-12-01 Lilly Co Eli Procédé de préparation de 1h-indol-3 glyoxamides substituées en position 4.
AR038136A1 (es) * 2002-01-24 2004-12-29 Merck Frosst Canada Inc Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento
AU2003296405A1 (en) 2003-01-06 2004-08-10 Eli Lilly And Company Fused heterocyclic derivatives as ppar modulators
FR2849811B1 (fr) 2003-01-10 2006-01-21 Renault Sas Systeme de controle longitudinal pour le maintien a l'arret d'un vehicule equipe d'une boite de vitesses automatique
CA2538759C (en) * 2003-09-12 2015-11-03 Elixir Pharmaceuticals, Inc. Substituted heterocyclic compounds as sirtuin inhitibitors
US20060074124A1 (en) * 2003-09-12 2006-04-06 Andrew Napper Methods of treating a disorder
US7534264B2 (en) 2004-01-28 2009-05-19 Ultradent Products, Inc. Delivery system for bone growth promoting material
AU2005208934A1 (en) * 2004-01-29 2005-08-11 Elixir Pharmaceuticals, Inc Treating a viral disorder
US7104702B2 (en) 2004-03-24 2006-09-12 Corning Cable Systems Llc Field installable optical fiber connector
US20060003065A1 (en) 2004-07-01 2006-01-05 Kateman Paul R Dry-base aerated food product dispensing method and apparatus
CA2588607A1 (en) * 2004-11-23 2006-06-01 Ptc Therapeutics, Inc. Carbazole, carboline and indole derivatives useful in the inhibition of vegf production
EP1856126A2 (en) * 2005-02-17 2007-11-21 Wyeth a Corporation of the State of Delaware Cycloalkylfused indole, benzothiophene, benzofuran and indene derivatives
WO2006099245A1 (en) * 2005-03-11 2006-09-21 Elixir Pharmaceuticals, Inc. Sirt inhibitors that bind to nad
WO2007047604A2 (en) * 2005-10-18 2007-04-26 Elixir Pharmaceuticals, Inc. Sirt1 inhibition
DE102006029320B3 (de) * 2006-06-23 2007-10-11 Röhm Gmbh Verfahren zur kontinuierlichen Herstellung von ungesättigten Carbonsäureanhydriden
WO2008019825A1 (en) * 2006-08-14 2008-02-21 Santhera Pharmaceuticals (Schweiz) Ag Use of tricyclic indole derivatives for the treatment of muscular diseases

Also Published As

Publication number Publication date
CN103958467B (zh) 2016-10-12
AU2012324824B2 (en) 2016-08-11
ES2585077T3 (es) 2016-10-03
AU2012324824A1 (en) 2014-05-08
US10329254B2 (en) 2019-06-25
JP6142459B2 (ja) 2017-06-07
JP2014530839A (ja) 2014-11-20
BR112014009297A2 (pt) 2017-04-11
IL232058A (en) 2016-02-29
HRP20160918T1 (hr) 2016-09-23
HK1200452A1 (en) 2015-08-07
AR088377A1 (es) 2014-05-28
HUE029282T2 (en) 2017-02-28
EP2768807A1 (en) 2014-08-27
CA2852797C (en) 2020-02-04
US20140303382A1 (en) 2014-10-09
WO2013057258A1 (en) 2013-04-25
CA2852797A1 (en) 2013-04-25
US20160304455A1 (en) 2016-10-20
IL232058A0 (en) 2014-05-28
PT2768807T (pt) 2016-08-08
CN103958467A (zh) 2014-07-30
EP2768807B1 (en) 2016-05-04
SI2768807T1 (sl) 2016-09-30

Similar Documents

Publication Publication Date Title
IL269322B (en) Methylphenidate-medications, processes for their preparation and use
PL2791093T3 (pl) Sposób wytwarzania 2,3,3,3-tetrafluoropropenu
PT2678332T (pt) Derivados de diaminopirimidina e processos para a preparação dos mesmos
IL232058A0 (en) Processes for the preparation of 6 - chloro - 2, 3, 4, 9 - tetrahydro - 1h - carbazole - 1 - carboxamide and its starting materials
SG11201400939YA (en) Process for the preparation of methoxymelonal
PL2901857T3 (pl) Sposób wytwarzania 3-chloro-4,5,6-trifluoro-pikolinonitrylu
EP2596007A4 (en) PROCESS FOR THE PREPARATION OF 17-DEOXY-CORTICOSTEROIDS
PL2603494T3 (pl) Sposób wytwarzania 3-haloalkilopirazoli
PT2702045T (pt) Método inovador para a preparação de etravirina
PL391776A1 (pl) Związki luminescencyjne, sposób wytwarzania związków luminescencyjnych oraz ich zastosowanie
PL398018A1 (pl) Nowa diacylo-sn-glicero-3-fosfocholina oraz sposób jej otrzymywania
PL398021A1 (pl) Nowa diacylo-sn-glicero-3-fosfocholina oraz sposób jej otrzymywania
PL2598504T3 (pl) Sposób otrzymywania dimiracetamu
PL390553A1 (pl) Sposób otrzymywania 1,2-epoksybutan-3-olu
PL392489A1 (pl) Sposób wytwarzania 3ß,7α-dihydroksy-5α-androst-17-onu
PL390554A1 (pl) Sposób otrzymywania 2,3-epoksybutan-1-olu
PL395184A1 (pl) Nowe pochodne benzimidazolu, sposób wytwarzania i zastosowanie pochodnych benzimidazolu
PL395175A1 (pl) Nowe pochodne dekstrometorfanu i sposób ich wytwarzania
PL396232A1 (pl) Surfaktanty kationowe, pochodne N,N-dimetylotrimetylenodiaminy oraz sposób wytwarzania surfaktantów kationowych N,N-dimetylotrimetylenodiaminy
PL396024A1 (pl) Sposób wytwarzania 4,2',4' -trihydroksy-6'-metoksy-3'-prenylo-α,ß-dihydrochalkonu
PL399423A1 (pl) Sposób wytwarzania 2'-hydroksydihydrochalkonu
PL399422A1 (pl) Sposób wytwarzania 2',4,4',6'-tetrahydroksydihydrochalkonu
PL398695A1 (pl) Sposób wytwarzania 2'-hydroksydihydrochalkonu
PL398984A1 (pl) Sposób wytwarzania (Z)-6,4'-dihydroksy-4-metoksy-7- prenyloauronu
GB201019078D0 (en) Process for the preparation of rosuvastatin