PE20050375A1 - COMBINATION OF INHIBITORS OF SEROTONIN RECAPTATION AND INHIBITORS OF NOREPINEPHRINE RECAPTATION - Google Patents
COMBINATION OF INHIBITORS OF SEROTONIN RECAPTATION AND INHIBITORS OF NOREPINEPHRINE RECAPTATIONInfo
- Publication number
- PE20050375A1 PE20050375A1 PE2004000863A PE2004000863A PE20050375A1 PE 20050375 A1 PE20050375 A1 PE 20050375A1 PE 2004000863 A PE2004000863 A PE 2004000863A PE 2004000863 A PE2004000863 A PE 2004000863A PE 20050375 A1 PE20050375 A1 PE 20050375A1
- Authority
- PE
- Peru
- Prior art keywords
- recaptation
- inhibitors
- norepinephrine
- serotonin
- combination
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 2
- QZAYGJVTTNCVMB-UHFFFAOYSA-N serotonin Chemical compound C1=C(O)C=C2C(CCN)=CNC2=C1 QZAYGJVTTNCVMB-UHFFFAOYSA-N 0.000 title 2
- SFLSHLFXELFNJZ-QMMMGPOBSA-N (-)-norepinephrine Chemical compound NC[C@H](O)C1=CC=C(O)C(O)=C1 SFLSHLFXELFNJZ-QMMMGPOBSA-N 0.000 title 1
- 229960002748 norepinephrine Drugs 0.000 title 1
- SFLSHLFXELFNJZ-UHFFFAOYSA-N norepinephrine Natural products NCC(O)C1=CC=C(O)C(O)=C1 SFLSHLFXELFNJZ-UHFFFAOYSA-N 0.000 title 1
- 229940076279 serotonin Drugs 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 206010046543 Urinary incontinence Diseases 0.000 abstract 1
- 230000001800 adrenalinergic effect Effects 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 208000004296 neuralgia Diseases 0.000 abstract 1
- 208000021722 neuropathic pain Diseases 0.000 abstract 1
- 230000000862 serotonergic effect Effects 0.000 abstract 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
REFERIDA A UN COMPUESTO DE FORMULA II DONDE n Y n1 SON CADA UNO 1-3, R Y R1 SON CADA UNO H, HALOGENO, HALO-ALQUILO C1-C6, ENTRE OTROS; A ES H, OR2; R2 ES H, ALQUILO C1-C12; R3 Y R4 SON CADA UNO H, ALQUILO C1-C6; O R3 Y R4 UNIDOS FORMAN UN GRUPO HETEROMONOCICLICO PENTATOMICO O HEXATOMICO. TAMBIEN REFERIDA A UN METODO DE TRATAMIENTO DE POTENCIACION DE LA NEUROTRANSMICION SEROTONERGICA, ADRENERGICA, O AMBAS, EN MAMIFEROS PARA TRASTORNOS TALES COMO DEPRESION, DOLOR NEUROPATICO, INCONTINENCIA URINARIA, ENTRE OTROSREFERRED TO A COMPOUND OF FORMULA II WHERE n AND n1 ARE EACH 1-3, R AND R1 ARE EACH H, HALOGEN, HALO-ALKYL C1-C6, AMONG OTHERS; A IS H, OR2; R2 IS H, C1-C12 ALKYL; R3 AND R4 ARE EACH H, C1-C6 ALKYL; OR R3 AND R4 TOGETHER FORM A HETEROMONOCICLIC PENTATOMIC OR HEXATOMIC GROUP. ALSO REFERRED TO A TREATMENT METHOD TO ENHANCE SEROTONERGIC, ADRENERGIC NEUROTRANSMITION, OR BOTH, IN MAMMALS FOR DISORDERS SUCH AS DEPRESSION, NEUROPATHIC PAIN, URINARY INCONTINENCE, AMONG OTHERS
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US50127503P | 2003-09-09 | 2003-09-09 | |
| US53889804P | 2004-01-23 | 2004-01-23 | |
| US54069604P | 2004-01-30 | 2004-01-30 | |
| US10/769,018 US20050014848A1 (en) | 2002-01-23 | 2004-01-30 | Combination of serotonin reuptake inhibitors and norephinephrine reuptake inhibitors |
| US10/860,721 US20050009927A1 (en) | 2002-01-23 | 2004-06-03 | Combination of serotonin reuptake inhibitors and norepinephrine reuptake inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20050375A1 true PE20050375A1 (en) | 2005-05-30 |
Family
ID=42778435
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2004000863A PE20050375A1 (en) | 2003-09-09 | 2004-09-07 | COMBINATION OF INHIBITORS OF SEROTONIN RECAPTATION AND INHIBITORS OF NOREPINEPHRINE RECAPTATION |
Country Status (2)
| Country | Link |
|---|---|
| AR (1) | AR045612A1 (en) |
| PE (1) | PE20050375A1 (en) |
-
2004
- 2004-09-07 PE PE2004000863A patent/PE20050375A1/en not_active Application Discontinuation
- 2004-09-08 AR ARP040103219 patent/AR045612A1/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR045612A1 (en) | 2005-11-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |