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IS5528A - Ný makrólíð - Google Patents

Ný makrólíð

Info

Publication number
IS5528A
IS5528A IS5528A IS5528A IS5528A IS 5528 A IS5528 A IS 5528A IS 5528 A IS5528 A IS 5528A IS 5528 A IS5528 A IS 5528A IS 5528 A IS5528 A IS 5528A
Authority
IS
Iceland
Prior art keywords
new macrolide
macrolide
new
Prior art date
Application number
IS5528A
Other languages
English (en)
Inventor
Philip Dirlam John
Alastair Irvine Mcarthur Hamish
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of IS5528A publication Critical patent/IS5528A/is

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
IS5528A 1998-01-02 2000-06-09 Ný makrólíð IS5528A (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US7034398P 1998-01-02 1998-01-02
PCT/IB1998/002099 WO1999035156A1 (en) 1998-01-02 1998-12-21 Novel macrolides

Publications (1)

Publication Number Publication Date
IS5528A true IS5528A (is) 2000-06-09

Family

ID=22094723

Family Applications (1)

Application Number Title Priority Date Filing Date
IS5528A IS5528A (is) 1998-01-02 2000-06-09 Ný makrólíð

Country Status (34)

Country Link
US (2) US6472371B1 (is)
EP (1) EP1044207A1 (is)
JP (1) JP2002500230A (is)
KR (1) KR100352809B1 (is)
CN (1) CN1284081A (is)
AP (1) AP9801420A0 (is)
AR (4) AR014948A1 (is)
AU (1) AU756409B2 (is)
BG (1) BG104644A (is)
BR (1) BR9814601A (is)
CA (1) CA2316919C (is)
CO (1) CO4970821A1 (is)
CZ (1) CZ20002458A3 (is)
DZ (1) DZ2698A1 (is)
EA (1) EA200000594A1 (is)
GT (1) GT199800206A (is)
HR (1) HRP20000442A2 (is)
HU (1) HUP0100420A3 (is)
IL (1) IL137024A0 (is)
IS (1) IS5528A (is)
MA (1) MA24729A1 (is)
NO (1) NO20003347L (is)
NZ (1) NZ504986A (is)
OA (1) OA11438A (is)
PA (1) PA8465301A1 (is)
PE (1) PE20000049A1 (is)
PL (1) PL341642A1 (is)
SK (1) SK9782000A3 (is)
TN (1) TNSN98238A1 (is)
TW (1) TW520374B (is)
UY (2) UY25330A1 (is)
WO (1) WO1999035156A1 (is)
YU (1) YU41500A (is)
ZA (1) ZA9811939B (is)

