JO2351B1 - Acylated piperidine derivatives as melanocortin-4 receptor agonists - Google Patents
Acylated piperidine derivatives as melanocortin-4 receptor agonistsInfo
- Publication number
- JO2351B1 JO2351B1 JO200281A JOP20020081A JO2351B1 JO 2351 B1 JO2351 B1 JO 2351B1 JO 200281 A JO200281 A JO 200281A JO P20020081 A JOP20020081 A JO P20020081A JO 2351 B1 JO2351 B1 JO 2351B1
- Authority
- JO
- Jordan
- Prior art keywords
- melanocortin
- piperidine derivatives
- receptor agonists
- acylated piperidine
- acylated
- Prior art date
Links
- 150000003053 piperidines Chemical class 0.000 title abstract 2
- 102000001796 Melanocortin 4 receptors Human genes 0.000 title 1
- 108010021436 Type 4 Melanocortin Receptor Proteins 0.000 title 1
- 239000000018 receptor agonist Substances 0.000 title 1
- 229940044601 receptor agonist Drugs 0.000 title 1
- 208000010228 Erectile Dysfunction Diseases 0.000 abstract 1
- 206010057671 Female sexual dysfunction Diseases 0.000 abstract 1
- 101000978418 Homo sapiens Melanocortin receptor 4 Proteins 0.000 abstract 1
- 208000008589 Obesity Diseases 0.000 abstract 1
- 201000001880 Sexual dysfunction Diseases 0.000 abstract 1
- 230000004913 activation Effects 0.000 abstract 1
- 239000000556 agonist Substances 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 230000006806 disease prevention Effects 0.000 abstract 1
- 208000037765 diseases and disorders Diseases 0.000 abstract 1
- 102000057094 human MC4R Human genes 0.000 abstract 1
- 201000001881 impotence Diseases 0.000 abstract 1
- 235000020824 obesity Nutrition 0.000 abstract 1
- 231100000872 sexual dysfunction Toxicity 0.000 abstract 1
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Certain novel 4-substituted N-acylated piperidine derivatives are agonists of the human melanocortin-4 receptor. They are useful for the treatment, control, or prevention of diseases and disorders responsive to the activation of MC-4R, such as obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JO200281A JO2351B1 (en) | 2002-07-13 | 2002-07-13 | Acylated piperidine derivatives as melanocortin-4 receptor agonists |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JO200281A JO2351B1 (en) | 2002-07-13 | 2002-07-13 | Acylated piperidine derivatives as melanocortin-4 receptor agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JO2351B1 true JO2351B1 (en) | 2006-06-28 |
Family
ID=48052157
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JO200281A JO2351B1 (en) | 2002-07-13 | 2002-07-13 | Acylated piperidine derivatives as melanocortin-4 receptor agonists |
Country Status (1)
| Country | Link |
|---|---|
| JO (1) | JO2351B1 (en) |
-
2002
- 2002-07-13 JO JO200281A patent/JO2351B1/en active
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