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PL2193131T3 - Związki imidazo[1,2-a]pirazyny w leczeniu infekcji wirusowych takich jak zapalenia wątroby - Google Patents

Związki imidazo[1,2-a]pirazyny w leczeniu infekcji wirusowych takich jak zapalenia wątroby

Info

Publication number
PL2193131T3
PL2193131T3 PL08787346T PL08787346T PL2193131T3 PL 2193131 T3 PL2193131 T3 PL 2193131T3 PL 08787346 T PL08787346 T PL 08787346T PL 08787346 T PL08787346 T PL 08787346T PL 2193131 T3 PL2193131 T3 PL 2193131T3
Authority
PL
Poland
Prior art keywords
imidazo
hepatitis
treatment
viral infections
pyrazine compounds
Prior art date
Application number
PL08787346T
Other languages
English (en)
Inventor
Angus Macleod
Dale Robert Mitchell
Nicholas John Palmer
Christophe Claude Parsy
Michael Daniel Goldsmith
Clifford John Harris
Original Assignee
Biofocus Dpi Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biofocus Dpi Ltd filed Critical Biofocus Dpi Ltd
Publication of PL2193131T3 publication Critical patent/PL2193131T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
PL08787346T 2007-08-21 2008-08-20 Związki imidazo[1,2-a]pirazyny w leczeniu infekcji wirusowych takich jak zapalenia wątroby PL2193131T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0716292.8A GB0716292D0 (en) 2007-08-21 2007-08-21 Imidazopyrazine compounds
PCT/EP2008/060896 WO2009024585A2 (en) 2007-08-21 2008-08-20 Imidazo [1,2-a] pyrazine compounds for treatment of viral infections such as hepatitis
EP08787346A EP2193131B1 (en) 2007-08-21 2008-08-20 Imidazo[1,2-a]pyrazine compounds for treatment of viral infections such as hepatitis

Publications (1)

Publication Number Publication Date
PL2193131T3 true PL2193131T3 (pl) 2013-07-31

Family

ID=38566736

Family Applications (1)

Application Number Title Priority Date Filing Date
PL08787346T PL2193131T3 (pl) 2007-08-21 2008-08-20 Związki imidazo[1,2-a]pirazyny w leczeniu infekcji wirusowych takich jak zapalenia wątroby

Country Status (20)

Country Link
US (1) US8362018B2 (pl)
EP (2) EP2567960A3 (pl)
JP (1) JP2010536825A (pl)
KR (1) KR20100081294A (pl)
CN (1) CN101835780B (pl)
AU (1) AU2008290531A1 (pl)
BR (1) BRPI0815717A2 (pl)
CA (1) CA2707521A1 (pl)
CY (1) CY1113872T1 (pl)
DK (1) DK2193131T3 (pl)
ES (1) ES2404415T3 (pl)
GB (1) GB0716292D0 (pl)
HR (1) HRP20130202T1 (pl)
MX (1) MX2010001733A (pl)
NZ (1) NZ584108A (pl)
PL (1) PL2193131T3 (pl)
PT (1) PT2193131E (pl)
SI (1) SI2193131T1 (pl)
WO (1) WO2009024585A2 (pl)
ZA (1) ZA201002009B (pl)

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CN104411314B (zh) 2012-07-09 2017-10-20 詹森药业有限公司 磷酸二酯酶10的抑制剂
WO2016130501A1 (en) 2015-02-09 2016-08-18 Incyte Corporation Aza-heteroaryl compounds as pi3k-gamma inhibitors
JP6800885B2 (ja) * 2015-04-29 2020-12-16 ヤンセン ファーマシューティカ エヌ.ベー. イミダゾピラジン及びピラゾロピリミジン、並びにampa受容体調節物質としてのこれらの使用
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JP6507976B2 (ja) * 2015-09-30 2019-05-08 東レ株式会社 イミダゾール−2−カルボン酸エステル誘導体又はその塩の製造方法
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BR112020007593A2 (pt) 2017-10-18 2020-09-24 Incyte Corporation derivados de imidazol condensados substituídos por grupos hidróxi terciários como inibidores de pi3k-gama
BR112020014431A2 (pt) 2018-01-17 2020-12-01 Glaxosmithkline Intellectual Property Development Limited inibidores de pl4kiiibeta
TWI811428B (zh) 2018-08-21 2023-08-11 日商杏林製藥股份有限公司 雙環雜芳香環衍生物
CR20250050A (es) 2018-09-05 2025-03-19 Incyte Corp Formas cristalinas de un inhibidor de fosfoinositida 3–quinasa (pi3k) (divisional 2021-0165)
CN109369545B (zh) * 2018-12-14 2020-04-10 东营曜康医药科技有限公司 2-甲基-5-甲酸吡嗪的合成工艺
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CN113929633A (zh) * 2021-10-27 2022-01-14 山东大学 一种法匹拉韦的合成方法及其应用
CN113831255B (zh) * 2021-11-25 2022-03-11 山东诚创蓝海医药科技有限公司 一种2-氨基丙二酰胺的制备方法
CN115489188B (zh) * 2022-10-09 2023-08-29 安徽国风新材料股份有限公司 一种家居保护用聚酯薄膜及其制备方法
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Also Published As

Publication number Publication date
US8362018B2 (en) 2013-01-29
ES2404415T3 (es) 2013-05-27
HRP20130202T1 (hr) 2013-04-30
EP2193131B1 (en) 2013-01-30
US20110166147A1 (en) 2011-07-07
WO2009024585A3 (en) 2009-08-06
GB0716292D0 (en) 2007-09-26
CA2707521A1 (en) 2009-02-26
WO2009024585A2 (en) 2009-02-26
KR20100081294A (ko) 2010-07-14
EP2193131A2 (en) 2010-06-09
DK2193131T3 (da) 2013-04-22
PT2193131E (pt) 2013-04-04
HK1143810A1 (en) 2011-01-14
AU2008290531A1 (en) 2009-02-26
SI2193131T1 (sl) 2013-06-28
NZ584108A (en) 2012-06-29
MX2010001733A (es) 2010-07-06
JP2010536825A (ja) 2010-12-02
CN101835780A (zh) 2010-09-15
ZA201002009B (en) 2010-12-29
BRPI0815717A2 (pt) 2015-02-10
CN101835780B (zh) 2013-09-18
EP2567960A2 (en) 2013-03-13
EP2567960A3 (en) 2013-06-05
CY1113872T1 (el) 2016-07-27

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