[go: up one dir, main page]

PE20170304A1 - Composiciones antimicrobianas con agentes efervescentes - Google Patents

Composiciones antimicrobianas con agentes efervescentes

Info

Publication number
PE20170304A1
PE20170304A1 PE2016002748A PE2016002748A PE20170304A1 PE 20170304 A1 PE20170304 A1 PE 20170304A1 PE 2016002748 A PE2016002748 A PE 2016002748A PE 2016002748 A PE2016002748 A PE 2016002748A PE 20170304 A1 PE20170304 A1 PE 20170304A1
Authority
PE
Peru
Prior art keywords
halogen
antimicrobial compositions
effervescent agents
composition
quinolinecarboxylate
Prior art date
Application number
PE2016002748A
Other languages
English (en)
Inventor
Danping Li
Original Assignee
Melinta Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54868661&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20170304(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Melinta Therapeutics Inc filed Critical Melinta Therapeutics Inc
Publication of PE20170304A1 publication Critical patent/PE20170304A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/133Amines having hydroxy groups, e.g. sphingosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Inorganic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Se refiere a una composicion farmaceutica que comprende: a) un derivado de acido quinolona carboxilico de formula I, donde R1 es H o un grupo protector carboxilo; R2 es hidroxilo, entre otros; R3 y R4 son H o halogeno; R5 es halogeno o un grupo amino ciclico saturado opcionalmente sustituido; R6 es H, halogeno, entre otros; X, Y y Z son, independientemente, N, -CH= o -CR7=; con la condicion de que al menos uno de X, Y y Z es N; y W es N o -CR8=; donde un compuesto seleccionado es D-glucitol, 1-desoxi-1-(metilamino), 1-(6- amino-3,5-difluoro- 2-piridinil)-8-cloro-6- fluor-1,4-dihidro-7- (3 -hidroxi-1-azetidinil)-4-oxo-3-quinolincarboxilato y b) un agente efervescente. Dicha composicion tiene tolerabilidad gastrointestinal mejorada y/o menos probabilidad de causar efectos secundarios; siendo util para el tatamiendo de infecciones microbianas
PE2016002748A 2014-06-20 2015-06-19 Composiciones antimicrobianas con agentes efervescentes PE20170304A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201462014786P 2014-06-20 2014-06-20

Publications (1)

Publication Number Publication Date
PE20170304A1 true PE20170304A1 (es) 2017-04-19

Family

ID=54868661

Family Applications (2)

Application Number Title Priority Date Filing Date
PE2016002748A PE20170304A1 (es) 2014-06-20 2015-06-19 Composiciones antimicrobianas con agentes efervescentes
PE2021000031A PE20210927A1 (es) 2014-06-20 2015-06-19 Composiciones antimicrobianas con agentes efervescentes

Family Applications After (1)

Application Number Title Priority Date Filing Date
PE2021000031A PE20210927A1 (es) 2014-06-20 2015-06-19 Composiciones antimicrobianas con agentes efervescentes

Country Status (32)

Country Link
US (2) US20150366857A1 (es)
EP (3) EP3157510B1 (es)
JP (2) JP6995479B2 (es)
CN (2) CN106572982B9 (es)
AR (1) AR100920A1 (es)
AU (3) AU2015276954B2 (es)
BR (1) BR112016029761B1 (es)
CA (1) CA2952950C (es)
CL (2) CL2016003273A1 (es)
CR (2) CR20160592A (es)
CY (2) CY1121995T1 (es)
DK (2) DK3157510T3 (es)
EA (1) EA034152B1 (es)
EC (1) ECSP16095540A (es)
ES (2) ES2732865T3 (es)
HR (2) HRP20191133T1 (es)
HU (2) HUE056298T2 (es)
IL (1) IL249622A0 (es)
LT (2) LT3581180T (es)
MX (2) MX386171B (es)
PE (2) PE20170304A1 (es)
PH (2) PH12022550979A1 (es)
PL (2) PL3581180T3 (es)
PT (2) PT3581180T (es)
RS (2) RS62538B1 (es)
SI (2) SI3157510T1 (es)
SM (2) SMT202100618T1 (es)
SV (1) SV2016005349A (es)
TR (1) TR201909417T4 (es)
TW (2) TWI732337B (es)
UY (1) UY36184A (es)
WO (1) WO2015196027A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022240897A1 (en) * 2021-05-10 2022-11-17 Sepelo Therapeutics, Llc Pharmaceutical composition comprising delafloxacin for administration into the lung

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5194617A (en) * 1988-12-17 1993-03-16 Meiji Seika Kaisha, Ltd. 2,3-disubstituted-4-hydroxyquinoline derivatives
US5223264A (en) * 1989-10-02 1993-06-29 Cima Labs, Inc. Pediatric effervescent dosage form
GB9402203D0 (en) * 1994-02-04 1994-03-30 Smithkline Beecham Plc Pharmaceutical formulation
DE69628466T2 (de) 1995-09-22 2004-04-01 Wakunaga Pharmaceutical Co., Ltd. Zwischenverbindungen zur Herstellung von neunen Pyridoncarbonsäurederivate oder deren Salzen
US6350470B1 (en) * 1998-04-29 2002-02-26 Cima Labs Inc. Effervescent drug delivery system for oral administration
DE19814256A1 (de) * 1998-03-31 1999-10-07 Asta Medica Ag Feste, schnellzerfallende Cetirizin-Formulierungen
IL141977A0 (en) 1998-09-14 2002-03-10 Ranbaxy Lab Ltd Orally administered controlled drug delivery system providing temporal and spatial control
US6187317B1 (en) * 1999-07-14 2001-02-13 Judith Taylor Natural anti-diarrheal composition and method
US6414036B1 (en) * 1999-09-01 2002-07-02 Van Beek Global/Ninkov Llc Composition for treatment of infections of humans and animals
JP2005097116A (ja) 1999-11-11 2005-04-14 Wakunaga Pharmaceut Co Ltd キノリンカルボン酸誘導体アルカリ金属塩及びこれを用いたキノリンカルボン酸誘導体の精製法
WO2003101431A1 (en) * 2002-06-04 2003-12-11 J.B. Chemicals & Pharmaceuticals Ltd. Pharmaceutical composition for controlled drug delivery system
EP2816033A1 (en) 2004-07-30 2014-12-24 Abbvie Inc. Preparation of pyridonecarboxylic acid antibacterials
MX2007004111A (es) * 2004-10-08 2007-06-14 Abbott Lab Sal y formas cristalinas de la misma de un farmaco.
EP2486942B1 (en) * 2004-11-24 2018-10-10 Meda Pharmaceuticals Inc. Compositions comprising azelastine and methods of use thereof
HRP20120502T1 (hr) 2005-04-11 2012-07-31 Abbott@Laboratories Farmaceutske smjese s poboljšanim profilom otapanja za slabo topljive lijekove
DE602005007205D1 (de) 2005-07-19 2008-07-10 Ethypharm Sa Gastroretentive Zusammensetzungen und Verfahren zur Herstellung
US7611739B2 (en) 2006-01-06 2009-11-03 Amerilab Technologies, Inc. Method of using guava extract and composition including guava extract
US20080171158A1 (en) * 2006-08-11 2008-07-17 Aqua Resources Corporation Nanoplatelet copper hydroxides and methods of preparing same
CN1943561A (zh) * 2006-08-23 2007-04-11 北京阜康仁生物制药科技有限公司 普卢利沙星口腔崩解片及其制备方法
PL2124884T3 (pl) 2006-12-22 2020-01-31 Ironwood Pharmaceuticals, Inc. Metody i kompozycje do leczenia zaburzeń przełyku
NZ580972A (en) * 2007-06-04 2012-02-24 Egalet Ltd Controlled release pharmaceutical compositions for prolonged effect
JP6063123B2 (ja) * 2008-11-15 2017-01-18 メリンタ セラピューティクス、インク 抗菌性組成物
WO2010096551A2 (en) * 2009-02-18 2010-08-26 Rib-X Pharmaceuticals, Inc. Antimicrobial compositions
GB201020076D0 (en) * 2010-11-26 2011-01-12 Liverpool School Tropical Medicine Antimalarial compounds
AR084824A1 (es) * 2011-01-10 2013-06-26 Intellikine Inc Procesos para preparar isoquinolinonas y formas solidas de isoquinolinonas
ES2705923T3 (es) * 2011-01-14 2019-03-27 Spero Trinem Inc Formas sólidas de inhibidor de girasa (R)-1-etil-3-[6-fluoro-5-[2-(1-hidroxi-1-metil-etil)pirimidin-5-il]-7-(tetrahidrofuran-2-il)-1H-bencimidazol-2-il]urea
JP2013034468A (ja) * 2011-08-10 2013-02-21 Nisshin Sugar Mfg Co Ltd 発泡成型甘味料
US20140328884A1 (en) * 2011-12-16 2014-11-06 Celanese Eva Performance Polymers, Inc. Controlled release vehicles having desired void volume architectures
CN102697751A (zh) * 2012-05-30 2012-10-03 河南牧翔动物药业有限公司 一种畜禽专用恩诺沙星泡腾分散片及其制备方法

