PL1989217T3 - 11-fosforowe pochodne steroidowe użyteczne jako modulatory receptora progesteronu - Google Patents

11-fosforowe pochodne steroidowe użyteczne jako modulatory receptora progesteronu

Info

Publication number: PL1989217T3
Authority: PL; Poland
Prior art keywords: receptor modulators; progesterone receptor; derivatives useful; steroid derivatives; phosphorous
Prior art date: 2006-02-17

Application number

PL07757084T

Other languages

English (en)

Other versions

PL1989217T4 (pl

Inventor

Weiqin Jiang

Zhihua Sui

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-02-17

Filing date

2007-02-16

Publication date

2012-11-30

2007-02-16 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2012-11-30 Publication of PL1989217T3 publication Critical patent/PL1989217T3/pl

2013-02-28 Publication of PL1989217T4 publication Critical patent/PL1989217T4/pl

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Gynecology & Obstetrics (AREA)
Emergency Medicine (AREA)
Hematology (AREA)
Obesity (AREA)
Pregnancy & Childbirth (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)

PL07757084T 2006-02-17 2007-02-16 11-fosforowe pochodne steroidowe użyteczne jako modulatory receptora progesteronu PL1989217T4 (pl)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US77473506P	2006-02-17	2006-02-17
EP07757084A EP1989217B1 (en)	2006-02-17	2007-02-16	11-phosphorous steroid derivatives useful as progesterone receptor modulators
PCT/US2007/062272 WO2007098381A2 (en)	2006-02-17	2007-02-16	11-phosphorous steroid derivatives useful as progesterone receptor modulators

Publications (2)

Publication Number	Publication Date
PL1989217T3 true PL1989217T3 (pl)	2012-11-30
PL1989217T4 PL1989217T4 (pl)	2013-02-28

Family

ID=38438062

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL07757084T PL1989217T4 (pl)	2006-02-17	2007-02-16	11-fosforowe pochodne steroidowe użyteczne jako modulatory receptora progesteronu

Country Status (13)

Country	Link
US (1)	US7678781B2 (pl)
EP (1)	EP1989217B1 (pl)
JP (1)	JP5230449B2 (pl)
CN (1)	CN101415720B (pl)
AU (1)	AU2007217094A1 (pl)
CA (1)	CA2642829A1 (pl)
CY (1)	CY1113146T1 (pl)
DK (1)	DK1989217T5 (pl)
ES (1)	ES2388752T3 (pl)
PL (1)	PL1989217T4 (pl)
PT (1)	PT1989217E (pl)
SI (1)	SI1989217T1 (pl)
WO (1)	WO2007098381A2 (pl)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2680119A1 (en) *	2007-03-07	2008-09-12	Janssen Pharmaceutica N.V.	Steroids derivatives as selective progesterone receptor modulators
CN101926806A (zh) *	2009-06-24	2010-12-29	天津金耀集团有限公司	一种17磷类雌甾化合物在制备紧急避孕药物中的应用
CN102617691B (zh) *	2012-01-18	2014-05-14	上海新华联制药有限公司	一种改进的米非司酮中间体制备方法
WO2014060888A1 (en)	2012-10-18	2014-04-24	Lupin Limited	Novel process and intermediate for preparation of ulipristal
RU2017112748A (ru)	2014-11-17	2018-12-19	Арно Терапьютикс, Инк.	Композиции онапристона пролонгированного действия и способы
US10308676B2 (en)	2015-09-25	2019-06-04	Context Biopharma Inc.	Methods of making onapristone intermediates
CN108883067B (zh)	2015-12-15	2021-03-09	康特斯生物制药公司	非晶奥那司酮组合物及其制备方法
WO2018102369A1 (en)	2016-11-30	2018-06-07	Arno Therapeutics, Inc.	Methods for onapristone synthesis dehydration and deprotection
WO2023000135A1 (en) *	2021-07-19	2023-01-26	Context Biopharma Inc.	Processes of making onapristone and intermediates thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9003939D0 (en) *	1990-02-21	1990-04-18	Imperial College	Sulphatase inhibitors
ZA929315B (en) *	1991-12-20	1993-05-24	Akzo Nv	17-spirofuran-3'-ylidene steroids.
CA2100514C (en) *	1992-07-29	2005-03-29	Johannes A. M. Hamersma	17-spiromethylene steroids
JPH0995496A (ja) *	1995-09-28	1997-04-08	Kaken Pharmaceut Co Ltd	ウルソデオキシコール酸誘導体
PT1448592E (pt) *	2001-10-18	2006-07-31	Sterix Ltd	Compostos esteroides para inibicao da esteroide sulfatase
EP1989218B1 (en) *	2006-02-17	2009-12-30	Janssen Pharmaceutica, N.V.	17-phosphorous steroid derivatives useful as progesterone receptor modulators

