JP5548129B2 - 不斉有機触媒 - Google Patents
不斉有機触媒 Download PDFInfo
- Publication number
- JP5548129B2 JP5548129B2 JP2010525576A JP2010525576A JP5548129B2 JP 5548129 B2 JP5548129 B2 JP 5548129B2 JP 2010525576 A JP2010525576 A JP 2010525576A JP 2010525576 A JP2010525576 A JP 2010525576A JP 5548129 B2 JP5548129 B2 JP 5548129B2
- Authority
- JP
- Japan
- Prior art keywords
- group
- formula
- asymmetric
- added
- carboxylic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- ASFQDNDZFGFMMP-UHFFFAOYSA-N CC(C)(OC1)OCC1=O Chemical compound CC(C)(OC1)OCC1=O ASFQDNDZFGFMMP-UHFFFAOYSA-N 0.000 description 1
- FGFGLSBDAMHTEX-NWDGAFQWSA-N CC(C)(OC1)O[C@@H]([C@H](c(cc2)ccc2[N+]([O-])=O)O)C1=O Chemical compound CC(C)(OC1)O[C@@H]([C@H](c(cc2)ccc2[N+]([O-])=O)O)C1=O FGFGLSBDAMHTEX-NWDGAFQWSA-N 0.000 description 1
- FGFGLSBDAMHTEX-RYUDHWBXSA-N CC(C)(OC1)O[C@H]([C@H](c(cc2)ccc2[N+]([O-])=O)O)C1=O Chemical compound CC(C)(OC1)O[C@H]([C@H](c(cc2)ccc2[N+]([O-])=O)O)C1=O FGFGLSBDAMHTEX-RYUDHWBXSA-N 0.000 description 1
- BXRFQSNOROATLV-UHFFFAOYSA-N [O-][N+](c1ccc(C=O)cc1)=O Chemical compound [O-][N+](c1ccc(C=O)cc1)=O BXRFQSNOROATLV-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/09—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton the carbon skeleton being further substituted by at least two halogen atoms
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
- B01J31/02—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides
- B01J31/04—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides containing carboxylic acids or their salts
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B53/00—Asymmetric syntheses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
- C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C255/56—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and doubly-bound oxygen atoms bound to the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C07C45/72—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction of compounds containing >C = O groups with the same or other compounds containing >C = O groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D319/04—1,3-Dioxanes; Hydrogenated 1,3-dioxanes
- C07D319/06—1,3-Dioxanes; Hydrogenated 1,3-dioxanes not condensed with other rings
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J2231/00—Catalytic reactions performed with catalysts classified in B01J31/00
- B01J2231/30—Addition reactions at carbon centres, i.e. to either C-C or C-X multiple bonds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Catalysts (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010525576A JP5548129B2 (ja) | 2008-08-18 | 2009-08-04 | 不斉有機触媒 |
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2008209411 | 2008-08-18 | ||
| JP2008209411 | 2008-08-18 | ||
| JP2010525576A JP5548129B2 (ja) | 2008-08-18 | 2009-08-04 | 不斉有機触媒 |
| PCT/JP2009/003699 WO2010021093A1 (fr) | 2008-08-18 | 2009-08-04 | Catalyseur organique asymétrique |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2010021093A1 JPWO2010021093A1 (ja) | 2012-01-26 |
| JP5548129B2 true JP5548129B2 (ja) | 2014-07-16 |
Family
ID=41706986
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2010525576A Expired - Fee Related JP5548129B2 (ja) | 2008-08-18 | 2009-08-04 | 不斉有機触媒 |
Country Status (2)
| Country | Link |
|---|---|
| JP (1) | JP5548129B2 (fr) |
| WO (1) | WO2010021093A1 (fr) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2793413C (fr) | 2010-03-19 | 2015-11-24 | Daiichi Sankyo Company, Limited | Forme cristalline d'edoxaban tosylate monohydrate et son procede de fabrication |
| JP5780657B2 (ja) * | 2010-07-02 | 2015-09-16 | 第一三共株式会社 | 光学活性ジアミン誘導体の塩の製造方法 |
| BR112015011574A2 (pt) * | 2012-11-23 | 2017-07-11 | Daiichi Sankyo Co Ltd | processo para produzir um composto |
| WO2014157612A1 (fr) * | 2013-03-29 | 2014-10-02 | 第一三共株式会社 | Procédé de production de (1s,4s,5s)-4-bromo-6- oxabicyclo[3.2.1]octane-7-one |
| CN105017121B (zh) * | 2015-06-09 | 2017-11-21 | 哈尔滨工程大学 | 带有Fmoc‑L‑羟脯氨酸的光学活性苯乙炔衍生物及制备和应用方法 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002275118A (ja) * | 2001-03-15 | 2002-09-25 | Central Glass Co Ltd | アルドール反応生成物の製造方法 |
-
2009
- 2009-08-04 JP JP2010525576A patent/JP5548129B2/ja not_active Expired - Fee Related
- 2009-08-04 WO PCT/JP2009/003699 patent/WO2010021093A1/fr not_active Ceased
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002275118A (ja) * | 2001-03-15 | 2002-09-25 | Central Glass Co Ltd | アルドール反応生成物の製造方法 |
Non-Patent Citations (4)
| Title |
|---|
| JPN6014018257; LUO Sanzhong et al.: 'Highly Enantioselective Direct syn- and anti-Aldol Reacitons of Dihydroxyacetones Catalyzed by Chira' Org. Lett. Vol.10,No.4, 20080221, page.653-656 * |
| JPN6014018258; GUIZZETTI Stefania et al.: 'Enantioselective Direct Aldol Reaction "on Water" Promoted by Chiral Organic Catalysts' Org. Lett. Vol.9,No.7, 20070329, page.1247-1250 * |
| JPN6014018262; NAKADAI Masakazu et al.: 'Diversity-based strategy for discovery of environmentally benign organocatalyst:diamine-protonic aci' Tetrahedron Vol.58,No.41, 20021007, page.8167-8177 * |
| JPN6014018264; NAKAYAMA Keiji et al.: 'Complete Switch of Product Selectivity in Asymmetric Direct Aldol Reaction with Two Different Chiral' J.Am.Chem.Coc Vol.130,No.52, 20081231, page.17666-17667 * |
Also Published As
| Publication number | Publication date |
|---|---|
| JPWO2010021093A1 (ja) | 2012-01-26 |
| WO2010021093A1 (fr) | 2010-02-25 |
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