Also Published As

Publication number Publication date
NZ727638A (en) 2023-08-25
PH12022550979A1 (en) 2023-06-26
RS59064B1 (sr) 2019-08-30
CR20160592A (es) 2017-02-21
BR112016029761B1 (pt) 2023-03-07
JP7149991B2 (ja) 2022-10-07
LT3581180T (lt) 2021-12-27
EA034152B1 (ru) 2020-01-09
AU2015276954B2 (en) 2020-07-23
CL2016003273A1 (es) 2017-08-04
AR100920A1 (es) 2016-11-09
HRP20191133T1 (hr) 2019-09-20
TR201909417T4 (tr) 2019-07-22
TWI705814B (zh) 2020-10-01
CN106572982B9 (zh) 2022-07-08
CR20200565A (es) 2021-01-14
AU2015276954A1 (en) 2017-01-12
LT3157510T (lt) 2019-09-25
JP2017518349A (ja) 2017-07-06
JP2020183415A (ja) 2020-11-12
SI3157510T1 (sl) 2019-09-30
CY1121995T1 (el) 2020-10-14
DK3581180T3 (da) 2021-11-08
HUE056298T2 (hu) 2022-02-28
ECSP16095540A (es) 2017-03-31
US20200237744A1 (en) 2020-07-30
EP3157510A1 (en) 2017-04-26
DK3157510T3 (da) 2019-07-01
PL3581180T3 (pl) 2022-02-07
JP6995479B2 (ja) 2022-01-14
BR112016029761A2 (pt) 2017-08-22
ES2897576T3 (es) 2022-03-01
PL3157510T3 (pl) 2019-12-31
US20150366857A1 (en) 2015-12-24
AU2021286284B2 (en) 2024-02-29
CY1125395T1 (el) 2023-03-24
TW201625249A (zh) 2016-07-16
ES2732865T3 (es) 2019-11-26
EP3581180B1 (en) 2021-08-04
MX2016017350A (es) 2017-04-06
PH12016502548B1 (en) 2023-05-24
TW202005650A (zh) 2020-02-01
AU2020256457B2 (en) 2021-09-30
UY36184A (es) 2016-01-29
EP3581180A1 (en) 2019-12-18
CN106572982A (zh) 2017-04-19
PT3581180T (pt) 2021-11-09
CN114831955A (zh) 2022-08-02
SMT202100618T1 (it) 2022-01-10
EP3157510B1 (en) 2019-03-27
PT3157510T (pt) 2019-06-21
HRP20211685T1 (hr) 2022-02-04
AU2021286284A1 (en) 2022-01-06
CN114831955B (zh) 2024-03-12
PE20210927A1 (es) 2021-05-19
CN106572982B (zh) 2022-06-03
CA2952950A1 (en) 2015-12-23
CA2952950C (en) 2023-11-14
RS62538B1 (sr) 2021-12-31
MX386171B (es) 2025-03-18
HUE044764T2 (hu) 2019-11-28
MX2019012608A (es) 2019-12-02
CL2020003153A1 (es) 2021-06-25
WO2015196027A1 (en) 2015-12-23
EA201692532A1 (ru) 2017-05-31
BR112016029761A8 (pt) 2021-06-29
IL249622A0 (en) 2017-02-28
EP3919057A1 (en) 2021-12-08
SMT201900348T1 (it) 2019-09-09
AU2020256457A1 (en) 2020-11-12
EP3157510A4 (en) 2018-02-21
MX368940B (es) 2019-10-21
PH12016502548A1 (en) 2017-04-10
SI3581180T1 (sl) 2021-12-31
SV2016005349A (es) 2017-08-31
TWI732337B (zh) 2021-07-01

Similar Documents

Publication Publication Date Title
CO2019004776A2 (es) Nuevos derivados de quinolina-3-carboxamida antihelmínticos
DOP2020000023A (es) Nuevos derivados de quinolina
MX373678B (es) Composición farmacéutica de clorhidrato de s-cetamina.
EA201690979A1 (ru) Производные азепана и способы лечения инфекций гепатита в
EA201492011A1 (ru) Безводные фармацевтические составы для местного применения
MX2021000189A (es) Compuestos heterociclicos que contienen bencilamina y composiciones utiles contra infeccion por micobacterias.
MX2017012545A (es) Compuestos heterociclicos y su uso en la prevencion o tratamiento de las infecciones bacterianas.
EA201690859A1 (ru) Предотвращение инфекций, вызываемых staphylococcus aureus, гликопротеиновыми вакцинами, синтезированными в escherichia coli
JOP20200004A1 (ar) تركيبات طويلة المفعول
BR112016024235A2 (pt) composições farmacêuticas compreendendo agentes antibacterianos
BR112018074985A2 (pt) composições antibacterianas
MX2019011908A (es) Macrociclos de peptidos anti-bacterianos y uso de los mismos.
MX2017012535A (es) Compuestos hetorociclicos novedosos y su uso en la prevencion o tratamiento de las infecciones bacterianas.
MX2017015812A (es) Formulaciones farmaceuticas inyectables de lefamulina.
MX2017014080A (es) Compuestos heterociclicos y su uso en la prevencion o tratamiento de las infecciones bacterianas.
EA202090750A1 (ru) Производные глюконовой кислоты для применения в лечении и/или предупреждении инфекций, вызываемых микроорганизмами
MX2018016339A (es) Compuestos heterociclicos antiinfecciosos y sus usos.
MX2015010790A (es) Derivados de anilina sustituidos con n-heteroarilo como antivirales de vhc.
PE20170304A1 (es) Composiciones antimicrobianas con agentes efervescentes
BR112016012053A2 (pt) Composições antibacterianas
BR112016024236A2 (pt) composições farmacêuticas compreendendo agentes antibacterianos
EA201692531A1 (ru) Способы лечения инфекций
UA113722C2 (uk) Фармацевтична композиція