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PE20090358A1 - Composiciones agonistas de dopamina de liberacion controlada - Google Patents

Composiciones agonistas de dopamina de liberacion controlada

Info

Publication number
PE20090358A1
PE20090358A1 PE2008000930A PE2008000930A PE20090358A1 PE 20090358 A1 PE20090358 A1 PE 20090358A1 PE 2008000930 A PE2008000930 A PE 2008000930A PE 2008000930 A PE2008000930 A PE 2008000930A PE 20090358 A1 PE20090358 A1 PE 20090358A1
Authority
PE
Peru
Prior art keywords
controlled release
dopamine agonist
release
agonist compositions
release dopamine
Prior art date
Application number
PE2008000930A
Other languages
English (en)
Inventor
Jonathan David Bortz
Michael N Grimshaw
David Erokoboni
Original Assignee
Drugtech Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Drugtech Corp filed Critical Drugtech Corp
Publication of PE20090358A1 publication Critical patent/PE20090358A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/428Thiazoles condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5084Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

REFERIDA A UNA FORMULACION FARMACEUTICA ORAL DE LIBERACION MULTIFASICA QUE COMPRENDE UN PRIMER Y SEGUNDO COMPONENTE QUE SON AGONISTAS DE DOPAMINA, DONDE EL PRIMER COMPONENTE PROPORCIONA UNA LIBERACION INMEDIATA Y EL SEGUNDO COMPONENTE PROPORCIONA UNA LIBERACION MODIFICADA DEL AGONISTA DE DOPAMINA, DONDE EL AGONISTA DE DOPAMINA ES (S)-2-AMINO-4,5,6,7-TETRAHIDRO-6-(PROPILAMINO)BENZOTIAZOL (PRAMIPEXOL). DICHA COMPOSICION ES UTIL EN EL TRATAMIENTO DE LA ENFERMEDAD DE PARKINSON, SINDROME DE PIERNAS INQUIETAS, TRANSTORNOS DEL SUENO, ENTRE OTROS
PE2008000930A 2007-06-04 2008-06-02 Composiciones agonistas de dopamina de liberacion controlada PE20090358A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US93327107P 2007-06-04 2007-06-04

Publications (1)

Publication Number Publication Date
PE20090358A1 true PE20090358A1 (es) 2009-04-24

Family

ID=40088517

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2008000930A PE20090358A1 (es) 2007-06-04 2008-06-02 Composiciones agonistas de dopamina de liberacion controlada

Country Status (5)

Country Link
US (1) US20080299189A1 (es)
AR (1) AR068792A1 (es)
CL (1) CL2008001622A1 (es)
PE (1) PE20090358A1 (es)
WO (1) WO2008150741A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20120021057A1 (en) * 2009-04-09 2012-01-26 Purdue Pharma Once-daily oral ir/cr pramipexole formulation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7670612B2 (en) * 2002-04-10 2010-03-02 Innercap Technologies, Inc. Multi-phase, multi-compartment capsular delivery apparatus and methods for using same
US20040166159A1 (en) * 2002-05-29 2004-08-26 Chien-Hsuan Han Pharmaceutical dosage forms having immediate and controlled release properties that contain an aromatic amino acid decarboxylase inhibitor and levodopa
US20050226926A1 (en) * 2002-07-25 2005-10-13 Pfizer Inc Sustained-release tablet composition of pramipexole
PA8578501A1 (es) * 2002-07-25 2005-02-04 Pharmacia Corp Forma de dosificacion una vez al dia de pramipexol
ES2337700T3 (es) * 2004-02-18 2010-04-28 Sepracor, Inc. Terapia combinada de agonista de dopamina con sedantes para mejorar la calidad del sueño.
US20060182805A1 (en) * 2005-02-15 2006-08-17 Jazz Pharmaceuticals Dosage form and method for sustained release of substituted pyrazine compound
US20070129329A1 (en) * 2005-12-02 2007-06-07 Alembic Limited Stabilized pharmaceutical composition of pramipexole and method of preparation thereof

Also Published As

Publication number Publication date
AR068792A1 (es) 2009-12-09
CL2008001622A1 (es) 2008-09-12
US20080299189A1 (en) 2008-12-04
WO2008150741A1 (en) 2008-12-11

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Legal Events

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