PL1828196T3 - Stereoselective process and crystalline forms of a camptothecin - Google Patents
Stereoselective process and crystalline forms of a camptothecinInfo
- Publication number
- PL1828196T3 PL1828196T3 PL05849781T PL05849781T PL1828196T3 PL 1828196 T3 PL1828196 T3 PL 1828196T3 PL 05849781 T PL05849781 T PL 05849781T PL 05849781 T PL05849781 T PL 05849781T PL 1828196 T3 PL1828196 T3 PL 1828196T3
- Authority
- PL
- Poland
- Prior art keywords
- camptothecin
- crystalline forms
- stereoselective process
- stereoselective
- crystalline
- Prior art date
Links
- KLWPJMFMVPTNCC-UHFFFAOYSA-N Camptothecin Natural products CCC1(O)C(=O)OCC2=C1C=C3C4Nc5ccccc5C=C4CN3C2=O KLWPJMFMVPTNCC-UHFFFAOYSA-N 0.000 title 1
- VSJKWCGYPAHWDS-FQEVSTJZSA-N camptothecin Chemical compound C1=CC=C2C=C(CN3C4=CC5=C(C3=O)COC(=O)[C@]5(O)CC)C4=NC2=C1 VSJKWCGYPAHWDS-FQEVSTJZSA-N 0.000 title 1
- 229940127093 camptothecin Drugs 0.000 title 1
- VSJKWCGYPAHWDS-UHFFFAOYSA-N dl-camptothecin Natural products C1=CC=C2C=C(CN3C4=CC5=C(C3=O)COC(=O)C5(O)CC)C4=NC2=C1 VSJKWCGYPAHWDS-UHFFFAOYSA-N 0.000 title 1
- 230000000707 stereoselective effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP04030246 | 2004-12-21 | ||
| EP05849781A EP1828196B1 (en) | 2004-12-21 | 2005-12-16 | Stereoselective process and crystalline forms of a camptothecin |
| PCT/EP2005/056849 WO2006067092A2 (en) | 2004-12-21 | 2005-12-16 | Stereoselective process and crystalline forms of a camptothecin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL1828196T3 true PL1828196T3 (en) | 2013-02-28 |
Family
ID=34927884
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL05849781T PL1828196T3 (en) | 2004-12-21 | 2005-12-16 | Stereoselective process and crystalline forms of a camptothecin |
Country Status (18)
| Country | Link |
|---|---|
| US (3) | US7799921B2 (en) |
| EP (1) | EP1828196B1 (en) |
| JP (2) | JP5491699B2 (en) |
| KR (1) | KR101355121B1 (en) |
| CN (1) | CN101084221B (en) |
| AU (1) | AU2005318227B2 (en) |
| BR (1) | BRPI0515832A (en) |
| CA (1) | CA2590756C (en) |
| CY (1) | CY1117243T1 (en) |
| DK (1) | DK1828196T3 (en) |
| ES (1) | ES2395930T3 (en) |
| HR (1) | HRP20120926T1 (en) |
| ME (1) | ME01495B (en) |
| PL (1) | PL1828196T3 (en) |
| PT (1) | PT1828196E (en) |
| RS (1) | RS52585B (en) |
| SI (1) | SI1828196T1 (en) |
| WO (1) | WO2006067092A2 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7799921B2 (en) * | 2004-12-21 | 2010-09-21 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Stereoselective process and crystalline forms of a camptothecin |
| ITRM20050418A1 (en) * | 2005-08-04 | 2007-02-05 | Sigma Tau Ind Farmaceuti | IMMEDIATE RELEASE THERAPEUTIC SYSTEMS FOR THE IMPROVED ORAL ABSORPTION OF 7 - [(E) -T-BUTYLOSSIMINOMETHYL] CAMPTOTECIN. |
| FR2938534B1 (en) | 2008-11-14 | 2012-10-26 | Sanofi Aventis | PROCESS FOR THE PREPARATION OF EPLIVANSERIN HEMIFUMARATE |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPH03271278A (en) * | 1990-03-16 | 1991-12-03 | Nissan Chem Ind Ltd | 2-anilinopyrimidine derivative and agricultural and horticultural fungicide |
| JP3046401B2 (en) * | 1991-06-18 | 2000-05-29 | イハラケミカル工業株式会社 | 6- [1- (N-Alkoxyimino) ethyl] salicylic acid derivative and method for producing the same |