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AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
AP9801420A0 (en) 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
EP1437360A3 (en) * 1998-08-19 2005-04-06 Pfizer Products Inc. C11 Carbamates of macrolide antibacterials
US6043227A (en) * 1998-08-19 2000-03-28 Pfizer Inc. C11 carbamates of macrolide antibacterials
EP1754700A3 (en) 1999-01-27 2007-05-09 Kosan Biosciences, Inc. Synthesis of oligoketides
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
US6451768B1 (en) 1999-04-16 2002-09-17 Kosan Biosciences, Inc. Macrolide antiinfective agents
CN1373767A (zh) 1999-04-16 2002-10-09 奥索-麦克尼尔药品公司 酮式大环内酯抗菌剂
HK1045523A1 (zh) 1999-05-24 2002-11-29 辉瑞产品公司 13-甲基红霉素衍生物
JPWO2003072589A1 (ja) * 2002-02-26 2005-06-16 明治製菓株式会社 新規１５員環アザライド及び新規１６員環ジアザライド誘導体とその製造法
US7312248B2 (en) 2004-09-23 2007-12-25 Schering-Plough Animal Health Corporation Control of parasites in animals by the use of novel trifluoromethanesulfonanilide oxime ether derivatives
MX2007006072A (es) * 2004-11-19 2007-07-11 Schering Plough Ltd Control de parasitos en animales mediante el uso de derivados del parasiticida 2-fenil-3-(1h-pirrol-2-il)acrilonitrilo.
DK1836211T3 (da) 2004-12-21 2010-05-17 Pfizer Prod Inc Makrolider
MX2007015729A (es) * 2005-06-09 2008-02-21 Schering Plough Ltd Control de parasitos en animales con derivados de n-[(feniloxi)fenil]-1,1,1-trifluorometansulfonamida y de n[(fenilsulfanil)fenil]-1,1,1-trifluorometansulfonamida.
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
EP2102154A1 (en) * 2006-12-13 2009-09-23 Schering-Plough Ltd. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
WO2008076259A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of florfenicol and its analogs
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
LT2957284T (lt) 2007-06-27 2018-04-10 E. I. Du Pont De Nemours And Company Kovos su gyvūnų kenkėjais būdas
WO2009064953A1 (en) * 2007-11-15 2009-05-22 Enanta Pharmaceuticals, Inc. Use of bridged macrolides or tylosin derivatives in treating inflammatory bowel diseases
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
CN102131772B (zh) * 2008-07-30 2015-03-11 英特威国际有限公司 用作氟苯尼考的中间体的*唑啉-保护的氨基二醇化合物的制备方法
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
BR112012002519A2 (pt) 2009-08-05 2019-09-24 Du Pont "pesticidas mesoiônicos"
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
WO2011017347A2 (en) 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
EP2576523B1 (en) 2010-05-27 2016-01-13 E. I. du Pont de Nemours and Company Crystalline form of 4-[5 - [3 -chloro-5 -(trifluoromethyl)phenyl] -4,5 -dihydro-5 -(trifluoromethyl)-3 - isoxazolyl]-n-[2-oxo-2-[(2,2,2-trifluoroethyl)amino]ethyl]-1- naphthalenecarboxamide
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
CA2826174A1 (en) * 2011-01-31 2012-08-09 Meiji Seika Pharma Co., Ltd. Novel macrolide derivative
EP2721006A1 (en) 2011-06-20 2014-04-23 E. I. Du Pont de Nemours and Company Heterocyclic compounds for treating helminth infections
CN102260306B (zh) * 2011-07-22 2012-07-18 山东鲁抗舍里乐药业有限公司 一种制备泰拉霉素的方法
KR20140094026A (ko) 2011-11-28 2014-07-29 이 아이 듀폰 디 네모아 앤드 캄파니 N-(4-퀴놀리닐메틸) 설폰아미드 유도체 및 구충제로서의 이의 용도
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
WO2014099837A1 (en) 2012-12-18 2014-06-26 E. I. Du Pont De Nemours And Company Sulfonamide anthelmintics
CN105669798B (zh) * 2013-08-23 2019-07-26 普莱柯生物工程股份有限公司 一种大环内酯类化合物
CN103965273B (zh) * 2013-08-23 2016-05-25 普莱柯生物工程股份有限公司 一种大环内酯类化合物

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US6043227A (en) 1998-08-19 2000-03-28 Pfizer Inc. C11 carbamates of macrolide antibacterials
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HK1045523A1 (zh) 1999-05-24 2002-11-29 辉瑞产品公司 13-甲基红霉素衍生物
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JP4311203B2 (ja) 2001-08-08 2009-08-12 大正製薬株式会社 １１ａ−アザライド化合物及びその製造方法

Also Published As

Publication number Publication date
UY25574A1 (es) 1999-09-27
CO4970821A1 (es) 2000-11-07
US6472371B1 (en) 2002-10-29
PE20000049A1 (es) 2000-02-07
AR020551A2 (es) 2002-05-15
AR020851A2 (es) 2002-05-29
AR014948A1 (es) 2001-04-11
BG104644A (en) 2001-01-31
NZ504986A (en) 2003-03-28
WO1999035156B1 (en) 1999-10-21
BR9814601A (pt) 2000-10-17
ZA9811939B (en) 2000-06-30
NO20003347L (no) 2000-08-28
HUP0100420A2 (hu) 2001-07-30
SK9782000A3 (en) 2001-12-03
US20040092459A1 (en) 2004-05-13
CZ20002458A3 (cs) 2001-10-17
WO1999035156A1 (en) 1999-07-15
EP1044207A1 (en) 2000-10-18
CA2316919C (en) 2004-10-26
DZ2698A1 (fr) 2003-03-29
YU41500A (sh) 2003-02-28
KR100352809B1 (ko) 2002-11-01
TNSN98238A1 (fr) 2005-03-15
NO20003347D0 (no) 2000-06-27
PA8465301A1 (es) 2000-09-29
UY25330A1 (es) 2000-12-29
AR019787A2 (es) 2002-03-13
CA2316919A1 (en) 1999-07-15
AU756409B2 (en) 2003-01-09
HRP20000442A2 (en) 2001-04-30
MA24729A1 (fr) 1999-07-01
AU1444799A (en) 1999-07-26
TW520374B (en) 2003-02-11
OA11438A (en) 2004-04-30
IL137024A0 (en) 2001-06-14
AP9801420A0 (en) 1998-12-31
GT199800206A (es) 2000-06-21
CN1284081A (zh) 2001-02-14
PL341642A1 (en) 2001-04-23
HUP0100420A3 (en) 2003-07-28
JP2002500230A (ja) 2002-01-08
KR20010024818A (ko) 2001-03-26
EA200000594A1 (ru) 2001-04-23
US7015203B2 (en) 2006-03-21

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