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PE20090625A1 - Composicion farmaceutica que contiene buprenorfina y nalmefeno - Google Patents

Composicion farmaceutica que contiene buprenorfina y nalmefeno

Info

Publication number
PE20090625A1
PE20090625A1 PE2008000411A PE2008000411A PE20090625A1 PE 20090625 A1 PE20090625 A1 PE 20090625A1 PE 2008000411 A PE2008000411 A PE 2008000411A PE 2008000411 A PE2008000411 A PE 2008000411A PE 20090625 A1 PE20090625 A1 PE 20090625A1
Authority
PE
Peru
Prior art keywords
pharmaceutical composition
composition containing
nalmefene
buprenorphine
containing buprenorphine
Prior art date
Application number
PE2008000411A
Other languages
English (en)
Inventor
Christopher Bourne Chapleo
Neil Hyde
Original Assignee
Reckitt Benckiser Healthcare
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reckitt Benckiser Healthcare filed Critical Reckitt Benckiser Healthcare
Publication of PE20090625A1 publication Critical patent/PE20090625A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36Opioid-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A UNA COMPOSICION ANALGESICA QUE CONTIENE: A) BUPRENORFINA QUE SE ENCUENTRA EN UNA CANTIDAD DE 10uG a 8MG; Y B) NALMEFENO, TAL QUE LA RELACION EN PESO DE BUPRENORFINA A NALMEFENO SE ENCUENTRA EN EL RANGO ENTRE 22,6:1 Y 40:1. SE REFIERE TAMBIEN A UN METODO DE TRATAMIENTO PARA EL DOLOR. DICHA COMPOSICION FARMACEUTICA SE PRESENTA EN UNA FORMA DE DOSIFICACION PARENTERAL UNITARIA O EN UNA FORMA DE DOSIFICACION UNITARIA ADECUADA PARA UNA ADMINISTRACION POR LA MUCOSA O LA DERMIS
PE2008000411A 2007-03-01 2008-02-29 Composicion farmaceutica que contiene buprenorfina y nalmefeno PE20090625A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB0703933A GB2447013A (en) 2007-03-01 2007-03-01 Analgesic composition containing buprenorphone and nalmefene

Publications (1)

Publication Number Publication Date
PE20090625A1 true PE20090625A1 (es) 2009-06-04

Family

ID=37965707

Family Applications (2)

Application Number Title Priority Date Filing Date
PE2012000471A PE20120956A1 (es) 2007-03-01 2008-02-29 Composicion farmaceutica que contiene buprenorfina y nalmefeno
PE2008000411A PE20090625A1 (es) 2007-03-01 2008-02-29 Composicion farmaceutica que contiene buprenorfina y nalmefeno

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PE2012000471A PE20120956A1 (es) 2007-03-01 2008-02-29 Composicion farmaceutica que contiene buprenorfina y nalmefeno

Country Status (21)

Country Link
US (1) US8497280B2 (es)
EP (1) EP2114452B1 (es)
JP (1) JP5577102B2 (es)
KR (1) KR101437461B1 (es)
CN (1) CN101622012B (es)
AR (1) AR065582A1 (es)
AU (1) AU2008220572B2 (es)
BR (1) BRPI0807903A2 (es)
CA (1) CA2678568C (es)
CL (1) CL2008000607A1 (es)
DK (1) DK2114452T3 (es)
ES (1) ES2476865T3 (es)
GB (1) GB2447013A (es)
HR (1) HRP20140591T1 (es)
MX (1) MX2009009134A (es)
PE (2) PE20120956A1 (es)
PL (1) PL2114452T3 (es)
PT (1) PT2114452E (es)
TW (1) TWI468163B (es)
WO (1) WO2008104736A1 (es)
ZA (1) ZA200905692B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA102128C2 (en) * 2008-12-05 2013-06-10 Х. Луннбек А/С Nalmefene hydrochloride dihydrate
HRP20160110T1 (hr) * 2009-05-25 2016-03-11 H. Lundbeck A/S Priprema nalmefen hidroklorida iz naltreksona
CN110101702A (zh) 2012-04-17 2019-08-09 普渡制药公司 用于治疗阿片样物质所致不良药效学响应的系统和方法
CN103637983B (zh) * 2013-12-16 2017-08-04 科贝源(北京)生物医药科技有限公司 一种含有盐酸纳美芬的药物组合物及其制备方法
US9849124B2 (en) 2014-10-17 2017-12-26 Purdue Pharma L.P. Systems and methods for treating an opioid-induced adverse pharmacodynamic response
CN104922061B (zh) * 2015-05-26 2017-09-22 成都天台山制药有限公司 盐酸纳美芬注射液药物组合物和制法
AU2018291397A1 (en) 2017-06-30 2020-01-16 Purdue Pharma L.P. Method of treatment and dosage forms thereof
CA3091443A1 (en) * 2018-02-22 2019-08-29 Avior, Inc. Transmucosal film composition and methods of making and using the same