2007
- 2007-02-16 PL PL07757084T patent/PL1989217T4/pl unknown
- 2007-02-16 US US11/675,647 patent/US7678781B2/en not_active Expired - Fee Related
- 2007-02-16 AU AU2007217094A patent/AU2007217094A1/en not_active Abandoned
- 2007-02-16 JP JP2008555503A patent/JP5230449B2/ja not_active Expired - Fee Related
- 2007-02-16 EP EP07757084A patent/EP1989217B1/en not_active Not-in-force
- 2007-02-16 SI SI200730988T patent/SI1989217T1/sl unknown
- 2007-02-16 CN CN2007800123141A patent/CN101415720B/zh not_active Expired - Fee Related
- 2007-02-16 DK DK07757084.4T patent/DK1989217T5/da active
- 2007-02-16 CA CA002642829A patent/CA2642829A1/en not_active Abandoned
- 2007-02-16 ES ES07757084T patent/ES2388752T3/es active Active
- 2007-02-16 PT PT07757084T patent/PT1989217E/pt unknown
- 2007-02-16 WO PCT/US2007/062272 patent/WO2007098381A2/en not_active Ceased
2012
- 2012-09-25 CY CY20121100875T patent/CY1113146T1/el unknown

Also Published As

Publication number	Publication date
CN101415720B (zh)	2011-10-05
WO2007098381A2 (en)	2007-08-30
PL1989217T4 (pl)	2013-02-28
EP1989217A2 (en)	2008-11-12
JP5230449B2 (ja)	2013-07-10
ES2388752T3 (es)	2012-10-18
CN101415720A (zh)	2009-04-22
PT1989217E (pt)	2012-08-30
WO2007098381A3 (en)	2008-01-03
DK1989217T3 (da)	2012-10-08
JP2009527489A (ja)	2009-07-30
SI1989217T1 (sl)	2012-09-28
US20070232570A1 (en)	2007-10-04
CY1113146T1 (el)	2016-04-13
US7678781B2 (en)	2010-03-16
AU2007217094A1 (en)	2007-08-30
HK1131396A1 (en)	2010-01-22
HK1125652A1 (en)	2009-08-14
DK1989217T5 (da)	2013-01-14
CA2642829A1 (en)	2007-08-30
EP1989217B1 (en)	2012-06-27

Publication	Publication Date	Title
ZA200904150B (en)	2010-11-24	Progesterone receptor antagonists
HRP20130374T1 (en)	2013-05-31	Pyrrolidin-2-one derivatives as androgen receptor modulators
ZA200903096B (en)	2010-07-28	Tetrahydrocyclopenta[b] indole compounds as androgen receptor modulators
SI1989217T1 (sl)	2012-09-28	11-fosforni steroidni derivati, uporabni kot modulatorji progesteronskega receptorja
IL191710A0 (en)	2009-09-22	Glucocorticoid receptor modulators as antiinflammatory agents
PL2564900T3 (pl)	2015-10-30	Steroidy C-19 do zastosowań terapeutycznych
IL184374A0 (en)	2007-10-31	Non steroidal glucocorticoid receptor modulators
ZA200800689B (en)	2009-07-29	Benzofuranone derivatives as nonsteroidal progesterone receptor modulators
ATE478078T1 (de)	2010-09-15	Pyridooxazepin-progesteronrezeptor-modulatoren
EP2049104A4 (en)	2009-09-09	PYRROLIDINONE ANILINES AS MODULATORS OF THE PROGESTERONE RECEPTOR
ZA200806237B (en)	2009-05-27	Cannibinoid receptor modulators
PL1991559T3 (pl)	2012-11-30	Pochodne oksy-steroidowe jako selektywne modulatory receptora progesteronu
HK1125945A (en)	2009-08-21	17-phosphorous steroid derivatives useful as progesterone receptor modulators
ZA200907546B (en)	2010-07-28	New progesterone receptor modulators
HK1139393A (en)	2010-09-17	Steroids derivatives as selective progesterone receptor modulators
HK1141515A (en)	2010-11-12	New progesterone receptor modulators
IL178010A0 (en)	2006-12-31	Progesterone receptor modulators
HK1122811A (en)	2009-05-29	Cannibinoid receptor modulators