IT1184285B - STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS - Google Patents
STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONSInfo
- Publication number
- IT1184285B IT1184285B IT48298/85A IT4829885A IT1184285B IT 1184285 B IT1184285 B IT 1184285B IT 48298/85 A IT48298/85 A IT 48298/85A IT 4829885 A IT4829885 A IT 4829885A IT 1184285 B IT1184285 B IT 1184285B
- Authority
- IT
- Italy
- Prior art keywords
- medications
- procedure
- preparation
- application
- beta position
- Prior art date
Links
- 229940079593 drug Drugs 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 150000003431 steroids Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8410304A FR2566779B2 (en) | 1984-06-29 | 1984-06-29 | NOVEL 11B SUBSTITUTED STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT8548298A0 IT8548298A0 (en) | 1985-06-28 |
| IT1184285B true IT1184285B (en) | 1987-10-22 |
Family
ID=9305596
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT48298/85A IT1184285B (en) | 1984-06-29 | 1985-06-28 | STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS |
Country Status (7)
| Country | Link |
|---|---|
| JP (1) | JPS6118798A (en) |
| CH (1) | CH666277A5 (en) |
| DE (1) | DE3523297A1 (en) |
| FR (1) | FR2566779B2 (en) |
| GB (1) | GB2160873B (en) |
| IT (1) | IT1184285B (en) |
| NL (1) | NL8501868A (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3619413C2 (en) * | 1986-06-10 | 2000-04-06 | Schering Ag | 9alpha, 10alpha-methylene-estrene, their preparation and pharmaceutical preparations containing them |
| DE3621024C2 (en) * | 1986-06-20 | 1999-10-28 | Schering Ag | 11beta-phenylestradienes, their preparation and pharmaceutical preparations containing them |
| JP2785023B2 (en) * | 1987-12-30 | 1998-08-13 | ルセル―ユクラフ | Novel derivative of 17β-OH-19-norsteroid substituted at 17α position, process for its preparation, its use as drug and pharmaceutical composition containing it |
| JP3202224B2 (en) * | 1989-08-04 | 2001-08-27 | シエーリング アクチエンゲゼルシヤフト | 11β-aryl-gon-4,9-dien-3-ones, process for their preparation and pharmaceutical preparations containing them |
| FR2651233B1 (en) * | 1989-08-23 | 1991-12-13 | Roussel Uclaf | NOVEL OMEGA-PHENYLAMINO ALKANOUIC ACIDS SUBSTITUTED ON THE AROMATIC CORE BY A RADICAL DERIVATIVE OF 19-NORSTEROUIDES, THEIR PREPARATION METHOD, THEIR APPLICATION AS MEDICAMENTS AND THE COMPOSITIONS CONTAINING THEM. |
| FR2651435A1 (en) * | 1989-09-07 | 1991-03-08 | Roussel Uclaf | NEW USE OF ANTI-PROGESTOMIMETIC COMPOUNDS. |
| FR2654337B1 (en) * | 1989-11-15 | 1994-08-05 | Roussel Uclaf | NOVEL BIODEGRADABLE INJECTABLE MICROSPHERES PREPARATION METHOD AND INJECTABLE SUSPENSIONS CONTAINING THEM. |
| US5407928A (en) * | 1990-08-15 | 1995-04-18 | Schering Aktiengesellschaft | 11β-aryl-gona-4,9-dien-3-ones |
| RU2165938C1 (en) * | 2000-06-23 | 2001-04-27 | Насыбуллин Радик Равильевич | METHOD OF SYNTHESIS OF 17β-HYDROXY-11β-[4-(DIMETHYLAMINO)- -PHENYL]-17α-(PROP-1-INYL)-ESTRA-4,9-DIENE-ONE |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2377418A1 (en) * | 1977-01-13 | 1978-08-11 | Roussel Uclaf | NEW 4,9-DIENIC 11B-SUBSTITUTE STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS |
| FR2528434B1 (en) * | 1982-06-11 | 1985-07-19 | Roussel Uclaf | NOVEL 19-NOR STEROIDS SUBSTITUTED IN 11B AND POSSIBLY IN 2, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS A MEDICAMENT |
| ZA8231B (en) * | 1981-01-09 | 1982-11-24 | Roussel Uclaf | New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained |
| DE3321826A1 (en) * | 1983-06-15 | 1984-12-20 | Schering AG, 1000 Berlin und 4709 Bergkamen | 13 alpha -Alkylgonanes, the preparation thereof and pharmaceutical products containing these |
-
1984
- 1984-06-29 FR FR8410304A patent/FR2566779B2/en not_active Expired
-
1985
- 1985-06-28 JP JP60140687A patent/JPS6118798A/en active Pending
- 1985-06-28 NL NL8501868A patent/NL8501868A/en not_active Application Discontinuation
- 1985-06-28 CH CH2772/85A patent/CH666277A5/en not_active IP Right Cessation
- 1985-06-28 DE DE19853523297 patent/DE3523297A1/en not_active Ceased
- 1985-06-28 GB GB08516387A patent/GB2160873B/en not_active Expired
- 1985-06-28 IT IT48298/85A patent/IT1184285B/en active
Also Published As
| Publication number | Publication date |
|---|---|
| FR2566779A2 (en) | 1986-01-03 |
| GB2160873A (en) | 1986-01-02 |
| NL8501868A (en) | 1986-01-16 |
| DE3523297A1 (en) | 1986-01-09 |
| JPS6118798A (en) | 1986-01-27 |
| GB8516387D0 (en) | 1985-07-31 |
| CH666277A5 (en) | 1988-07-15 |
| IT8548298A0 (en) | 1985-06-28 |
| GB2160873B (en) | 1988-03-09 |
| FR2566779B2 (en) | 1987-03-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| TA | Fee payment date (situation as of event date), data collected since 19931001 |
Effective date: 19960517 |