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PE20151334A1 - Metodo de produccion de compuestos de piridazinona - Google Patents

Metodo de produccion de compuestos de piridazinona

Info

Publication number
PE20151334A1
PE20151334A1 PE2015001778A PE2015001778A PE20151334A1 PE 20151334 A1 PE20151334 A1 PE 20151334A1 PE 2015001778 A PE2015001778 A PE 2015001778A PE 2015001778 A PE2015001778 A PE 2015001778A PE 20151334 A1 PE20151334 A1 PE 20151334A1
Authority
PE
Peru
Prior art keywords
production
pyridazinone compounds
pyridazinone
compounds
symbol
Prior art date
Application number
PE2015001778A
Other languages
English (en)
Inventor
Naohiro Fukuda
Tomomi Ikemoto
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50272674&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20151334(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of PE20151334A1 publication Critical patent/PE20151334A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Compounds Of Alkaline-Earth Elements, Aluminum Or Rare-Earth Metals (AREA)

Abstract

La presente invencion proporciona un metodo de produccion industrialmente ventajoso de un compuesto piridazinona de formula (I) o (I') en donde cada simbolo es como se describe en la memoria descriptiva
PE2015001778A 2013-02-21 2014-02-20 Metodo de produccion de compuestos de piridazinona PE20151334A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2013032326 2013-02-21

Publications (1)

Publication Number Publication Date
PE20151334A1 true PE20151334A1 (es) 2015-10-14

Family

ID=50272674

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2015001778A PE20151334A1 (es) 2013-02-21 2014-02-20 Metodo de produccion de compuestos de piridazinona

Country Status (27)

Country Link
US (1) US10174004B2 (es)
EP (1) EP2958896B1 (es)
JP (1) JP6364420B2 (es)
KR (1) KR20150119428A (es)
CN (1) CN105189463B (es)
AP (1) AP2015008724A0 (es)
AR (1) AR094717A1 (es)
AU (1) AU2014219665A1 (es)
BR (1) BR112015019942A2 (es)
CA (1) CA2901088C (es)
CL (1) CL2015002286A1 (es)
CR (1) CR20150484A (es)
DO (1) DOP2015000186A (es)
EA (1) EA201591540A1 (es)
EC (1) ECSP15040447A (es)
ES (1) ES2645510T3 (es)
HK (1) HK1219274A1 (es)
IL (1) IL240471A0 (es)
MA (1) MA38427A1 (es)
MX (1) MX2015010940A (es)
PE (1) PE20151334A1 (es)
PH (1) PH12015501840A1 (es)
SG (1) SG11201506302YA (es)
TN (1) TN2015000336A1 (es)
TW (1) TW201444825A (es)
UY (1) UY35341A (es)
WO (1) WO2014129668A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3115B1 (ar) 2011-08-22 2017-09-20 Takeda Pharmaceuticals Co مركبات بيريدازينون واستخدامها كمثبطات daao
EP3856185A1 (en) * 2018-09-28 2021-08-04 Takeda Pharmaceutical Company Limited Balipodect for treating or preventing autism spectrum disorders

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9506382D0 (en) * 1995-03-29 1995-05-17 Boots Co Plc Pharmaceutical compositions
JP5502890B2 (ja) 2008-12-04 2014-05-28 エフ.ホフマン−ラ ロシュ アーゲー ピリダジノン誘導体
BRPI1008498B8 (pt) 2009-02-05 2021-05-25 Takeda Pharmaceuticals Co compostos de piridazinona úteis como inibidores da fosfodiesterase 10a, composição farmacêutica, e, uso de um composto
US9187455B2 (en) * 2009-02-23 2015-11-17 Hoffmann-La Roche Inc. Substituted pyridazines as PDE10A inhibitors
US9090586B2 (en) 2010-08-04 2015-07-28 Takeda Pharmaceutical Company Limited Heterocyclic compound
WO2012018058A1 (ja) 2010-08-04 2012-02-09 武田薬品工業株式会社 縮合複素環化合物
EP2604597B1 (en) 2010-08-10 2017-01-04 Takeda Pharmaceutical Company Limited Heterocyclic compound and use thereof inhibitor of phosphodiesterase 10a
JP6153513B2 (ja) 2011-08-22 2017-06-28 武田薬品工業株式会社 哺乳類中のホスホジエステラーゼ(pde10a)を定量的に画像化する放射性トレーサとしての放射標識された化合物及びその用途

Also Published As

Publication number Publication date
CN105189463A (zh) 2015-12-23
CR20150484A (es) 2015-10-26
ES2645510T3 (es) 2017-12-05
EP2958896B1 (en) 2017-08-30
HK1219274A1 (zh) 2017-03-31
TW201444825A (zh) 2014-12-01
SG11201506302YA (en) 2015-09-29
AP2015008724A0 (en) 2015-09-30
DOP2015000186A (es) 2015-08-31
TN2015000336A1 (en) 2017-01-03
ECSP15040447A (es) 2017-10-31
MA38427A1 (fr) 2018-08-31
CA2901088A1 (en) 2014-08-28
JP2016513070A (ja) 2016-05-12
UY35341A (es) 2014-09-30
MX2015010940A (es) 2015-10-29
WO2014129668A1 (en) 2014-08-28
EA201591540A1 (ru) 2016-01-29
BR112015019942A2 (pt) 2017-07-18
CN105189463B (zh) 2018-05-18
US10174004B2 (en) 2019-01-08
JP6364420B2 (ja) 2018-07-25
IL240471A0 (en) 2015-09-24
US20160002209A1 (en) 2016-01-07
AU2014219665A1 (en) 2015-10-08
CA2901088C (en) 2021-06-29
KR20150119428A (ko) 2015-10-23
PH12015501840A1 (en) 2015-11-09
CL2015002286A1 (es) 2016-02-19
EP2958896A1 (en) 2015-12-30
AR094717A1 (es) 2015-08-19

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Legal Events

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