PE20090358A1 - Composiciones agonistas de dopamina de liberacion controlada - Google Patents
Composiciones agonistas de dopamina de liberacion controladaInfo
- Publication number
- PE20090358A1 PE20090358A1 PE2008000930A PE2008000930A PE20090358A1 PE 20090358 A1 PE20090358 A1 PE 20090358A1 PE 2008000930 A PE2008000930 A PE 2008000930A PE 2008000930 A PE2008000930 A PE 2008000930A PE 20090358 A1 PE20090358 A1 PE 20090358A1
- Authority
- PE
- Peru
- Prior art keywords
- controlled release
- dopamine agonist
- release
- agonist compositions
- release dopamine
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 238000013270 controlled release Methods 0.000 title 1
- 239000003136 dopamine receptor stimulating agent Substances 0.000 title 1
- VYFYYTLLBUKUHU-WTJCDBBSSA-N 4-(2-amino-1,1-ditritioethyl)benzene-1,2-diol Chemical compound NCC([3H])([3H])C1=CC=C(O)C(O)=C1 VYFYYTLLBUKUHU-WTJCDBBSSA-N 0.000 abstract 2
- 208000018737 Parkinson disease Diseases 0.000 abstract 1
- 208000005793 Restless legs syndrome Diseases 0.000 abstract 1
- 239000000556 agonist Substances 0.000 abstract 1
- 239000012729 immediate-release (IR) formulation Substances 0.000 abstract 1
- 239000008203 oral pharmaceutical composition Substances 0.000 abstract 1
- FASDKYOPVNHBLU-ZETCQYMHSA-N pramipexole Chemical compound C1[C@@H](NCCC)CCC2=C1SC(N)=N2 FASDKYOPVNHBLU-ZETCQYMHSA-N 0.000 abstract 1
- 208000019116 sleep disease Diseases 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
REFERIDA A UNA FORMULACION FARMACEUTICA ORAL DE LIBERACION MULTIFASICA QUE COMPRENDE UN PRIMER Y SEGUNDO COMPONENTE QUE SON AGONISTAS DE DOPAMINA, DONDE EL PRIMER COMPONENTE PROPORCIONA UNA LIBERACION INMEDIATA Y EL SEGUNDO COMPONENTE PROPORCIONA UNA LIBERACION MODIFICADA DEL AGONISTA DE DOPAMINA, DONDE EL AGONISTA DE DOPAMINA ES (S)-2-AMINO-4,5,6,7-TETRAHIDRO-6-(PROPILAMINO)BENZOTIAZOL (PRAMIPEXOL). DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE LA ENFERMEDAD DE PARKINSON, SINDROME DE PIERNAS INQUIETAS, TRANSTORNOS DEL SUENO, ENTRE OTROS
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US93327107P | 2007-06-04 | 2007-06-04 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20090358A1 true PE20090358A1 (es) | 2009-04-24 |
Family
ID=40088517
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2008000930A PE20090358A1 (es) | 2007-06-04 | 2008-06-02 | Composiciones agonistas de dopamina de liberacion controlada |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US20080299189A1 (es) |
| AR (1) | AR068792A1 (es) |
| CL (1) | CL2008001622A1 (es) |
| PE (1) | PE20090358A1 (es) |
| WO (1) | WO2008150741A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20120021057A1 (en) * | 2009-04-09 | 2012-01-26 | Purdue Pharma | Once-daily oral ir/cr pramipexole formulation |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7670612B2 (en) * | 2002-04-10 | 2010-03-02 | Innercap Technologies, Inc. | Multi-phase, multi-compartment capsular delivery apparatus and methods for using same |
| US20040166159A1 (en) * | 2002-05-29 | 2004-08-26 | Chien-Hsuan Han | Pharmaceutical dosage forms having immediate and controlled release properties that contain an aromatic amino acid decarboxylase inhibitor and levodopa |
| US20050226926A1 (en) * | 2002-07-25 | 2005-10-13 | Pfizer Inc | Sustained-release tablet composition of pramipexole |
| PA8578501A1 (es) * | 2002-07-25 | 2005-02-04 | Pharmacia Corp | Forma de dosificacion una vez al dia de pramipexol |
| ES2337700T3 (es) * | 2004-02-18 | 2010-04-28 | Sepracor, Inc. | Terapia combinada de agonista de dopamina con sedantes para mejorar la calidad del sueño. |
| US20060182805A1 (en) * | 2005-02-15 | 2006-08-17 | Jazz Pharmaceuticals | Dosage form and method for sustained release of substituted pyrazine compound |
| US20070129329A1 (en) * | 2005-12-02 | 2007-06-07 | Alembic Limited | Stabilized pharmaceutical composition of pramipexole and method of preparation thereof |
-
2008
- 2008-05-23 US US12/126,575 patent/US20080299189A1/en not_active Abandoned
- 2008-05-23 WO PCT/US2008/064772 patent/WO2008150741A1/en not_active Ceased
- 2008-06-02 AR ARP080102321A patent/AR068792A1/es unknown
- 2008-06-02 PE PE2008000930A patent/PE20090358A1/es not_active Application Discontinuation
- 2008-06-04 CL CL200801622A patent/CL2008001622A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR068792A1 (es) | 2009-12-09 |
| CL2008001622A1 (es) | 2008-09-12 |
| US20080299189A1 (en) | 2008-12-04 |
| WO2008150741A1 (en) | 2008-12-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Application declared void or lapsed |