PL2406253T3 - Pochodne benzofuranylu jako inhibitory glukokinazy - Google Patents
Pochodne benzofuranylu jako inhibitory glukokinazyInfo
- Publication number
- PL2406253T3 PL2406253T3 PL10708644T PL10708644T PL2406253T3 PL 2406253 T3 PL2406253 T3 PL 2406253T3 PL 10708644 T PL10708644 T PL 10708644T PL 10708644 T PL10708644 T PL 10708644T PL 2406253 T3 PL2406253 T3 PL 2406253T3
- Authority
- PL
- Poland
- Prior art keywords
- derivatives used
- glucokinase inhibitors
- benzofuranyl derivatives
- benzofuranyl
- glucokinase
- Prior art date
Links
- 102000030595 Glucokinase Human genes 0.000 title 1
- 108010021582 Glucokinase Proteins 0.000 title 1
- 125000000499 benzofuranyl group Chemical group O1C(=CC2=C1C=CC=C2)* 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US15909909P | 2009-03-11 | 2009-03-11 | |
| PCT/IB2010/050943 WO2010103437A1 (en) | 2009-03-11 | 2010-03-04 | Benzofuranyl derivatives used as glucokinase inhibitors |
| EP10708644.9A EP2406253B1 (en) | 2009-03-11 | 2010-03-04 | Benzofuranyl derivatives used as glucokinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL2406253T3 true PL2406253T3 (pl) | 2013-10-31 |
Family
ID=42124287
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL10708644T PL2406253T3 (pl) | 2009-03-11 | 2010-03-04 | Pochodne benzofuranylu jako inhibitory glukokinazy |
Country Status (37)
| Country | Link |
|---|---|
| US (2) | US8455496B2 (pl) |
| EP (2) | EP2406253B1 (pl) |
| JP (1) | JP5086480B2 (pl) |
| KR (1) | KR101295937B1 (pl) |
| CN (1) | CN102388038B (pl) |
| AP (1) | AP3179A (pl) |
| AR (1) | AR075729A1 (pl) |
| AU (1) | AU2010222589B2 (pl) |
| BR (1) | BRPI1013246B1 (pl) |
| CA (1) | CA2754681C (pl) |
| CL (1) | CL2011002185A1 (pl) |
| CO (1) | CO6430427A2 (pl) |
| CR (1) | CR20110467A (pl) |
| CU (1) | CU24036B1 (pl) |
| DK (1) | DK2406253T3 (pl) |
| DO (1) | DOP2011000279A (pl) |
| EA (1) | EA018894B1 (pl) |
| EC (1) | ECSP11011306A (pl) |
| ES (1) | ES2427279T3 (pl) |
| GE (1) | GEP20156239B (pl) |
| HR (1) | HRP20130661T1 (pl) |
| IL (1) | IL214942A (pl) |
| MA (1) | MA33119B1 (pl) |
| MY (1) | MY151246A (pl) |
| NI (1) | NI201100166A (pl) |
| NZ (1) | NZ595024A (pl) |
| PE (1) | PE20120668A1 (pl) |
| PL (1) | PL2406253T3 (pl) |
| PT (1) | PT2406253E (pl) |
| RS (1) | RS52903B (pl) |
| SI (1) | SI2406253T1 (pl) |
| TN (1) | TN2011000454A1 (pl) |
| TW (1) | TWI383981B (pl) |
| UA (1) | UA99882C2 (pl) |
| UY (1) | UY32480A (pl) |
| WO (1) | WO2010103437A1 (pl) |
| ZA (1) | ZA201106632B (pl) |
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