[go: up one dir, main page]

IT1184285B - STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS - Google Patents

STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS

Info

Publication number
IT1184285B
IT1184285B IT48298/85A IT4829885A IT1184285B IT 1184285 B IT1184285 B IT 1184285B IT 48298/85 A IT48298/85 A IT 48298/85A IT 4829885 A IT4829885 A IT 4829885A IT 1184285 B IT1184285 B IT 1184285B
Authority
IT
Italy
Prior art keywords
medications
procedure
preparation
application
beta position
Prior art date
Application number
IT48298/85A
Other languages
Italian (it)
Other versions
IT8548298A0 (en
Inventor
Torelli Vesperto
Jean George Teutsch
Daniel Philibert
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of IT8548298A0 publication Critical patent/IT8548298A0/en
Application granted granted Critical
Publication of IT1184285B publication Critical patent/IT1184285B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J41/00Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C07J41/0083Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IT48298/85A 1984-06-29 1985-06-28 STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS IT1184285B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8410304A FR2566779B2 (en) 1984-06-29 1984-06-29 NOVEL 11B SUBSTITUTED STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS

Publications (2)

Publication Number Publication Date
IT8548298A0 IT8548298A0 (en) 1985-06-28
IT1184285B true IT1184285B (en) 1987-10-22

Family

ID=9305596

Family Applications (1)

Application Number Title Priority Date Filing Date
IT48298/85A IT1184285B (en) 1984-06-29 1985-06-28 STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS

Country Status (7)

Country Link
JP (1) JPS6118798A (en)
CH (1) CH666277A5 (en)
DE (1) DE3523297A1 (en)
FR (1) FR2566779B2 (en)
GB (1) GB2160873B (en)
IT (1) IT1184285B (en)
NL (1) NL8501868A (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3619413C2 (en) * 1986-06-10 2000-04-06 Schering Ag 9alpha, 10alpha-methylene-estrene, their preparation and pharmaceutical preparations containing them
DE3621024C2 (en) * 1986-06-20 1999-10-28 Schering Ag 11beta-phenylestradienes, their preparation and pharmaceutical preparations containing them
JP2785023B2 (en) * 1987-12-30 1998-08-13 ルセル―ユクラフ Novel derivative of 17β-OH-19-norsteroid substituted at 17α position, process for its preparation, its use as drug and pharmaceutical composition containing it
JP3202224B2 (en) * 1989-08-04 2001-08-27 シエーリング アクチエンゲゼルシヤフト 11β-aryl-gon-4,9-dien-3-ones, process for their preparation and pharmaceutical preparations containing them
FR2651233B1 (en) * 1989-08-23 1991-12-13 Roussel Uclaf NOVEL OMEGA-PHENYLAMINO ALKANOUIC ACIDS SUBSTITUTED ON THE AROMATIC CORE BY A RADICAL DERIVATIVE OF 19-NORSTEROUIDES, THEIR PREPARATION METHOD, THEIR APPLICATION AS MEDICAMENTS AND THE COMPOSITIONS CONTAINING THEM.
FR2651435A1 (en) * 1989-09-07 1991-03-08 Roussel Uclaf NEW USE OF ANTI-PROGESTOMIMETIC COMPOUNDS.
FR2654337B1 (en) * 1989-11-15 1994-08-05 Roussel Uclaf NOVEL BIODEGRADABLE INJECTABLE MICROSPHERES PREPARATION METHOD AND INJECTABLE SUSPENSIONS CONTAINING THEM.
US5407928A (en) * 1990-08-15 1995-04-18 Schering Aktiengesellschaft 11β-aryl-gona-4,9-dien-3-ones
RU2165938C1 (en) * 2000-06-23 2001-04-27 Насыбуллин Радик Равильевич METHOD OF SYNTHESIS OF 17β-HYDROXY-11β-[4-(DIMETHYLAMINO)- -PHENYL]-17α-(PROP-1-INYL)-ESTRA-4,9-DIENE-ONE

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2377418A1 (en) * 1977-01-13 1978-08-11 Roussel Uclaf NEW 4,9-DIENIC 11B-SUBSTITUTE STEROID DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICINAL PRODUCTS
FR2528434B1 (en) * 1982-06-11 1985-07-19 Roussel Uclaf NOVEL 19-NOR STEROIDS SUBSTITUTED IN 11B AND POSSIBLY IN 2, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS A MEDICAMENT
ZA8231B (en) * 1981-01-09 1982-11-24 Roussel Uclaf New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained
DE3321826A1 (en) * 1983-06-15 1984-12-20 Schering AG, 1000 Berlin und 4709 Bergkamen 13 alpha -Alkylgonanes, the preparation thereof and pharmaceutical products containing these

Also Published As

Publication number Publication date
FR2566779A2 (en) 1986-01-03
GB2160873A (en) 1986-01-02
NL8501868A (en) 1986-01-16
DE3523297A1 (en) 1986-01-09
JPS6118798A (en) 1986-01-27
GB8516387D0 (en) 1985-07-31
CH666277A5 (en) 1988-07-15
IT8548298A0 (en) 1985-06-28
GB2160873B (en) 1988-03-09
FR2566779B2 (en) 1987-03-06

Similar Documents

Publication Publication Date Title
IT1200092B (en) AMINOPROPOSED DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1219811B (en) PEPTIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT8348580A0 (en) PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICINES
IT1153437B (en) 5-AMINOMETHY-OXYZOLIDINE DERIVATIVES, PROCEDURE FOR THEIR PREPARATION, AND THEIR APPLICATION IN THERAPY
IT1213246B (en) 6-VINYL-FURO- (3,4-C) -PYRIDINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM.
IT1219542B (en) PEPTICIDAL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1169765B (en) DESOXYURIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT8621125A0 (en) POLY-4-AMINOPYRROL-2-CARBOXAMIDO DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION.
IT1184285B (en) STEROID DERIVATIVES REPLACED IN 11-BETA POSITION, PROCEDURE FOR THEIR PREPARATION AND APPLICATION AS MEDICATIONS
IT1199143B (en) 1,4-DIHYDROPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1197655B (en) 2 (HI) -PYRIDINONE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT8547862A0 (en) PYRIDINE DERIVATIVES AND PROCEDURES FOR THEIR PREPARATION
IT1185828B (en) CALCONE DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION
IT1178353B (en) 1,4-DIHYDROPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1199212B (en) 1,2-DITIOLAN DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1170578B (en) CHINAZOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1197634B (en) PLEUROMUTILINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1200079B (en) NAPHTHOXYZINE DERIVATIVES, THEIR PREPARATION, THEIR APPLICATION AS MEDICATIONS AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM
IT1197546B (en) INDOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS
IT1168389B (en) ALCANDIOL DERIVATIVES WITH HYPOLIPIDEMIZING ACTIVITY, METHODS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM
IT1197588B (en) 1,4 DIHYDROPYRIDINE DERIVATIVES, THEIR PREPARATION AND MEDICATIONS CONTAINING THESE DERIVATIVES
IT1181803B (en) ACYLAMINOPHENOL DERIVATIVES, THEIR PREPARATION AND THEIR USE AS A MEDICATION
IT1188188B (en) 6-AMINOMETHY-FURO- (3,4-C) -PYRIDINE DERIVATIVES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME
IT8823183A0 (en) DIOXAZOCIN DERIVATIVES, THEIR PREPARATION AND COMPOSITIONS THAT CONTAIN THEM
IT1200155B (en) 1,4-DIHYDROPYRIDINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICATIONS

Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19960517