IT1283951B1 - Uso della acetil l-carnitina o dei suoi sali farmacologicamente accettabili per il trattamento terapeutico o la profilassi di - Google Patents
Uso della acetil l-carnitina o dei suoi sali farmacologicamente accettabili per il trattamento terapeutico o la profilassi diInfo
- Publication number
- IT1283951B1 IT1283951B1 IT96RM000171A ITRM960171A IT1283951B1 IT 1283951 B1 IT1283951 B1 IT 1283951B1 IT 96RM000171 A IT96RM000171 A IT 96RM000171A IT RM960171 A ITRM960171 A IT RM960171A IT 1283951 B1 IT1283951 B1 IT 1283951B1
- Authority
- IT
- Italy
- Prior art keywords
- carnitine
- prophylaxis
- acetyl
- acceptable salts
- pharmacologically acceptable
- Prior art date
Links
- RDHQFKQIGNGIED-MRVPVSSYSA-N O-acetyl-L-carnitine Chemical compound CC(=O)O[C@H](CC([O-])=O)C[N+](C)(C)C RDHQFKQIGNGIED-MRVPVSSYSA-N 0.000 title 1
- 238000011321 prophylaxis Methods 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
- 238000011282 treatment Methods 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
- A61K31/221—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin with compounds having an amino group, e.g. acetylcholine, acetylcarnitine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Priority Applications (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT96RM000171A IT1283951B1 (it) | 1996-03-15 | 1996-03-15 | Uso della acetil l-carnitina o dei suoi sali farmacologicamente accettabili per il trattamento terapeutico o la profilassi di |
| TW086102934A TW513304B (en) | 1996-03-15 | 1997-03-10 | Use of an alkanoyl L-carnitine or a pharmacologically acceptable salt thereof for the therapeutic treatment or prophylaxis of glutamate-mediated disturbances or diseases |
| US09/147,034 US6037372A (en) | 1996-03-15 | 1997-03-12 | Use of an alkanoyl-L-carnitine for the treatment of glutamate mediated diseases |
| EP97907268A EP0888113A1 (en) | 1996-03-15 | 1997-03-12 | Use of an alkanoyl-l-carnitine for the treatment of glutamate mediated diseases |
| CA002248879A CA2248879A1 (en) | 1996-03-15 | 1997-03-12 | Use of an alkanoyl-l-carnitine for the treatment of glutamate mediated diseases |
| PCT/IT1997/000056 WO1997034596A1 (en) | 1996-03-15 | 1997-03-12 | Use of an alkanoyl-l-carnitine for the treatment of glutamate mediated diseases |
| KR10-1998-0707309A KR100481188B1 (ko) | 1996-03-15 | 1997-03-12 | 글루타민산염관련질환치료용알카노일-l-카르니틴의용도 |
| JP53332497A JP2001503731A (ja) | 1996-03-15 | 1997-03-12 | グルタメート仲介疾患の処置のためアルカノイル―l―カルニチンの使用 |
| ZA9702219A ZA972219B (en) | 1996-03-15 | 1997-03-14 | Alkanoyl L-carnitine composition against glutamate-mediated conditions. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT96RM000171A IT1283951B1 (it) | 1996-03-15 | 1996-03-15 | Uso della acetil l-carnitina o dei suoi sali farmacologicamente accettabili per il trattamento terapeutico o la profilassi di |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| ITRM960171A0 ITRM960171A0 (it) | 1996-03-15 |
| ITRM960171A1 ITRM960171A1 (it) | 1997-09-15 |
| IT1283951B1 true IT1283951B1 (it) | 1998-05-07 |
Family
ID=11403995
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT96RM000171A IT1283951B1 (it) | 1996-03-15 | 1996-03-15 | Uso della acetil l-carnitina o dei suoi sali farmacologicamente accettabili per il trattamento terapeutico o la profilassi di |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US6037372A (it) |
| EP (1) | EP0888113A1 (it) |
| JP (1) | JP2001503731A (it) |
| KR (1) | KR100481188B1 (it) |
| CA (1) | CA2248879A1 (it) |
| IT (1) | IT1283951B1 (it) |
| TW (1) | TW513304B (it) |
| WO (1) | WO1997034596A1 (it) |
| ZA (1) | ZA972219B (it) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1277897B1 (it) * | 1995-08-03 | 1997-11-12 | Mendes Srl | Uso della l-carnitina,di suoi derivati e di loro sali farmaceuticamen- te accettabili in combinazione con farmaci antiretrovirali per ridurre |
| IT1277898B1 (it) * | 1995-08-03 | 1997-11-12 | Mendes Srl | Uso di amminoacidi basici, di acil derivati di amminoacidi basici e di loro sali farmaceuticamente accettabili per la profilassi di malattie |
| US6348495B1 (en) * | 1996-06-06 | 2002-02-19 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Method for treating celiac disease |