| IL106786A (en) * | 1992-09-10 | 1997-02-18 | Basf Ag | Substituted pyridine derivatives and fungicidal compositions containing them |
| DE69901379T2 (en) * | 1999-03-09 | 2002-11-07 | Istituto Nazionale Per Lo Studio E La Cura Dei Tumori, Mailand/Milano | Camptothecin derivatives with anti-tumor effects |
| MXPA04008484A (en) | 2002-03-01 | 2004-12-06 | Pharmacia Italia Spa | Crystalline polymorphic form of irinotecan hydrochloride. |
| US7799921B2 (en) * | 2004-12-21 | 2010-09-21 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Stereoselective process and crystalline forms of a camptothecin |
-
2005
- 2005-12-16 US US11/721,282 patent/US7799921B2/en not_active Expired - Fee Related
- 2005-12-16 SI SI200531610T patent/SI1828196T1/en unknown
- 2005-12-16 JP JP2007547467A patent/JP5491699B2/en not_active Expired - Fee Related
- 2005-12-16 AU AU2005318227A patent/AU2005318227B2/en not_active Ceased
- 2005-12-16 ES ES05849781T patent/ES2395930T3/en active Active
- 2005-12-16 BR BRPI0515832-0A patent/BRPI0515832A/en not_active Application Discontinuation
- 2005-12-16 CA CA2590756A patent/CA2590756C/en not_active Expired - Fee Related
- 2005-12-16 PL PL05849781T patent/PL1828196T3/en unknown
- 2005-12-16 PT PT05849781T patent/PT1828196E/en unknown
- 2005-12-16 DK DK05849781.9T patent/DK1828196T3/en active
- 2005-12-16 KR KR1020077016814A patent/KR101355121B1/en not_active Expired - Fee Related
- 2005-12-16 HR HRP20120926TT patent/HRP20120926T1/en unknown
- 2005-12-16 RS RS20120505A patent/RS52585B/en unknown
- 2005-12-16 WO PCT/EP2005/056849 patent/WO2006067092A2/en not_active Ceased
- 2005-12-16 ME MEP-2012-128A patent/ME01495B/en unknown
- 2005-12-16 CN CN2005800440829A patent/CN101084221B/en active Active
- 2005-12-16 EP EP05849781A patent/EP1828196B1/en active Active
-
2010
- 2010-08-17 US US12/857,743 patent/US8124769B2/en not_active Expired - Fee Related
- 2010-08-17 US US12/857,776 patent/US8101758B2/en not_active Expired - Fee Related
-
2012
- 2012-10-30 CY CY20121101034T patent/CY1117243T1/en unknown
- 2012-11-09 JP JP2012247587A patent/JP5982261B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2590756C (en) | 2014-09-02 |
| CA2590756A1 (en) | 2006-06-29 |
| HRP20120926T1 (en) | 2012-12-31 |
| CN101084221B (en) | 2011-05-11 |
| US20090239893A1 (en) | 2009-09-24 |
| CY1117243T1 (en) | 2017-04-05 |
| BRPI0515832A (en) | 2008-08-05 |
| KR101355121B1 (en) | 2014-01-24 |
| DK1828196T3 (en) | 2012-11-26 |
| PT1828196E (en) | 2012-11-19 |
| SI1828196T1 (en) | 2012-12-31 |
| CN101084221A (en) | 2007-12-05 |
| WO2006067092A2 (en) | 2006-06-29 |
| WO2006067092A3 (en) | 2006-11-02 |
| AU2005318227B2 (en) | 2011-08-18 |
| JP5491699B2 (en) | 2014-05-14 |
| US20100311783A1 (en) | 2010-12-09 |
| EP1828196A2 (en) | 2007-09-05 |
| US8101758B2 (en) | 2012-01-24 |
| EP1828196B1 (en) | 2012-10-17 |
| JP5982261B2 (en) | 2016-08-31 |
| US7799921B2 (en) | 2010-09-21 |
| US8124769B2 (en) | 2012-02-28 |
| KR20070097535A (en) | 2007-10-04 |
| US20100311784A1 (en) | 2010-12-09 |
| JP2008524306A (en) | 2008-07-10 |
| RS52585B (en) | 2013-04-30 |
| AU2005318227A1 (en) | 2006-06-29 |
| JP2013067629A (en) | 2013-04-18 |
| HK1113487A1 (en) | 2008-10-03 |
| ME01495B (en) | 2014-04-20 |
| ES2395930T3 (en) | 2013-02-18 |
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