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8728294D0 (en) * 1987-12-03 1988-01-06 Reckitt & Colmann Prod Ltd Treatment compositions
US5149538A (en) * 1991-06-14 1992-09-22 Warner-Lambert Company Misuse-resistive transdermal opioid dosage form
US5272149A (en) * 1992-05-05 1993-12-21 Stalling Reginald W Symptom controlled receptor substitution for addiction withdrawl
US6096756A (en) * 1992-09-21 2000-08-01 Albert Einstein College Of Medicine Of Yeshiva University Method of simultaneously enhancing analgesic potency and attenuating dependence liability caused by morphine and other bimodally-acting opioid agonists
AU755790B2 (en) * 1997-12-22 2002-12-19 Euro-Celtique S.A. A method of preventing abuse of opioid dosage forms
AR031682A1 (es) * 1999-11-19 2003-10-01 Reckitt Benckiser Helthcare Uk Composiciones farmaceuticas
US20050191340A1 (en) * 2002-08-09 2005-09-01 Gruenenthal Gmbh Opioid-receptor antagonists in transdermal systems having buprenorphine
US9539303B2 (en) * 2006-04-24 2017-01-10 Celgene Corporation Treatment of Ras-expressing tumors
US8957027B2 (en) * 2006-06-08 2015-02-17 Celgene Corporation Deacetylase inhibitor therapy
US20110015168A1 (en) * 2007-01-19 2011-01-20 Mitchell Keegan Methods for increasing levels of human fetal hemoglobin

Also Published As

Publication number Publication date
JP2010520184A (ja) 2010-06-10
KR20090115862A (ko) 2009-11-09
CN101622012B (zh) 2012-05-30
US20100152222A1 (en) 2010-06-17
PE20120956A1 (es) 2012-08-01
GB2447013A (en) 2008-09-03
DK2114452T3 (da) 2014-06-30
PT2114452E (pt) 2014-07-15
MX2009009134A (es) 2009-09-03
CL2008000607A1 (es) 2008-10-03
HK1139868A1 (en) 2010-09-30
US8497280B2 (en) 2013-07-30
WO2008104736A1 (en) 2008-09-04
CN101622012A (zh) 2010-01-06
HRP20140591T1 (hr) 2014-09-12
AU2008220572B2 (en) 2014-03-27
ZA200905692B (en) 2010-10-27
JP5577102B2 (ja) 2014-08-20
KR101437461B1 (ko) 2014-09-05
PL2114452T3 (pl) 2014-09-30
GB0703933D0 (en) 2007-04-11
TWI468163B (zh) 2015-01-11
ES2476865T3 (es) 2014-07-15
CA2678568A1 (en) 2008-09-04
CA2678568C (en) 2015-06-16
EP2114452B1 (en) 2014-04-09
TW200900067A (en) 2009-01-01
BRPI0807903A2 (pt) 2014-06-17
EP2114452A1 (en) 2009-11-11
AR065582A1 (es) 2009-06-17
AU2008220572A1 (en) 2008-09-04

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