| US6589994B1 (en) | 1996-08-30 | 2003-07-08 | Nps Pharmaceuticals, Inc. | Treating a variety of pathological conditions, including spasticity and convulsions, by effecting a modulation of CNS activity with isovaleramide, isovaleric acid, or a related compound |
| IT1299161B1 (it) * | 1998-04-17 | 2000-02-29 | Sigma Tau Healthscience Spa | Composizione comprendente l-carnitina o un'alcanoil l-carnitina e nadh e/o nadph |
| DE69923322T2 (de) * | 1998-07-30 | 2005-12-22 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Verwendung von propionyl-l-carnitin und acetyl-l-carnitin zur herstellung von arzneimittel mit antikrebs wirkung |
| IT1302289B1 (it) * | 1998-09-30 | 2000-09-05 | Univ Catania | Composizioni farmaceutiche ad attivita' antineoplastica |
| AU1294600A (en) * | 1998-11-11 | 2000-05-29 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Use of propionyl l-carnitine for the preparation of a medicament capable of inducing apoptosis |
| CA2352485A1 (en) * | 1998-11-26 | 2000-06-02 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Use of fumarate salt of l-carnitine or its alkanoyl derivatives in ischaemia |
| IT1306130B1 (it) * | 1999-04-16 | 2001-05-30 | Sigma Tau Healthscience Spa | Composizione comprendente una carnitina e glutatione, atta adaumentare l'assorbimento del glutatione sinergizzandone gli effetti. |
| US20050232911A1 (en) * | 2004-04-19 | 2005-10-20 | Schreiber Brian D | Prevention and treatment of metabolic abnormalities associated with excess intramyocellular lipid |
| JP2006347935A (ja) * | 2005-06-15 | 2006-12-28 | Masanori Ogata | 炎症性サイトカインの産生が関与する疾患の予防及び/又は治療のための医薬 |
| WO2008036682A2 (en) | 2006-09-18 | 2008-03-27 | Raptor Pharmaceutical Inc. | Treatment of liver disorders by administration of receptor-associated protein (rap)-conjugates |
| US20120093809A1 (en) * | 2008-12-01 | 2012-04-19 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Use of alkanoyl l-carnitine in combination with chemotherapeutic agents for the treatment of neoplasms |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
| EP2586438A1 (en) | 2011-10-28 | 2013-05-01 | SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A. | Compound useful for preventing cognitive deficit disorders in a new born from HIV-seropositive pregnant female who is in treatment with azidothymidine |
| CN114522158B (zh) * | 2022-01-21 | 2023-06-27 | 武汉大学 | 用于制备治疗肝癌药物的代谢物及其应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU518617B2 (en) * | 1977-04-29 | 1981-10-08 | Sigma-Tau Industrie Farmaceutiche Riunite S.P.A. | Therapeutic application of acetyl-d, 1-carnitine |
| IT1224842B (it) * | 1988-12-27 | 1990-10-24 | Sigma Tau Ind Farmaceuti | Uso di derivati della l-carnitina nel trattamento terapeutico delle alterazioni degenerative del sistema nervoso |
| IT1244636B (it) * | 1991-01-04 | 1994-08-08 | Sigma Tau Ind Farmaceuti | Uso dell'acetil l-carnitina nel trattamento terapeutico del coma e composizioni farmaceutiche utili in tale trattamento. |
| AU6922994A (en) * | 1993-06-21 | 1995-01-17 | Bernardini, Attilio | Use of acylcarnitin to treat illnesses caused by aids |
-
1996
- 1996-03-15 IT IT96RM000171A patent/IT1283951B1/it active IP Right Grant
-
1997
- 1997-03-10 TW TW086102934A patent/TW513304B/zh not_active IP Right Cessation
- 1997-03-12 KR KR10-1998-0707309A patent/KR100481188B1/ko not_active Expired - Fee Related
- 1997-03-12 EP EP97907268A patent/EP0888113A1/en not_active Ceased
- 1997-03-12 US US09/147,034 patent/US6037372A/en not_active Expired - Fee Related
- 1997-03-12 CA CA002248879A patent/CA2248879A1/en not_active Abandoned
- 1997-03-12 JP JP53332497A patent/JP2001503731A/ja not_active Withdrawn
- 1997-03-12 WO PCT/IT1997/000056 patent/WO1997034596A1/en not_active Ceased
- 1997-03-14 ZA ZA9702219A patent/ZA972219B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| TW513304B (en) | 2002-12-11 |
| ITRM960171A0 (it) | 1996-03-15 |
| KR100481188B1 (ko) | 2005-07-07 |
| CA2248879A1 (en) | 1997-09-25 |
| JP2001503731A (ja) | 2001-03-21 |
| US6037372A (en) | 2000-03-14 |
| WO1997034596A1 (en) | 1997-09-25 |
| ZA972219B (en) | 1997-09-17 |
| EP0888113A1 (en) | 1999-01-07 |
| ITRM960171A1 (it) | 1997-09-15 |
| KR20000064614A (ko) | 2000-11-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 0001 | Granted |